Synthesis and antinociceptive activities of some pyrazoline derivatives

European Journal of Medicinal Chemistry

Volumn 44, Issue 6, 2009, Pages 2606-2610

  Kaplancikli, Zafer Asim ^a   Turan Zitouni, Gülhan ^a   Özdemir, Ahmet ^a   Devrim Can, Özgür ^a   Chevallet, Pierre ^b  

^a ANADOLU UNIVERSITY   (Turkey)

^b UNIVERSITÉ DE MONTPELLIER   (France)

Author keywords

Benzimidazole; Benzoxazole; Hot plate; Pyrazoline; Rota Rod; Writhing test

Indexed keywords

1 [(BENZAZOLE 2 YL)THIOACETYLAMINO] 3,5 DIARYL 2 PYRAZOLINE DERIVATIVE; BENZIMIDAZOLE; MORPHINE SULFATE; NALOXONE; PYRAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANTINOCICEPTION; ARTICLE; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; MALE; MOUSE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PROTON NUCLEAR MAGNETIC RESONANCE;

ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; DRUG EVALUATION, PRECLINICAL; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; MICE; MOLECULAR STRUCTURE; NALOXONE; PAIN MEASUREMENT; PYRAZOLES; SPECTROPHOTOMETRY, INFRARED;

EID: 64249127655     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2008.09.002     Document Type: Article

References (33)

