메뉴 건너뛰기




Volumn 399, Issue 1-2, 2009, Pages 83-87

Telmisartan pharmacokinetics in Japanese renal transplant recipients

Author keywords

MRP2; OATP; Pharmacokinetics; Telmisartan; UGT

Indexed keywords

BREAST CANCER RESISTANCE PROTEIN; CANDESARTAN; GLUCURONOSYLTRANSFERASE 1A1; GLUCURONOSYLTRANSFERASE 1A6; GLUCURONOSYLTRANSFERASE 1A7; GLUCURONOSYLTRANSFERASE 1A9; GLUCURONOSYLTRANSFERASE 2B7; MULTIDRUG RESISTANCE PROTEIN 1; MULTIDRUG RESISTANCE PROTEIN 2; PROTEIN ABCC2; PROTEIN SLCO 1B1; PROTEIN SLCO 1B3; PROTEIN SLCO 2B1; TELMISARTAN; UNCLASSIFIED DRUG;

EID: 57049170781     PISSN: 00098981     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.cca.2008.09.020     Document Type: Article
Times cited : (31)

References (35)
  • 1
    • 0347589286 scopus 로고    scopus 로고
    • Therapeutic effects of angiotensin II inhibition or blockade on the progression of chronic renal disease
    • Cantarovich F., and Rangoonwala B. Therapeutic effects of angiotensin II inhibition or blockade on the progression of chronic renal disease. Int J Clin Pract 57 (2003) 801-822
    • (2003) Int J Clin Pract , vol.57 , pp. 801-822
    • Cantarovich, F.1    Rangoonwala, B.2
  • 2
    • 0033748477 scopus 로고    scopus 로고
    • Pharmacokinetics and safety of intravenous and oral telmisartan 20 mg and 120 mg in subjects with hepatic impairment compared with healthy volunteers
    • Stangier J., Su C.A., Schondorfer G., and Roth W. Pharmacokinetics and safety of intravenous and oral telmisartan 20 mg and 120 mg in subjects with hepatic impairment compared with healthy volunteers. J Clin Pharmacol 40 (2000) 1355-1364
    • (2000) J Clin Pharmacol , vol.40 , pp. 1355-1364
    • Stangier, J.1    Su, C.A.2    Schondorfer, G.3    Roth, W.4
  • 5
    • 0037733365 scopus 로고    scopus 로고
    • A novel human organic anion transporting polypeptide localized to the basolateral hepatocyte membrane
    • Konig J., Cui Y., Nies A.T., and Keppler D. A novel human organic anion transporting polypeptide localized to the basolateral hepatocyte membrane. Am J Physiol Gastrointest Liver Physiol 278 (2000) G156-G164
    • (2000) Am J Physiol Gastrointest Liver Physiol , vol.278
    • Konig, J.1    Cui, Y.2    Nies, A.T.3    Keppler, D.4
  • 6
    • 0034725617 scopus 로고    scopus 로고
    • Localization and genomic organization of a new hepatocellular organic anion transporting polypeptide
    • Konig J., Cui Y., Nies A.T., and Keppler D. Localization and genomic organization of a new hepatocellular organic anion transporting polypeptide. J Biol Chem 275 (2000) 23161-23168
    • (2000) J Biol Chem , vol.275 , pp. 23161-23168
    • Konig, J.1    Cui, Y.2    Nies, A.T.3    Keppler, D.4
  • 7
    • 0037907742 scopus 로고    scopus 로고
    • Role of organic anion-transporting polypeptides, OATP-A, OATP-C and OATP-8, in the human placenta-maternal liver tandem excretory pathway for foetal bilirubin
    • Briz O., Serrano M.A., Maclas R.I., Gonzalez-Gallego J., and Marin J.J. Role of organic anion-transporting polypeptides, OATP-A, OATP-C and OATP-8, in the human placenta-maternal liver tandem excretory pathway for foetal bilirubin. Biochem J 371 (2003) 897-905
    • (2003) Biochem J , vol.371 , pp. 897-905
    • Briz, O.1    Serrano, M.A.2    Maclas, R.I.3    Gonzalez-Gallego, J.4    Marin, J.J.5
  • 8
    • 0035125407 scopus 로고    scopus 로고
    • Organic anion-transporting polypeptide B (OATP-B) and its functional comparison with three other OATPs of human liver
    • Kullak-Ublick G.A., Ismair M.G., Stieger B., et al. Organic anion-transporting polypeptide B (OATP-B) and its functional comparison with three other OATPs of human liver. Gastroenterology 120 (2001) 525-533
