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Volumn 449, Issue 3, 2002, Pages 229-237

Biochemical characterization of desloratadine, a potent antagonist of the human histamine H1 receptor

(11) Anthes, John C a Gilchrest, Helen a Richard, Christian a Eckel, Stephen a Hesk, Dave a West Jr , Robert E a Williams, Shirley M a Greenfeder, Scott a Billah, Motasim a Kreutner, William a Egan, Robert W a

a MERCK RESEARCH LABORATORIES (United States)

Author keywords

Desloratadine; Human

Indexed keywords

ASTEMIZOLE; AZELASTINE; CALCIUM ION; CAREBASTINE; CETIRIZINE; CHLORPHENIRAMINE; DESLORATADINE; DIPHENHYDRAMINE; EBASTINE; EPINASTINE; FEXOFENADINE; HISTAMINE H1 RECEPTOR; HISTAMINE H1 RECEPTOR ANTAGONIST; HYDROXYZINE; KETOTIFEN; LORATADINE; MEPYRAMINE; MIZOLASTINE; NORASTEMIZOLE; TERFENADINE;

ANIMAL CELL; ARTICLE; BINDING COMPETITION; BINDING KINETICS; CALCULATION; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DISSOCIATION; DRUG ACTIVITY; DRUG MECHANISM; DRUG POTENCY; DRUG RECEPTOR BINDING; FEMALE; INCUBATION TIME; NONHUMAN; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL;

EID: 0037047697 PISSN: 00142999 EISSN: None Source Type: Journal
DOI: 10.1016/S0014-2999(02)02049-6 Document Type: Article

Times cited : (116)

References (32)

1
- 0033982162
- 1 receptor antagonists
- (2000) Eur. J. Pharmacol. , vol.387
- Bakker, R.A.¹ Wieland, K.² Timmerman, H.³ Leurs, R.⁴

2
- 0034752736
- q/11-subunits in constitutive and agonist mediated signalling
- (2001) Mol. Pharmacol. , vol.60 , pp. 1133-1142
- Bakker, R.A.¹ Schoonus, S.B.J.² Smit, M.J.³ Timmerman, H.⁴ Leurs, R.⁵

3
- 0030979265
- 1 receptor antagonist
- (1997) Eur. J. Pharmacol. , vol.325 , pp. 253-261
- Cascieri, M.A.¹ Ber, E.² Fong, T.M.³ Hale, J.J.⁴ Tang, F.⁵ Shiao, L.L.⁶ Mills, S.G.⁷ MacCoss, M.⁸ Sadowski, S.⁹ Tota, M.R.¹⁰ Strader, C.D.¹¹

4
- 0015861774
- 50) of an enzymatic reaction
- (1973) Biochem. Pharmacol. , vol.22 , pp. 3094-3108
- Cheng, Y.C.¹ Prusoff, W.H.²

5
- 0032732550
- The assessment of antagonist potency under conditions of transient response kinetics
- (1999) Eur. J. Pharmacol. , vol.382 , pp. 217-227
- Christopoulos, A.¹ Parson, A.M.² Lew, M.J.³ El-Fakahany, E.E.⁴

6
- 0001695201
- Torsades de pointes after astemizole overdose
- (1986) BMJ , vol.192 , pp. 660-664
- Craft, T.M.¹

7
- 0027772522
- 1 receptor
- (1993) Biochem. Biophys. Res. Commun. , vol.197 , pp. 1601-1608
- DeBacker, M.D.¹ Gommeren, W.² Moereels, H.³ Nobels, G.⁴ Van Gompel, P.⁵ Leysen, J.E.⁶ Luyten, W.⁷

8
- 0025946154
- 2 receptor
- (1991) Biochem. Biophys. Res. Commun. , vol.178 , pp. 1386-1392
- Gantz, I.¹ Munzert, G.² Tashiro, T.³ Schaffer, M.⁴ Wang, L.⁵ Delvalle, J.⁶ Yamada, T.⁷

9
- 0033494989
- Advancement of the third generation of antihistamines
- (1999) Pediatr. Allergy Immunol. , vol.13 , pp. 163-168
- Handley, D.A.¹

10
- 0010013730
- Descarboxyloratadine, a metabolite of loratadine, is a superior antihistamine
- abstract
- (1997) Ann. Allergy, Asthma, & Immun. , vol.78 , pp. 144
- Handley, D.A.¹ McCullough, J.R.² Fang, F.Q.³ Wright, S.E.⁴ Smith, E.R.⁵

11
- 0001339720
- 1 receptor antagonist
- (2000) J. Allergy Clin. Immunol. , vol.104 , Issue.1 PART 2
- Hey, J.¹ Anthes, J.² Barnett, A.³ Tozzi, S.⁴ Kreutner, W.⁵

12
- 0030772640
- International union of pharmacology: XIII. Classification of histamine receptors
- (1997) Pharmacol. Rev. , vol.49 , pp. 253-278
- Hill, S.J.¹ Ganellin, C.R.² Timmerman, H.³ Schwartz, J.C.⁴ Shankley, N.P.⁵ Young, J.M.⁶ Schunack, W.⁷ Levi, R.⁸ Hass, H.L.⁹

13
- 0023511488
- Histamine-induced calcium release and phorbol antagonism in cultured airway smooth muscle cells
- (1987) Am. J. Physiol. , vol.253
- Kotlikoff, M.I.¹ Murray, R.K.² Reynolds, E.E.³

14
- 0033999939
- 1 receptor antagonist: 1st communication: Receptor selectivity, antihistaminic activity, and antiallergenic effects
- (2000) Arzneim.-Forsch. , vol.50 , pp. 345-352
- Kreutner, W.¹ Hey, J.A.² Anthes, J.³ Barnett, A.⁴ Young, S.⁵ Tozzi, S.⁶

