How to increase the reactivity of [18F]fluoroethyl bromide: [18F]fluoroethylation of amine, phenol and amide functional groups with [18F]FEtBr, [18F]FEtBr/NaI and [18F]FEtOTf

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 46, Issue 6, 2003, Pages 587-598

  Zhang, Ming Rong ^a,b   Furutsuka, Kenji ^a,b   Yoshida, Yuichiro ^a,b   Suzuki, Kazutoshi ^a  

^a NATIONAL INSTITUTE OF RADIOLOGICAL SCIENCES   (Japan)

^b Japan   (Japan)

Author keywords

PET tracer; 18F FEtBr; 18F FEtBr NaI; 18F FEtOTf; 18F fluoroethylation

Indexed keywords

AMIDES; EFFICIENCY; IODINE COMPOUNDS; PHENOLS; SUBSTRATES;

AMIDE FUNCTIONAL GROUP; AMINE FUNCTIONAL GROUPS; AMINE MOIETIES; PET TRACER; PHENOL FUNCTIONAL GROUPS; SYNTHETIC PRECURSORS; [18F]FETBR; [18F]FETBR/NAI; [18F]FETOTF; [18F]FLUOROETHYLATION;

SODIUM IODIDE;

AMIDE; AMINE; FLUORINE 18; FLUOROETHYL BROMIDE F 18; FLUOROETHYL SODIUM IODIDE F 18; FLUOROETHYL TRIFLATE F 18; PHENOL; SODIUM IODIDE; TRACER; UNCLASSIFIED DRUG;

ARTICLE; DRUG ACTIVITY; DRUG STRUCTURE; ISOTOPE LABELING; POSITRON EMISSION TOMOGRAPHY;

EID: 0038541684     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/jlcr.703     Document Type: Article

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