    • (2001) Gastroenterology , vol.120 , pp. 525-533
    • Kullak-Ublick, G.A.1    Ismair, M.G.2    Stieger, B.3
  • 9
    • 0038637144 scopus 로고    scopus 로고
    • Involvement of human organic anion transporting polypeptide OATP-B (SLC21A9) in pH-dependent transport across intestinal apical membrane
    • Kobayashi D., Nozawa T., Imai K., Nezu J., Tsuji A., and Tamai I. Involvement of human organic anion transporting polypeptide OATP-B (SLC21A9) in pH-dependent transport across intestinal apical membrane. J Pharmacol Exp Ther 306 (2003) 703-708
    • (2003) J Pharmacol Exp Ther , vol.306 , pp. 703-708
    • Kobayashi, D.1    Nozawa, T.2    Imai, K.3    Nezu, J.4    Tsuji, A.5    Tamai, I.6
  • 10
    • 0033032730 scopus 로고    scopus 로고
    • Expression of the MRP2 gene-encoded conjugate export pump in human kidney proximal tubules and in renal cell carcinoma
    • Schaub T.P., Kartenbeck J., Konig J., et al. Expression of the MRP2 gene-encoded conjugate export pump in human kidney proximal tubules and in renal cell carcinoma. J Am Soc Nephrol 10 (1999) 1159-1169
    • (1999) J Am Soc Nephrol , vol.10 , pp. 1159-1169
    • Schaub, T.P.1    Kartenbeck, J.2    Konig, J.3
  • 11
    • 22944446686 scopus 로고    scopus 로고
    • Identification of the hepatic efflux transporters of organic anions using double-transfected Madin-Darby canine kidney II cells expressing human organic anion-transporting polypeptide 1B1 (OATP1B1)/multidrug resistance-associated protein 2, OATP1B1/multidrug resistance 1, and OATP1B1/breast cancer resistance protein
    • Matsushima S., Maeda K., Kondo C., et al. Identification of the hepatic efflux transporters of organic anions using double-transfected Madin-Darby canine kidney II cells expressing human organic anion-transporting polypeptide 1B1 (OATP1B1)/multidrug resistance-associated protein 2, OATP1B1/multidrug resistance 1, and OATP1B1/breast cancer resistance protein. J Pharmacol Exp Ther 314 (2005) 1059-1067
    • (2005) J Pharmacol Exp Ther , vol.314 , pp. 1059-1067
    • Matsushima, S.1    Maeda, K.2    Kondo, C.3
  • 12
    • 33745253947 scopus 로고    scopus 로고
    • Predominant contribution of OATP1B3 to the hepatic uptake of telmisartan, an angiotensin II receptor antagonist, in humans
    • Ishiguro N., Maeda K., Kishimoto W., et al. Predominant contribution of OATP1B3 to the hepatic uptake of telmisartan, an angiotensin II receptor antagonist, in humans. Drug Metab Dispos 34 (2006) 1109-1115
    • (2006) Drug Metab Dispos , vol.34 , pp. 1109-1115
    • Ishiguro, N.1    Maeda, K.2    Kishimoto, W.3
  • 13
    • 41549098278 scopus 로고    scopus 로고
    • Establishment of a set of double transfectants coexpressing organic anion transporting polypeptide 1B3 and hepatic efflux transporters for the characterization of the hepatobiliary transport of telmisartan acylglucuronide
    • Ishiguro N., Maeda K., Saito A., et al. Establishment of a set of double transfectants coexpressing organic anion transporting polypeptide 1B3 and hepatic efflux transporters for the characterization of the hepatobiliary transport of telmisartan acylglucuronide. Drug Metab Dispos 36 (2008) 796-805
    • (2008) Drug Metab Dispos , vol.36 , pp. 796-805
    • Ishiguro, N.1    Maeda, K.2    Saito, A.3
  • 14
    • 0034671387 scopus 로고    scopus 로고
    • Polymorphisms of UDP-glucuronosyltransferase gene and irinotecan toxicity: a pharmacogenetic analysis
    • Ando Y., Saka H., Ando M., et al. Polymorphisms of UDP-glucuronosyltransferase gene and irinotecan toxicity: a pharmacogenetic analysis. Cancer Res 60 (2000) 6921-6926
