메뉴 건너뛰기




Volumn 97, Issue 5, 2008, Pages 1843-1852

Theoretical dissolution model of poly-disperse drug particles in biorelevant media

Author keywords

Absorption; Dissolution; Gastrointestinal; Particle size; Phospholipids; Surfactants

Indexed keywords

BILE SALT; DANAZOL; GRISEOFULVIN; PHOSPHATIDYLCHOLINE; TAUROCHOLIC ACID; DRUG;

EID: 48549102969     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.21070     Document Type: Article
Times cited : (72)

References (42)
  • 2
    • 84956640361 scopus 로고    scopus 로고
    • Processing of biopharmaceutical profiling data in drug discovery
    • Testa B, Krämer SD, Wunderli-Allenspach H, Folkers G, Guy R, editors, Zurich: Wiley-VCH. pp
    • Sugano K, Obata K, Saitoh R, Higashida A, Hamada H. 2006. Processing of biopharmaceutical profiling data in drug discovery. In: Testa B, Krämer SD, Wunderli-Allenspach H, Folkers G, Guy R, editors. Pharmacokinetic profiling in drug research. Zurich: Wiley-VCH. pp 441-458.
    • (2006) Pharmacokinetic profiling in drug research , pp. 441-458
    • Sugano, K.1    Obata, K.2    Saitoh, R.3    Higashida, A.4    Hamada, H.5
  • 3
    • 0034461768 scopus 로고    scopus 로고
    • Drug-like properties and the causes of poor solubility and poor permeability
    • Lipinski CA. 2000. Drug-like properties and the causes of poor solubility and poor permeability. J Pharmacol Toxicol Methods 44:235-249.
    • (2000) J Pharmacol Toxicol Methods , vol.44 , pp. 235-249
    • Lipinski, C.A.1
  • 4
    • 0031024171 scopus 로고    scopus 로고
    • Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
    • Lipinski CA, Lombardo F, Dominy BW, Feeney PJ. 1997. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings. Adv Drug Deliv Rev 23:3-25.
    • (1997) Adv Drug Deliv Rev , vol.23 , pp. 3-25
    • Lipinski, C.A.1    Lombardo, F.2    Dominy, B.W.3    Feeney, P.J.4
  • 5
    • 0034655372 scopus 로고    scopus 로고
    • A high-throughput screening method for the determination of aqueous drug solubility using laser nephelometry in micro-titer plates
    • Bevan CD, Lloyd RS. 2000. A high-throughput screening method for the determination of aqueous drug solubility using laser nephelometry in micro-titer plates. Anal Chem 72:1781-1787.
    • (2000) Anal Chem , vol.72 , pp. 1781-1787
    • Bevan, C.D.1    Lloyd, R.S.2
  • 6
    • 0035150465 scopus 로고    scopus 로고
    • High throughput physicochemical profiling for drug discovery
    • Kerns EH. 2001. High throughput physicochemical profiling for drug discovery. J Pharm Sci 90:1838-1858.
    • (2001) J Pharm Sci , vol.90 , pp. 1838-1858
    • Kerns, E.H.1
  • 7
    • 0035120237 scopus 로고    scopus 로고
    • Determination of the aqueous solubility of drugs using a convenient 96-well plate-based assay
    • Roy D, Ducher F, Laumain A, Legendre JY. 2001. Determination of the aqueous solubility of drugs using a convenient 96-well plate-based assay. Drug Dev Ind Pharm 27:107-109.
    • (2001) Drug Dev Ind Pharm , vol.27 , pp. 107-109
    • Roy, D.1    Ducher, F.2    Laumain, A.3    Legendre, J.Y.4
  • 8
    • 0035468033 scopus 로고    scopus 로고
    • Physicochemical profiling (solubility, permeability and charge state)
    • Avdeef A. 2001. Physicochemical profiling (solubility, permeability and charge state). Curr Top Med Chem 1:277-351.
    • (2001) Curr Top Med Chem , vol.1 , pp. 277-351
    • Avdeef, A.1
  • 9
    • 1842432543 scopus 로고    scopus 로고
    • Biopharmaceutics classification by high throughput solubility assay and PAMPA
    • Obata K, Sugano K, Machida M, Aso Y. 2004. Biopharmaceutics classification by high throughput solubility assay and PAMPA. Drug Dev Ind Pharm 30:181.
