New N-pyridinyl(methyl)-indolalkanamides acting as topical inflammation inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 21, 2004, Pages 5441-5444

  Dassonville, Alexandra ^a   Bretéché, Anne ^a   Evano, Johan ^a   Duflos, Muriel ^a   Le Baut, Guillaume ^a   Grimaud, Nicole ^a   Petit, Jean Yves ^a  

^a UNIVERSITÉ DE NANTES   (France)

Author keywords

1 and 3 Indol(alkyl)carboxamides; Amino(methyl)pyridines; Nonacidic and nonsteroidal anti inflammatory drugs

Indexed keywords

2,3 DIHYDRO 5 METHYL 3 (MORPHOLINOMETHYL) 6 (1 NAPHTHOYL)PYRROLO[1,2,3 DE][1,4]BENZOXAZINE; ACID; AMIDE; DEXAMETHASONE; IBUPROFEN; N (PYRIDIN 3 YLMETHYL) 3 [5 CHLORO 1 (4 CHLOROBENZYL)INDOL 3 YL]PROPANAMIDE; NONSTEROID ANTIINFLAMMATORY AGENT; PROPIONAMIDE DERIVATIVE; TISSUE PLASMINOGEN ACTIVATOR; UNCLASSIFIED DRUG;

ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG MECHANISM; DRUG POTENCY; DRUG SCREENING; EDEMA; MOUSE; NONHUMAN; OTITIS;

ADMINISTRATION, CUTANEOUS; ADMINISTRATION, ORAL; AMIDES; ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; EAR, EXTERNAL; EDEMA; INDOLES; MICE; POLYUNSATURATED ALKAMIDES; PROPANE; PYRIDINES; STRUCTURE-ACTIVITY RELATIONSHIP; TETRADECANOYLPHORBOL ACETATE;

EID: 5344244051     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.07.057     Document Type: Article

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