    • (2000) Cancer Res , vol.60 , pp. 6921-6926
    • Ando, Y.1    Saka, H.2    Ando, M.3
  • 15
    • 21444446551 scopus 로고    scopus 로고
    • Urinary excretion of phenytoin metabolites, 5-(4'-hydroxyphenyl)-5-phenylhydantoin and its O-glucuronide in humans and analysis of genetic polymorphisms of UDP-glucuronosyltransferases
    • Yamanaka H., Nakajima M., Hara Y., et al. Urinary excretion of phenytoin metabolites, 5-(4'-hydroxyphenyl)-5-phenylhydantoin and its O-glucuronide in humans and analysis of genetic polymorphisms of UDP-glucuronosyltransferases. Drug Metab Pharmacokinet 20 (2005) 135-143
    • (2005) Drug Metab Pharmacokinet , vol.20 , pp. 135-143
    • Yamanaka, H.1    Nakajima, M.2    Hara, Y.3
  • 16
    • 33645130789 scopus 로고    scopus 로고
    • Polymorphisms of UDP-glucuronosyltransferase 1A7 are not involved in pancreatic diseases
    • Verlaan M., Drenth J.P., and Truninger K. Polymorphisms of UDP-glucuronosyltransferase 1A7 are not involved in pancreatic diseases. J Med Genet 42 (2005) e62
    • (2005) J Med Genet , vol.42
    • Verlaan, M.1    Drenth, J.P.2    Truninger, K.3
  • 17
    • 10344233143 scopus 로고    scopus 로고
    • Genetic polymorphisms in UDP-glucuronosyltransferases and glutathione S-transferases and colorectal cancer risk
    • van der Logt E.M., Bergevoet S.M., Roelofs H.M., et al. Genetic polymorphisms in UDP-glucuronosyltransferases and glutathione S-transferases and colorectal cancer risk. Carcinogenesis 25 (2004) 2407-2415
    • (2004) Carcinogenesis , vol.25 , pp. 2407-2415
    • van der Logt, E.M.1    Bergevoet, S.M.2    Roelofs, H.M.3
  • 18
    • 33745242349 scopus 로고    scopus 로고
    • The novel UGT1A9 intronic I399 polymorphism appears as a predictor of 7-ethyl-10-hydroxycamptothecin glucuronidation levels in the liver
    • Girard H., Villeneuve L., Court M.H., et al. The novel UGT1A9 intronic I399 polymorphism appears as a predictor of 7-ethyl-10-hydroxycamptothecin glucuronidation levels in the liver. Drug Metab Dispos 34 (2006) 1220-1228
    • (2006) Drug Metab Dispos , vol.34 , pp. 1220-1228
    • Girard, H.1    Villeneuve, L.2    Court, M.H.3
  • 19
    • 0036073404 scopus 로고    scopus 로고
    • Genetic polymorphisms of human organic anion transporters OATP-C (SLC21A6) and OATP-B (SLC21A9): allele frequencies in the Japanese population and functional analysis
    • Nozawa T., Nakajima M., Tamai I., et al. Genetic polymorphisms of human organic anion transporters OATP-C (SLC21A6) and OATP-B (SLC21A9): allele frequencies in the Japanese population and functional analysis. J Pharmacol Exp Ther 302 (2002) 804-813
    • (2002) J Pharmacol Exp Ther , vol.302 , pp. 804-813
    • Nozawa, T.1    Nakajima, M.2    Tamai, I.3
  • 20
    • 33744991123 scopus 로고    scopus 로고
    • Polymorphisms and linkage disequilibrium of the OATP8 (OATP1B3) gene in Japanese subjects
    • Tsujimoto M., Hirata S., Dan Y., Ohtani H., and Sawada Y. Polymorphisms and linkage disequilibrium of the OATP8 (OATP1B3) gene in Japanese subjects. Drug Metab Pharmacokinet 21 (2006) 165-169
    • (2006) Drug Metab Pharmacokinet , vol.21 , pp. 165-169
    • Tsujimoto, M.1    Hirata, S.2    Dan, Y.3    Ohtani, H.4    Sawada, Y.5
  • 21
    • 0035104031 scopus 로고    scopus 로고
    • Frequency of single nucleotide polymorphisms in the P-glycoprotein drug transporter MDR1 gene in white subjects
    • Cascorbi I., Gerloff T., Johne A., et al. Frequency of single nucleotide polymorphisms in the P-glycoprotein drug transporter MDR1 gene in white subjects. Clin Pharmacol Ther 69 (2001) 169-174