    • (2004) Drug Dev Ind Pharm , vol.30 , pp. 181
    • Obata, K.1    Sugano, K.2    Machida, M.3    Aso, Y.4
  • 10
    • 33750000906 scopus 로고    scopus 로고
    • High throughput solubility measurement with automated polarized light microscopy analysis
    • Sugano K, Kato T, Suzuki K, Keiko K, Sujaku T, Mano T. 2006. High throughput solubility measurement with automated polarized light microscopy analysis. J Pharm Sci 95:2115-2122.
    • (2006) J Pharm Sci , vol.95 , pp. 2115-2122
    • Sugano, K.1    Kato, T.2    Suzuki, K.3    Keiko, K.4    Sujaku, T.5    Mano, T.6
  • 12
    • 0027263353 scopus 로고
    • Comparison of the mechanism of dissolution of hydrocortisone in simple and mixed micelle systems
    • Naylor LJ, Bakatselou V, Dressman JB. 1993. Comparison of the mechanism of dissolution of hydrocortisone in simple and mixed micelle systems. Pharm Res 10:865-870.
    • (1993) Pharm Res , vol.10 , pp. 865-870
    • Naylor, L.J.1    Bakatselou, V.2    Dressman, J.B.3
  • 13
    • 0030967838 scopus 로고    scopus 로고
    • A mechanistic study of griseofulvin dissolution into surfactant solutions under laminar flow conditions
    • Rao VM, Lin M, Larive CK, Southard MZ. 1997. A mechanistic study of griseofulvin dissolution into surfactant solutions under laminar flow conditions. J Pharm Sci 86:1132-1137.
    • (1997) J Pharm Sci , vol.86 , pp. 1132-1137
    • Rao, V.M.1    Lin, M.2    Larive, C.K.3    Southard, M.Z.4
  • 14
    • 12244261581 scopus 로고    scopus 로고
    • A mechanistic study of danazol dissolution in ionic surfactant solutions
    • Sun W, Larive CK, Southard MZ. 2003. A mechanistic study of danazol dissolution in ionic surfactant solutions. J Pharm Sci 92:424-435.
    • (2003) J Pharm Sci , vol.92 , pp. 424-435
    • Sun, W.1    Larive, C.K.2    Southard, M.Z.3
  • 15
    • 3843128718 scopus 로고    scopus 로고
    • Surfactant-mediated dissolution: Contributions of solubility enhancement and relatively low micelle diffusivity
    • Balakrishnan A, Rege BD, Amidon GL, Polli JE. 2004. Surfactant-mediated dissolution: Contributions of solubility enhancement and relatively low micelle diffusivity. J Pharm Sci 93:2064-2075.
    • (2004) J Pharm Sci , vol.93 , pp. 2064-2075
    • Balakrishnan, A.1    Rege, B.D.2    Amidon, G.L.3    Polli, J.E.4
  • 16
    • 0021828101 scopus 로고
    • Prediction of available surface area of powdered particles of flufenamic acid in tablets
    • Kouchiwa S, Nemoto M, Itai S, Murayama H, Nagai T. 1985. Prediction of available surface area of powdered particles of flufenamic acid in tablets. Chem Pharm Bull 33:1641-1651.
    • (1985) Chem Pharm Bull , vol.33 , pp. 1641-1651
    • Kouchiwa, S.1    Nemoto, M.2    Itai, S.3    Murayama, H.4    Nagai, T.5
  • 17
    • 0021798852 scopus 로고
    • Dissolution profiles of nalidixic acid powders having weibull particle size distribution
    • Kouchiwa S, Nemoto M, Itai S, Murayama H, Nagai T. 1985. Dissolution profiles of nalidixic acid powders having weibull particle size distribution. Chem Pharm Bull 33:2452-2460.
    • (1985) Chem Pharm Bull , vol.33 , pp. 2452-2460
    • Kouchiwa, S.1    Nemoto, M.2    Itai, S.3    Murayama, H.4    Nagai, T.5
  • 18
    • 0022409189 scopus 로고
    • Influence of wetting factors on the dissolution behavior of flufenamic acid
    • Itai S, Nemoto M, Kouchiwa S, Murayama H, Nagai T. 1985. Influence of wetting factors on the dissolution behavior of flufenamic acid. Chem Pharm Bull 33:5464-5473.
