High-Potency Olfactory Receptor Agonists Discovered by Virtual High-Throughput Screening: Molecular Probes for Receptor Structure and Olfactory Function

Neuron

Volumn 60, Issue 5, 2008, Pages 767-774

  Triballeau, Nicolas ^a,b   Van Name, Eric ^c   Laslier, Guillaume ^a   Cai, Diana ^d   Paillard, Guillaume ^b   Sorensen, Peter W ^d   Hoffmann, Rémy ^b   Bertrand, Hugues Olivier ^b   Ngai, John ^c   Acher, Francine C ^a  

^a UNIVERSITÉ PARIS DESCARTES   (France)

^b Parc Club Orsay Universite   (France)

^c UNIVERSITY OF CALIFORNIA   (United States)

^d UNIVERSITY OF MINNESOTA   (United States)

Author keywords

CELLBIO; CHEMBIO; MOLNEURO

Indexed keywords

ARGININE; G PROTEIN COUPLED RECEPTOR; LYSINE;

ARTICLE; BINDING AFFINITY; CHEMICAL STRUCTURE; CONTROLLED STUDY; HUMAN; HUMAN CELL; IN VIVO STUDY; LIGAND BINDING; MOLECULAR MODEL; OLFACTORY SYSTEM; PRIORITY JOURNAL; SENSORY RECEPTOR; STRUCTURE ANALYSIS;

AMINO ACIDS; ANIMALS; CALCIUM; CELL LINE, TRANSFORMED; COMPUTER-AIDED DESIGN; DRUG EVALUATION, PRECLINICAL; GOLDFISH; HUMANS; LIGANDS; MODELS, MOLECULAR; MOLECULAR PROBES; OLFACTORY RECEPTOR NEURONS; PROTEIN BINDING; PROTEIN CONFORMATION; RECEPTORS, ODORANT; ROC CURVE; SMALL MOLECULE LIBRARIES; SMELL; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 57049164250     PISSN: 08966273     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuron.2008.11.014     Document Type: Article

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