15
- 0033051582
- 3 receptor
- (1999) Mol. Pharmacol. , vol.55 , pp. 1101-1107
- Lovenberg, T.W.¹ Roland, B.L.² Wilson, S.J.³ Jiang, X.⁴ Pyati, J.⁵ Huvar, A.⁶ Jackson, M.R.⁷ Erlander, M.G.⁸

16
- 0031861820
- Pharmacological treatment options for allergic rhinitis and asthma
- (1998) Clin. Exp. Allergy , vol.28 , pp. 27-36
- Meltzer, E.O.¹

17
- 0032723296
- 1-histamine receptor antagonists in fluorescent imaging plate reader based calcium assays
- (1999) J. Biomol. Screen. , vol.4 , pp. 249-258
- Miller, T.R.¹ Witte, D.G.² Ireland, L.M.³ Kang, C.H.⁴ Roh, J.M.⁵ Masters, J.N.⁶ Esbenshade, T.A.⁷ Hancock, J.⁸

18
- 0028105946
- 1 histamine receptor cDNA in Chinese hamster ovary cells
- (1994) Eur. J. Biochem. , vol.224 , pp. 489-495
- Moguilevsky, N.¹ Varsolona, F.² Noyer, M.³ Gillard, M.⁴ Guillaume, J.P.⁵ Garcia, L.⁶ Szpirer, C.⁷ Szpirer, G.⁸ Bollen, A.⁹

19
- 0025222965
- Torsades de pointes occurring in association with terfenadine use
- (1990) JAMA , vol.264 , pp. 2788-2790
- Monahan, B.P.¹ Ferguson, C.L.² Killeavy, E.S.³ Lloyd, B.K.⁴ Troy, J.⁵ Cantilena L.R., Jr.⁶

20
- 0035120049
- Cloning and characterization of a novel human histamine receptor
- (2001) J. Pharmacol. Exp. Ther. , vol.296 , pp. 1058-1066
- Morse, K.L.¹ Behan, J.² Laz, T.³ West R.E., Jr.⁴ Greenfeder, S.⁵ Anthes, J.C.⁶ Umland, S.⁷ Wan, Y.⁸ Hipkin, R.W.⁹ Gonsiorek, W.¹⁰ Shin, N.¹¹ Gustafson, E.L.¹² Qiao, X.¹³ Wang, S.¹⁴ Hedrick, J.A.¹⁵ Greene, J.¹⁶ Bayne, M.¹⁷ Monsma F.J., Jr.¹⁸

21
- 0025865173
- Receptor activated calcium influx in human airway smooth muscle cells
- (1991) J. Physiol. , vol.435 , pp. 123-144
- Murray, R.K.¹ Kotlikoff, M.I.²

22
- 0034711258
- Molecular cloning and characterization of novel type of histamine receptor preferentially expressed in leukocytes
- (2000) J. Biol. Chem. , vol.275 , pp. 36781-36786
- Oda, T.¹ Morkiawa, N.² Saito, Y.³ Masuho, Y.⁴ Matsumoto, S.⁵

23
- 0031987855
- 1 receptors
- (1998) Int. J. Mol. Med. , vol.1 , pp. 355-360
- Ohuchi, Y.¹ Yanai, K.² Sakura, E.³ Fukui, H.⁴ Yanagisawa, T.⁵ Watanabe, T.⁶

24
- 0029078461
- 1 antagonism
- (1995) J. Pharmacol. Exp. Ther. , vol.273 , pp. 753-761
- Panek, R.L.¹ Lu, G.H.² Overhiser, R.W.³ Major, T.C.⁴ Hodges, J.C.⁵ Taylor, D.G.⁶

25
- 0001075185
- Efficacy and safety of desloratadine in seasonal allergic rhinitis
- (2000) J. Allergy Clin. Immunol. , vol.104 , Issue.1 PART 2
- Salmun, L.M.¹ Lorber, R.² Danzig, M.³ Staudinger, H.⁴

26
- 0027459122
- Prolonged QT interval and torsade de pointes following astemizole overdose
- (1993) J. Toxicol., Clin. Toxicol. , vol.31 , pp. 121-125
- Saviuc, P.¹ Danel, V.² Dixmerias, F.³

27
- 0032919046
- Second generation anti-histamines: A comparative review
- (1999) Drugs , vol.57 , pp. 31-38
- Slater, J.W.¹ Zehnich, A.D.² Haxby, D.G.³

28
- 0027405484
- 1 receptor antagonists for CNS and peripheral receptors?
- (1993) Eur. J. Pharmacol. , vol.232 , pp. 199-205
- Ter Laak, A.M.¹ Donne-Op den Kelder, G.M.² Bast, A.³ Timmerman, H.⁴

29
- 0023912788
- 3H]-mepyramine
- (1988) Br. J. Pharmacol. , vol.94 , pp. 811-822
- Treherne, J.M.¹ Young, J.M.²

30
- 0033569709
- 1 receptor
- (1999) J. Biol. Chem. , vol.274 , pp. 29994-30000
- Wieland, K.¹ Ter Laak, A.² Smit, H.J.³ Kuhne, R.⁴ Timmerman, H.⁵ Leurs, R.⁶

31
- 0027474601
- Mechanism of the cardiotoxic actions of terfenadine
- (1993) JAMA , vol.269 , pp. 1532-1535
- Woosley, R.L.¹ Chen, Y.² Freiman, J.P.³

32
- 0026327418
- 1 receptor
- (1991) Proc. Natl. Acad. Sci. , vol.88 , pp. 11515-11520
- Yamashita, M.¹ Fukui, H.² Sugama, K.³ Horio, I.⁴ Ito, S.⁵ Mizuguchi, H.⁶ Wada, H.⁷

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