Hansch analysis of veratric acid derivatives as antimicrobial agents

European Journal of Medicinal Chemistry

Volumn 44, Issue 2, 2009, Pages 689-700

  Narasimhan, Balasubramanian ^a   Ohlan, Sucheta ^a   Ohlan, Ruchita ^a   Judge, Vikramjeet ^a   Narang, Rakesh ^a  

^a GURU JAMBHESHWAR UNIVERSITY OF SCIENCE AND TECHNOLOGY   (India)

Author keywords

Antibacterial activity; Antifungal activity; QSAR; Veratric acid

Indexed keywords

3 NITROVERATRANILIDE; 4 BROMOVERATRANILIDE; 8 QUINOLINYL VERATRATE; ANTIINFECTIVE AGENT; CIPROFLOXACIN; FLUCONAZOLE; UNCLASSIFIED DRUG; VERATRIC ACID DERIVATIVE;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; ASPERGILLUS NIGER; BACILLUS SUBTILIS; CANDIDA ALBICANS; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STAPHYLOCOCCUS AUREUS; TABEBUIA;

ANTI-INFECTIVE AGENTS; FUNGI; GRAM-NEGATIVE BACTERIA; GRAM-POSITIVE BACTERIA; MICROBIAL SENSITIVITY TESTS; STRUCTURE-ACTIVITY RELATIONSHIP; VANILLIC ACID;

EID: 60149102773     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2008.05.008     Document Type: Article

References (44)

