[18F]FEAC and [18F]FEDAC: Two novel positron emission tomography ligands for peripheral-type benzodiazepine receptor in the brain

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 6, 2009, Pages 1707-1710

  Yanamoto, Kazuhiko ^a   Kumata, Katsushi ^a   Yamasaki, Tomoteru ^a   Odawara, Chika ^a   Kawamura, Kazunori ^a   Yui, Joji ^a   Hatori, Akiko ^a   Suzuki, Kazutoshi ^a   Zhang, Ming Rong ^a  

^a NATIONAL INSTITUTE OF RADIOLOGICAL SCIENCES   (Japan)

Author keywords

18F FEAC; 18F FEDAC; Fluorine 18; Peripheral type benzodiazepine receptor; Positron emission tomography

Indexed keywords

BENZODIAZEPINE RECEPTOR; EMAPUNIL; FAC F 18; FEAC F 18; FEDAC F 18; FLUORODEOXYGLUCOSE F 18; KAINIC ACID; N SEC BUTYL 1 (2 CHLOROPHENYL) N METHYL 3 ISOQUINOLINECARBOXAMIDE; TRACER; UNCLASSIFIED DRUG; 4 AMINOBUTYRIC ACID A RECEPTOR; FLUORINE; LIGAND; RADIOPHARMACEUTICAL AGENT;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; CORPUS STRIATUM; DRUG STRUCTURE; DRUG SYNTHESIS; ENCEPHALITIS; IN VITRO STUDY; LIPOPHILICITY; MALE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; RAT; ANIMAL; BRAIN; CHEMICAL MODEL; CHEMISTRY; DRUG DESIGN; DRUG EFFECT; HUMAN; INFLAMMATION; INSTRUMENTATION; METABOLISM; METHODOLOGY; SPRAGUE DAWLEY RAT; SYNTHESIS;

ANIMALIA; RATTUS;

ANIMALS; BRAIN; CHEMISTRY, PHARMACEUTICAL; DRUG DESIGN; FLUORINE RADIOISOTOPES; HUMANS; INFLAMMATION; LIGANDS; MALE; MODELS, CHEMICAL; POSITRON-EMISSION TOMOGRAPHY; RADIOPHARMACEUTICALS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GABA-A;

EID: 61349126690     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.01.093     Document Type: Article

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