    • (1985) Chem Pharm Bull , vol.33 , pp. 5464-5473
    • Itai, S.1    Nemoto, M.2    Kouchiwa, S.3    Murayama, H.4    Nagai, T.5
  • 19
    • 0022636263 scopus 로고
    • Effect of compression pressure and formulation on the available surface area of flufenamic acid in tablets
    • Itai S, Kouchiwa S, Nemoto M, Murayama H, Nagai T. 1986. Effect of compression pressure and formulation on the available surface area of flufenamic acid in tablets. Chem Pharm Bull 34:1264-1274.
    • (1986) Chem Pharm Bull , vol.34 , pp. 1264-1274
    • Itai, S.1    Kouchiwa, S.2    Nemoto, M.3    Murayama, H.4    Nagai, T.5
  • 20
    • 0024596954 scopus 로고
    • The effect of particle size distribution on dissolution rate and oral absorption
    • Hintz RJ, Johnson KC. 1989. The effect of particle size distribution on dissolution rate and oral absorption. Int J Pharm 51:9-17.
    • (1989) Int J Pharm , vol.51 , pp. 9-17
    • Hintz, R.J.1    Johnson, K.C.2
  • 21
    • 0030444550 scopus 로고    scopus 로고
    • Guidance in the setting of drug particle size specifications to minimize variability in absorption
    • Johnson KC, Swindell AC. 1996. Guidance in the setting of drug particle size specifications to minimize variability in absorption. Pharm Res 13:1795-1798.
    • (1996) Pharm Res , vol.13 , pp. 1795-1798
    • Johnson, K.C.1    Swindell, A.C.2
  • 22
    • 0031750861 scopus 로고    scopus 로고
    • Evaluation of various dissolution media for predicting in vivo performance of class I and II drugs
    • Galia E, Nicolaides E, Horter D, Lobenberg R, Reppas C, Dressman JB. 1998. Evaluation of various dissolution media for predicting in vivo performance of class I and II drugs. Pharm Res 15:698-705.
    • (1998) Pharm Res , vol.15 , pp. 698-705
    • Galia, E.1    Nicolaides, E.2    Horter, D.3    Lobenberg, R.4    Reppas, C.5    Dressman, J.B.6
  • 23
    • 0033452575 scopus 로고    scopus 로고
    • Forecasting the in vivo performance of four low solubility drugs from their in vitro dissolution data
    • Nicolaides E, Galia E, Efthymiopoulos C, Dressman JB, Reppas C. 1999. Forecasting the in vivo performance of four low solubility drugs from their in vitro dissolution data. Pharm Res 16:1876-1882.
    • (1999) Pharm Res , vol.16 , pp. 1876-1882
    • Nicolaides, E.1    Galia, E.2    Efthymiopoulos, C.3    Dressman, J.B.4    Reppas, C.5
  • 24
    • 0034948871 scopus 로고    scopus 로고
    • Biorelevant dissolution testing to predict the plasma profile of lipophilic drugs after oral administration
    • Nicolaides E, Symillides M, Dressman JB, Reppas C. 2001. Biorelevant dissolution testing to predict the plasma profile of lipophilic drugs after oral administration. Pharm Res 18:380-388.
    • (2001) Pharm Res , vol.18 , pp. 380-388
    • Nicolaides, E.1    Symillides, M.2    Dressman, J.B.3    Reppas, C.4
  • 25
    • 33748936522 scopus 로고    scopus 로고
    • Effect of food intake on the oral absorption of poorly water-soluble drugs: In vitro assessment of drug dissolution and permeation assay system
    • Kataoka M, Masaoka Y, Sakuma S, Yamashita S. 2006. Effect of food intake on the oral absorption of poorly water-soluble drugs: In vitro assessment of drug dissolution and permeation assay system. J Pharm Sci 95:2051-2061.