    • (2001) Clin Pharmacol Ther , vol.69 , pp. 169-174
    • Cascorbi, I.1    Gerloff, T.2    Johne, A.3
  • 22
    • 33750346955 scopus 로고    scopus 로고
    • Multidrug resistance protein 2 genetic polymorphisms influence mycophenolic acid exposure in renal allograft recipients
    • Naesens M., Kuypers D.R., Verbeke K., and Vanrenterghem Y. Multidrug resistance protein 2 genetic polymorphisms influence mycophenolic acid exposure in renal allograft recipients. Transplantation 82 (2006) 1074-1084
    • (2006) Transplantation , vol.82 , pp. 1074-1084
    • Naesens, M.1    Kuypers, D.R.2    Verbeke, K.3    Vanrenterghem, Y.4
  • 23
    • 33750958330 scopus 로고    scopus 로고
    • High-dose methotrexate in pediatric acute lymphoblastic leukemia: impact of ABCC2 polymorphisms on plasma concentrations
    • Rau T., Erney B., Gores R., Eschenhagen T., Beck J., and Langer T. High-dose methotrexate in pediatric acute lymphoblastic leukemia: impact of ABCC2 polymorphisms on plasma concentrations. Clin Pharmacol Ther 80 (2006) 468-476
    • (2006) Clin Pharmacol Ther , vol.80 , pp. 468-476
    • Rau, T.1    Erney, B.2    Gores, R.3    Eschenhagen, T.4    Beck, J.5    Langer, T.6
  • 24
    • 19944399722 scopus 로고    scopus 로고
    • Functional assessment of ABCG2 (BCRP) gene polymorphisms to protein expression in human placenta
    • Kobayashi D., Ieiri I., Hirota T., et al. Functional assessment of ABCG2 (BCRP) gene polymorphisms to protein expression in human placenta. Drug Metab Dispos 33 (2005) 94-101
    • (2005) Drug Metab Dispos , vol.33 , pp. 94-101
    • Kobayashi, D.1    Ieiri, I.2    Hirota, T.3
  • 25
    • 0036030902 scopus 로고    scopus 로고
    • Pharmacokinetic evaluation of an angiotensin II AT1 receptor antagonist BIBR277 (temisartan) in hypertensive patients
    • Ogihara T., Minami F., Kainuma H., et al. Pharmacokinetic evaluation of an angiotensin II AT1 receptor antagonist BIBR277 (temisartan) in hypertensive patients. Jpn Pharmacol Ther 30 (2002) S-271-S-283
    • (2002) Jpn Pharmacol Ther , vol.30
    • Ogihara, T.1    Minami, F.2    Kainuma, H.3
  • 26
    • 33747131444 scopus 로고    scopus 로고
    • Telmisartan improves insulin sensitivity in nondiabetic patients with essential hypertension
    • Benndorf R.A., Rudolph T., Appel D., et al. Telmisartan improves insulin sensitivity in nondiabetic patients with essential hypertension. Metabolism 55 (2006) 1159-1164
    • (2006) Metabolism , vol.55 , pp. 1159-1164
    • Benndorf, R.A.1    Rudolph, T.2    Appel, D.3
  • 27
    • 1842537144 scopus 로고    scopus 로고
    • Insulin-sensitizing effects of telmisartan: implications for treating insulin-resistant hypertension and cardiovascular disease
    • Pershadsingh H.A., and Kurtz T.W. Insulin-sensitizing effects of telmisartan: implications for treating insulin-resistant hypertension and cardiovascular disease. Diabetes Care 27 (2004) 1015
    • (2004) Diabetes Care , vol.27 , pp. 1015
    • Pershadsingh, H.A.1    Kurtz, T.W.2
  • 28
    • 14644444519 scopus 로고    scopus 로고
    • Replacement of valsartan and candesartan by telmisartan in hypertensive patients with type 2 diabetes: metabolic and antiatherogenic consequences
    • Miura Y., Yamamoto N., Tsunekawa S., et al. Replacement of valsartan and candesartan by telmisartan in hypertensive patients with type 2 diabetes: metabolic and antiatherogenic consequences. Diabetes Care 28 (2005) 757-758
    • (2005) Diabetes Care , vol.28 , pp. 757-758
    • Miura, Y.1    Yamamoto, N.2    Tsunekawa, S.3
  • 29
    • 0030800075 scopus 로고    scopus 로고
