Towards a species-selective acetylcholinesterase inhibitor to control the mosquito vector of malaria, Anopheles gambiae

Chemico-Biological Interactions

Volumn 175, Issue 1-3, 2008, Pages 368-375

  Carlier, Paul R ^a   Anderson, Troy D ^a   Wong, Dawn M ^a   Hsu, Danny C ^a   Hartsel, Joshua ^a   Ma, Ming ^a   Wong, Eric A ^a   Choudhury, Ranginee ^a   Lam, Polo C H ^b   Totrov, Maxim M ^b   Bloomquist, Jeffrey R ^a  

^a VIRGINIA POLYTECHNIC INSTITUTE AND STATE UNIVERSITY   (United States)

^b MOLSOFT LLC   (United States)

Author keywords

Acetylcholinesterase; Anopheles; Human; Inhibitor; Insecticide; Mosquito

Indexed keywords

1,5 BIS(4 ALLYLDIMETHYLAMMONIUMPHENYL)PENTAN 3 ONE DIBROMIDE; ACETYLCHOLINESTERASE; BIS(7) TACRINE; CHOLINESTERASE INHIBITOR; FASCICULIN II; GALANTAMINE; INSECTICIDE; PHYSOSTIGMINE; PROFENAMINE; PROPIDIUM IODIDE; PROPOXUR; PYRETHROID; TACRINE; UNCLASSIFIED DRUG;

AFRICA; ANIMAL CELL; ANOPHELES GAMBIAE; ARTICLE; BED NET; CRYSTAL STRUCTURE; DRUG POTENCY; DRUG SAFETY; DRUG SELECTIVITY; ENDEMIC DISEASE; ENZYME INHIBITION; ENZYME STRUCTURE; MALARIA; NONHUMAN; NUCLEOTIDE SEQUENCE; STRUCTURE ACTIVITY RELATION;

ACETYLCHOLINESTERASE; AMINO ACID SEQUENCE; ANIMALS; ANOPHELES; CHOLINESTERASE INHIBITORS; HUMANS; INSECT VECTORS; MALARIA; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; SPECIES SPECIFICITY;

ANOPHELES GAMBIAE;

EID: 50649083260     PISSN: 00092797     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.cbi.2008.04.037     Document Type: Article

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