    • (2006) J Pharm Sci , vol.95 , pp. 2051-2061
    • Kataoka, M.1    Masaoka, Y.2    Sakuma, S.3    Yamashita, S.4
  • 26
    • 33745416604 scopus 로고    scopus 로고
    • Oral absorption of poorly water-soluble drugs: Computer simulation of fraction absorbed in humans from a miniscale dissolution test
    • Takano R, Sugano K, Higashida A, Hayashi Y, Machida M, Aso Y, Yamashita S. 2006. Oral absorption of poorly water-soluble drugs: Computer simulation of fraction absorbed in humans from a miniscale dissolution test. Pharm Res 23:1144-1156.
    • (2006) Pharm Res , vol.23 , pp. 1144-1156
    • Takano, R.1    Sugano, K.2    Higashida, A.3    Hayashi, Y.4    Machida, M.5    Aso, Y.6    Yamashita, S.7
  • 27
    • 0002642747 scopus 로고
    • Theorie der Reaktionsgeschwin-digkeit in heterogenen Systemen
    • Nernst W. 1904. Theorie der Reaktionsgeschwin-digkeit in heterogenen Systemen. Z Phys Chem 47: 52-55.
    • (1904) Z Phys Chem , vol.47 , pp. 52-55
    • Nernst, W.1
  • 28
    • 33747373878 scopus 로고    scopus 로고
    • A century of dissolution research: From Noyes and Whitney to the Biopharmaceutics Classification System
    • Dokoumetzidis A, Macheras P. 2006. A century of dissolution research: From Noyes and Whitney to the Biopharmaceutics Classification System. Int J Pharm 321:1-11.
    • (2006) Int J Pharm , vol.321 , pp. 1-11
    • Dokoumetzidis, A.1    Macheras, P.2
  • 30
    • 0029879771 scopus 로고    scopus 로고
    • Control of poorly soluble drug dissolution in conditions simulating the gastrointestinal tract flow. 1. Effect of tablet geometry in buffered medium
    • Chakrabarti S, Southard MZ. 1996. Control of poorly soluble drug dissolution in conditions simulating the gastrointestinal tract flow. 1. Effect of tablet geometry in buffered medium. J Pharm Sci 86:313-319.
    • (1996) J Pharm Sci , vol.86 , pp. 313-319
    • Chakrabarti, S.1    Southard, M.Z.2
  • 31
    • 0030992126 scopus 로고    scopus 로고
    • Control of poorly soluble drug dissolution in conditions simulating the gastrointestinal tract flow. 2. Cocom-pression of drugs with buffers
    • Chakrabarti S, Southard MZ. 1997. Control of poorly soluble drug dissolution in conditions simulating the gastrointestinal tract flow. 2. Cocom-pression of drugs with buffers. J Pharm Sci 86:465-469.
    • (1997) J Pharm Sci , vol.86 , pp. 465-469
    • Chakrabarti, S.1    Southard, M.Z.2
  • 33
    • 0020471096 scopus 로고
    • Effect of food on the bioavailability of griseofulvin from microsize and PEG ultramicrosize (GRIS-PEG) plain tablets
    • Aoyagi N, Ogata H, Kaniwa N, Ejima A. 1982. Effect of food on the bioavailability of griseofulvin from microsize and PEG ultramicrosize (GRIS-PEG) plain tablets. J Pharmacobio-Dyn 5:120-124.
    • (1982) J Pharmacobio-Dyn , vol.5 , pp. 120-124
    • Aoyagi, N.1    Ogata, H.2    Kaniwa, N.3    Ejima, A.4
  • 34
    • 0027287976 scopus 로고
    • Effect of food and a monoglyceride emulsion formulation on danazol bioavailability
    • Charman WN, Rogge MC, Boddy AW, Berger BM. 1993. Effect of food and a monoglyceride emulsion formulation on danazol bioavailability. J Clin Pharmacol 33:381-386.
    • (1993) J Clin Pharmacol , vol.33 , pp. 381-386
    • Charman, W.N.1    Rogge, M.C.2    Boddy, A.W.3    Berger, B.M.4
  • 35
    • 0034707091 scopus 로고    scopus 로고
    • Phase boundaries in mixtures of membrane-forming amphiphiles and micelle-forming amphiphiles
    • Lichtenberg D, Opatowski E, Kozlov MM. 2000. Phase boundaries in mixtures of membrane-forming amphiphiles and micelle-forming amphiphiles. Biochim Biophys Acta 1508:1-19.