1. Vongtau H.O., Abbah J., Mosugu O., Chindo B.A., Ngazal I.E., Salawu A.O., Kwanashie H.O., and Gamaniel K.S. J. Ethnopharmacol. 92 (2004) 317-324
2. Wilkerson W.W., Galbraith W., Gans-Brangs K., Grubb M., Hewes W.E., Jaffee B., Kenney J.P., Kerr J., and Wong N. J. Med. Chem. 37 (1994) 988-998
3. Wilkerson W.W., Copeland R.A., Covington M., and Trzaskos J.M. J. Med. Chem. 38 (1995) 389-391
4. Khanna I.K., Weier R.M., Yu Y., Collins P.W., Miyashiro J.M., Koboldt C.M., Veenhuizen A.W., Currie J.L., Seibert K., and Isakson P.C. J. Med. Chem. 40 (1997) 1619-1633
5. Khanna I.K., Weier R.M., Yu Y., Xu X.D., Koszyk F.J., Collins P.W., Koboldt C.M., Veenhuizen A.W., Perkins W.E., Casler J.J., Masferrer J.L., Zhang Y.Y., Gregory S.A., Seibert K., and Isakson P.C. J. Med. Chem. 40 (1997) 1634-1647
6. Tsuji K., Nakamura K., Konishi N., Tojo T., Ochi T., Senoh H., and Matsuo M. Chem. Pharm. Bull. 45 (1997) 987-995
7. Tsuji K., Konishi N., Spears G.W., Ogino T., Nakamura K., Tojo T., Ochi T., Shimojo F., Senoh H., and Matsuo M. Chem. Pharm. Bull. 45 (1997) 1475-1481
8. Bansal E., Srivastava V.K., and Kumar A. Eur. J. Med. Chem. 36 (2001) 81-92
9. Mana F., Chimenti F., Bolasco A., Cenicola M.L., Parrillo M.D.C., Rossi F., and Marmo E. Eur. J. Med. Chem. 27 (1992) 633-639
10. Milano J., Oliveira S.M., Rossato M.F., Sauzem P.D., Machado P., Beck P., Zanatta N., Martins M.A.P., Mello C.F., Rubin M.A., Ferreira J., and Bonacorso H.G. Eur. J. Pharmacol. 581 (2008) 86-96
11. Tabarelli Z., Rubin M.A., Berlese D.B., Sauzem P.D., Missio T.P., Teixeira M.V., Sinhorin A.P., Martins M.A.P., Zanatta N., Bonacorso H.G., and Mello C.F. Braz. J. Med. Biol. Res. 37 (2004) 1531-1540
12. Godoy M.C., Fighera M.R., Souza F.R., Flores A.E., Rubin M.A., Oliveira M.R., Zanatta N., Martins M.A., Bonacorso H.G., and Mello C.F. Eur. J. Pharmacol. 496 (2004) 93-97
13. Sondhi S.M., Singh N., Kumar A., Lozach O., and Meijer L. Bioorg. Med. Chem. 14 (2006) 3758-3765
14. Köksal M., Gökhan N., Küpeli E., Yesilada E., and Erdogan H. Arch. Pharm. Res. 30 (2007) 419-424
15. Önkol T., Sahin M.F., Yildirim E., Erol K., and Ito S. Arch. Pharm. Res. 27 (2004) 1086-1092
16. Sondhi S.M., Rajvanshi S., Johar M., Bharti N., Azam A., and Kumar Singh A. Eur. J. Med. Chem. 37 (2002) 835-843
17. Kawanaka Y., Kobayashi K., Kusuda S., Tatsumi T., Murota M., Nishiyama T., Hisaichi K., Fujii A., Hirai K., Naka M., Komeno M., Nakai H., and Toda M. Bioorg. Med. Chem. Lett. 12 (2002) 2291-2294
18. Shankaran K., Donnelly K.L., Shah S.K., Humes J.L., Pacholok S.G., Grant S.K., Green B.G., and MacCoss M. Bioorg. Med. Chem. Lett. 7 (1997) 2887-2892
19. Vicini P., Incerti M., Amoretti L., Ballabeni V., Tognolini M., and Barocelli E. Farmaco 57 (2002) 363-367
20. Palin R., Clark J.K., Evans L., Houghton A.K., Jones P.S., Prosser A., Wishart G., and Yoshiizumi K. Bioorg. Med. Chem. 16 (2008) 2829-2851
21. Aydin S., Beis R., and Can O.D. Pharmazie 58 (2003) 405-408
22. Kabli R.A., Khalaf A.A., Zimaity M.T., Khalil A.M., Kaddah A.M., and Al-Rifaie H.A. J. Ind. Chem. Soc. 68 (1991) 47-51
23. Khalaf A.A., Kabli R.A., Zimaity M.T., Khalil A.M., Kaddah A.M., and Al-Rifaie H.A. Ind. J. Chem. Sect. B. 32B (1993) 1125-1129
24. Woolfe G., and Mcdonald A.D. J. Pharmacol. Exp. Ther. 80 (1944) 300-307
25. Gabra B.H., and Sirois P. Peptides 24 (2003) 1131-1139
26. Asongalem E.A., Foyet H.S., Ngogang J., Folefoc G.N., Dimo T., and Kamtchouing P.J. J. Ethnopharmacol. 91 (2004) 301-308
27. Koster R., Anderson M., and DeBeer E.J. Fed. Proc. 18 (1959) 412-418
28. Gülçin I., Küfrevioglu O.I., Oktay M., and Büyükokuroglu M.E. J. Ethnopharmacol. 90 (2004) 205-215
29. Adzu B., Amos S., Muazzam I., Inyang U.S., and Gamaniel K.S. J. Ethnopharmacol. 83 (2002) 139-143
30. Wong C.H., Day P., Yarmush J., Wu W., and Zbuzek U.K. Anesth. Analg. 79 (1994) 303-306
31. Coelho L.P., Reis P.A., De Castro F.L., Gayer C.R., Da Silva Lopes C., Da Costa Silva M.C., De Carvalho Sabino K.C., Todeschini A.R., and Coelho M.G. J. Ethnopharmacol. 98 (2005) 109-116
32. Le Bars D., Gozariu M., and Cadden S.W. Pharmacol. Rev. 53 (2001) 597-652
33. Tortorici V., Vásquez E., and Vanegas H. Brain Res. 725 (1996) 106-110