Homology modelling and binding site mapping of the human histamine H1 receptor

European Journal of Medicinal Chemistry

Volumn 39, Issue 11, 2004, Pages 959-967

  Kiss, Róbert ^a   Kovári, Zoltán ^a,b   Keseru, György M ^a,b  

^a GEDEON RICHTER LTD   (Hungary)

^b BUDAPEST UNIVERSITY OF TECHNOLOGY AND ECONOMICS   (Hungary)

Author keywords

Antagonist; Binding site mapping; Homology model; Human histamine H1 receptor

Indexed keywords

ACRIVASTINE; AMINO ACID; DESLORATADINE; HISTAMINE H1 RECEPTOR; LORATADINE; MEPYRAMINE; RHODOPSIN;

ARTICLE; BINDING AFFINITY; BINDING SITE; CALCULATION; GENETIC ALGORITHM; LIPOPHILICITY; MOLECULAR INTERACTION; MOLECULAR MODEL; PROTEIN BINDING; PROTEIN STRUCTURE; SEQUENCE HOMOLOGY;

ALGORITHMS; AMINO ACID SEQUENCE; ANIMALS; BINDING SITES; CATTLE; COMPUTER SIMULATION; DRUG INTERACTIONS; HISTAMINE AGONISTS; HISTAMINE ANTAGONISTS; HUMANS; LORATADINE; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; PROTEIN CONFORMATION; PYRILAMINE; RECEPTORS, HISTAMINE H1; RHODOPSIN; SEQUENCE HOMOLOGY, AMINO ACID; TRIPROLIDINE;

EID: 6344221642     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejmech.2004.07.009     Document Type: Article

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