    • (2000) Biochim Biophys Acta , vol.1508 , pp. 1-19
    • Lichtenberg, D.1    Opatowski, E.2    Kozlov, M.M.3
  • 36
    • 14144250013 scopus 로고    scopus 로고
    • In vivo in vitro correlations for a poorly soluble drug, danazol, using the flow-through dissolution method with biorelevant dissolution media
    • Sunesen VH, Pedersen BL, Kristensen HG, Mullertz A. 2005. In vivo in vitro correlations for a poorly soluble drug, danazol, using the flow-through dissolution method with biorelevant dissolution media. Eur J Pharm Sci 24:305-313.
    • (2005) Eur J Pharm Sci , vol.24 , pp. 305-313
    • Sunesen, V.H.1    Pedersen, B.L.2    Kristensen, H.G.3    Mullertz, A.4
  • 37
    • 32644443825 scopus 로고    scopus 로고
    • Biorelevant dissolution media: Aggregation of amphiphiles and solubility of estradiol
    • Ilardia-Arana D, Kristensen HG, Mullertz A. 2006. Biorelevant dissolution media: Aggregation of amphiphiles and solubility of estradiol. J Pharm Sci 95:248-255.
    • (2006) J Pharm Sci , vol.95 , pp. 248-255
    • Ilardia-Arana, D.1    Kristensen, H.G.2    Mullertz, A.3
  • 38
    • 0036803219 scopus 로고    scopus 로고
    • Prediction of intestinal absorption: Comparative assessment of GASTRO-PLUS and IDEA
    • Parrott N, Lave T. 2002. Prediction of intestinal absorption: Comparative assessment of GASTRO-PLUS and IDEA. Eur J Pharm Sci 17:51-61.
    • (2002) Eur J Pharm Sci , vol.17 , pp. 51-61
    • Parrott, N.1    Lave, T.2
  • 39
    • 28444451169 scopus 로고    scopus 로고
    • A strategy for preclinical formulation development using GastroPlus(TM) as pharmacokinetic simulation tool and a statistical screening design applied to a dog study
    • Kuentz M, Nick S, Parrott N, Rothlisberger D. 2006. A strategy for preclinical formulation development using GastroPlus(TM) as pharmacokinetic simulation tool and a statistical screening design applied to a dog study. Eur J Pharm Sci 27:91-99.
    • (2006) Eur J Pharm Sci , vol.27 , pp. 91-99
    • Kuentz, M.1    Nick, S.2    Parrott, N.3    Rothlisberger, D.4
  • 40
    • 84956632541 scopus 로고    scopus 로고
    • Predicting the intestinal solubility of poorly soluble drugs
    • Testa B, Krämer SD, Wunderli-Allenspach H, Folkers G, Guy R, editors, Zurich: Wiley-VCH. pp
    • Glomme A, März J, Dressman JB. 2006. Predicting the intestinal solubility of poorly soluble drugs. In: Testa B, Krämer SD, Wunderli-Allenspach H, Folkers G, Guy R, editors. Pharmacokinetic profiling in drug research. Zurich: Wiley-VCH. pp 260-280.
    • (2006) Pharmacokinetic profiling in drug research , pp. 260-280
    • Glomme, A.1    März, J.2    Dressman, J.B.3
  • 41
    • 84956610645 scopus 로고    scopus 로고
    • Calculation of lipophilicity: A classification of methods
    • Testa B, Krämer SD, Wunderli-Allenspach H, Folkers G, Guy R, editors, Zurich: Wiley-VCH. pp
    • Mannhold R. 2006. Calculation of lipophilicity: A classification of methods. In: Testa B, Krämer SD, Wunderli-Allenspach H, Folkers G, Guy R, editors. Pharmacokinetic profiling in drug research. Zurich: Wiley-VCH. pp 333-352.
    • (2006) Pharmacokinetic profiling in drug research , pp. 333-352
    • Mannhold, R.1
  • 42
    • 13544270908 scopus 로고    scopus 로고
    • Predicting aqueous solubility from structure
    • Delaney JS. 2005. Predicting aqueous solubility from structure. Drug Discov Today 10:289-295.
    • (2005) Drug Discov Today , vol.10 , pp. 289-295
    • Delaney, J.S.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.