1. Zanatta N., Alves S.H., Coelho H.S., Borchhardt D.M., Santurio J.M., Bonacorso H.G., and Martin M.A.P. Bioorg. Med. Chem. Lett. 15 (2007) 1947-1956
2. Nezhad A.K., Rad M.N.S., Mohabatkar H., Asrari Z., and Hemmateenejad B. Bioorg. Med. Chem. Lett. 13 (2005) 1931-1938
3. Antolini M., Boaaoli A., Ghiron C., Kennedy G., Rossi T., and Ursini A. Bioorg. Med. Chem. Lett. 9 (1999) 1023-1028
4. Awale S., Kawakami T., Tezuka K., Ueda J., Tanaka K., and Kodata S. Chem. Pharm. Bull. 53 6 (2005) 710-713
5. Malarczyk E., and Pazdzioch-czochra M. Cell Biol. Int. 24 8 (2000) 515-527
6. Zemek J., Valen M., Podova M., Kasikova B., and Joniak D. Folia Microbiol. (Praha) 32 5 (1987) 421-425
7. Szwajgier D., Pielecki J., and Targonski Z. Acta Sci. Pol., Technol. Aliment. 4 2 (2005) 129-149
8. Zheng J., Zhao D.S., Wu B., and Wu L. Zhongguo Zhong Yao Za Zhi 27 10 (2002) 749-751
9. Sommers D.K., Snyman J.R., Van W.M., and Eloff J.N. Eur. J. Clin. Pharmacol. 53 3-4 (1997) 247-249
10. Hansch C., and Fujita T. J. Am. Chem. Soc. 86 (1964) 1616-1626
11. Narasimhan B., Kothawade U.R., Pharande D.S., Mourya V.K., and Dhake A.S. Indian J. Chem. 42B (2003) 2828-2834
12. Narasimhan B., Belsare D.P., Pharande D.S., Mourya V.K., and Dhake A.S. Eur. J. Med. Chem. 39 10 (2004) 827-834
13. Narasimhan B., Mourya V.K., and Dhake A.S. Bioorg. Med. Chem. Lett. 16 (2006) 3023-3029
14. Narasimhan B., Mourya V.K., and Dhake A.S. Khim. Farm. Zh. 41 3 (2007) 16-21
15. Narasimhan B., Narang R., Judge V., Ohlan S., and Ohlan R. ARKIVOC xv (2007) 112-126
16. Narasimhan B., Judge V., Narang R., Ohlan S., and Ohlan R. Bioorg. Med. Chem. Lett. 17 (2007) 5836-5845
17. Gangwal N.A., Narasimhan B., Mourya V.K., Dhake A.S., and Indian J. Heteroat. Chem. 12 (2003) 201-204
18. Narasimhan B., Ansari A.H., Singh N., Mourya V.K., and Dhake A.S. Chem. Pharm. Bull. 54 8 (2006) 1067-1071
19. Narasimhan B., Kumari M., Jain N., Dhake A.S., and Sundaravelan C. Bioorg. Med. Chem. Lett. 16 (2006) 4951-4958
20. Narasimhan B., Kumari M., Dhake A.S., and Sundaravelan C. ARKIVOC xiii (2006) 73-82
21. Kumar A., Narasimhan B., and Kumar D. Bioorg. Med. Chem. 15 (2007) 4113-4124
22. Narasimhan B., Dhake A.S., and Mourya V.K. ARKIVOC I (2007) 189-204
23. Narasimhan B., Ohlan R., Ohlan S., Judge V., Narang R., and Ahuja M. ARKIVOC xiv (2007) 172-184
24. Park J., Lee J., Jung E., Park Y., Kim K., Park B., Jung K., Park E., Kim J., and Park D. Eur. J. Pharmacol. 496 1-3 (2004) 189-195
25. Pharmacopoeia of India vol. II (1996), Ministry of Health Department, Govt. of India, New Delhi A-88
26. Hansch C., Leo A., Unger S.H., Kim K.H., Nikaitani D., and Lien E.J. J. Med. Chem. 16 11 (1973) 1207-1216
27. Kier L.B., and Hall L.H. Molecular Connectivity in Chemistry and Drug Research (1976), Academic Press, New York
28. Randic M. J. Am. Chem. Soc. 97 (1975) 6609-6615
29. Balaban A.T. Chem. Phys. Lett. 89 (1982) 399-404
30. Wiener H. J. Am. Chem. Soc. 69 (1947) 17-20
31. Randic M. Croat. Chem. Acta 66 (1993) 289-312
32. Sharma P., Rane N., and Gurram V.K. Bioorg. Med. Chem. Lett. 14 (2004) 4185-4190
33. Sortino M., Delgado P., Jaurez S., Quiroga J., Abonia R., Insuasey B., Nogueras M., Rodero L., Garibotto F.M., Enriz R.D., and Zacchino S.A. Bioorg. Med. Chem. Lett. 15 (2007) 484-494
34. Gupta S.P., Kumar A.N., Nagazppa A.N., Kumar D., and Kumaran S. Eur. J. Med. Chem. 38 (2003) 867-873
35. Karelson M., Lobanov V.S., and Katritzky A.R. Chem. Rev. 96 3 (1996) 1027-1044
36. Wold S., and Erikkson L. Statistical validation of QSAR results. Chemometrics Methods in Molecular Design (1995), VCH Publishers, New York
37. Golbraikh A., and Tropsha A. J. Mol. Graph. Model. 20 4 (2002) 269-276
38. Bajaj S., Sambi S.S., and Madan A.K. Croat. Chem. Acta 78 2 (2005) 165-174
39. Sharma P., Kumar A., and Sharma M. Eur. J. Med. Chem. 41 (2006) 833-840
40. Hatya S.A., Aki-sener E., Tekiner-Gulbas B., Yildiz I., Temiz-Arpaci O., Yalcin I., and Altanlar N. Eur. J. Med. Chem. 41 (2006) 1398-1404
41. Kumar A., Sharma P., Gurram V.K., and Rane N. Bioorg. Med. Chem. Lett. 16 (2006) 2484-2491
42. TSAR 3D Version 3.3 (2000), Oxford Molecular Limited
43. SPSS for Windows, Version 10.05 (1999), SPSS Inc., Bangalore, India
44. Schaper K.J. Quant. Struct.-Act. Relat. 18 (1999) 354-360