    • Differential expression of the UGT1A locus in human liver, biliary, and gastric tissue: identification of UGT1A7 and UGT1A10 transcripts in extrahepatic tissue
    • Strassburg C.P., Oldhafer K., Manns M.P., and Tukey R.H. Differential expression of the UGT1A locus in human liver, biliary, and gastric tissue: identification of UGT1A7 and UGT1A10 transcripts in extrahepatic tissue. Mol Pharmacol 52 (1997) 212-220
    • (1997) Mol Pharmacol , vol.52 , pp. 212-220
    • Strassburg, C.P.1    Oldhafer, K.2    Manns, M.P.3    Tukey, R.H.4
  • 30
    • 0034128936 scopus 로고    scopus 로고
    • Human UDP-glucuronosyltransferases: metabolism, expression, and disease
    • Tukey R.H., and Strassburg C.P. Human UDP-glucuronosyltransferases: metabolism, expression, and disease. Annu Rev Pharmacol Toxicol 40 (2000) 581-616
    • (2000) Annu Rev Pharmacol Toxicol , vol.40 , pp. 581-616
    • Tukey, R.H.1    Strassburg, C.P.2
  • 31
    • 0035209568 scopus 로고    scopus 로고
    • The role of hepatic and extrahepatic UDP-glucuronosyltransferases in human drug metabolism
    • Fisher M.B., Paine M.F., Strelevitz T.J., and Wrighton S.A. The role of hepatic and extrahepatic UDP-glucuronosyltransferases in human drug metabolism. Drug Metab Rev 33 (2001) 273-297
    • (2001) Drug Metab Rev , vol.33 , pp. 273-297
    • Fisher, M.B.1    Paine, M.F.2    Strelevitz, T.J.3    Wrighton, S.A.4
  • 32
    • 2442716361 scopus 로고    scopus 로고
    • Cyclosporin A, but not tacrolimus, inhibits the biliary excretion of mycophenolic acid glucuronide possibly mediated by multidrug resistance-associated protein 2 in rats
    • Kobayashi M., Saitoh H., Kobayashi M., Tadano K., Takahashi Y., and Hirano T. Cyclosporin A, but not tacrolimus, inhibits the biliary excretion of mycophenolic acid glucuronide possibly mediated by multidrug resistance-associated protein 2 in rats. J Pharmacol Exp Ther 309 (2004) 1029-1035
    • (2004) J Pharmacol Exp Ther , vol.309 , pp. 1029-1035
    • Kobayashi, M.1    Saitoh, H.2    Kobayashi, M.3    Tadano, K.4    Takahashi, Y.5    Hirano, T.6
  • 33
    • 25144489979 scopus 로고    scopus 로고
    • Population pharmacokinetics of mycophenolic acid in renal transplant recipients
    • van Hest R.M., van Gelder T., Vulto A.G., and Mathot R.A. Population pharmacokinetics of mycophenolic acid in renal transplant recipients. Clin Pharmacokinet 44 (2005) 1083-1096
    • (2005) Clin Pharmacokinet , vol.44 , pp. 1083-1096
    • van Hest, R.M.1    van Gelder, T.2    Vulto, A.G.3    Mathot, R.A.4
  • 34
    • 36148991372 scopus 로고    scopus 로고
    • Influence of SLCO1B1, 1B3, 2B1 and ABCC2 genetic polymorphisms on mycophenolic acid pharmacokinetics in Japanese renal transplant recipients
    • Miura M., Satoh S., Inoue K., et al. Influence of SLCO1B1, 1B3, 2B1 and ABCC2 genetic polymorphisms on mycophenolic acid pharmacokinetics in Japanese renal transplant recipients. Eur J Clin Pharmacol 63 (2007) 1161-1169
    • (2007) Eur J Clin Pharmacol , vol.63 , pp. 1161-1169
    • Miura, M.1    Satoh, S.2    Inoue, K.3
  • 35
    • 55349106941 scopus 로고    scopus 로고
    • Miura M, Kagaya H, Satoh S, et al. Influence of Drug Transporters and UGT Polymorphisms on Pharmacokinetics of Phenolic glucuronide Metabolite of Mycophenolic Acid in Japanese Renal Transplant Recipients. Ther Drug Monit 2008; In press.
    • Miura M, Kagaya H, Satoh S, et al. Influence of Drug Transporters and UGT Polymorphisms on Pharmacokinetics of Phenolic glucuronide Metabolite of Mycophenolic Acid in Japanese Renal Transplant Recipients. Ther Drug Monit 2008; In press.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.