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Volumn 13, Issue 7-8, 2008, Pages 360-367

Snapshot PK: a rapid rodent in vivo preclinical screening approach

Author keywords

[No Author keywords available]

Indexed keywords

AUTOMATION; DATA ANALYSIS; DRUG EXPOSURE; IN VIVO STUDY; METHODOLOGY; PHARMACOKINETICS; REVIEW; RODENT; SAMPLING; SNAPSHOT PHARMACOKINETICS;

EID: 41549121839     PISSN: 13596446     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.drudis.2007.10.014     Document Type: Review
Times cited : (62)

References (28)
  • 1
    • 0037277752 scopus 로고    scopus 로고
    • Drug metabolism and pharmacokinetics in drug discovery
    • Roberts S.A. Drug metabolism and pharmacokinetics in drug discovery. Curr. Opin. Drug Discov. Dev. 6 (2003) 66-80
    • (2003) Curr. Opin. Drug Discov. Dev. , vol.6 , pp. 66-80
    • Roberts, S.A.1
  • 2
    • 4344645978 scopus 로고    scopus 로고
    • Can the pharmaceutical industry reduce attrition rates?
    • Kola I., and Landis J. Can the pharmaceutical industry reduce attrition rates?. Nat. Rev. Drug Discov. 3 (2004) 711-715
    • (2004) Nat. Rev. Drug Discov. , vol.3 , pp. 711-715
    • Kola, I.1    Landis, J.2
  • 3
    • 0037376928 scopus 로고    scopus 로고
    • Pharmaceutical profiling in drug discovery
    • Kerns E.H., and Di L. Pharmaceutical profiling in drug discovery. DDT 8 (2003) 316-323
    • (2003) DDT , vol.8 , pp. 316-323
    • Kerns, E.H.1    Di, L.2
  • 4
    • 0033178249 scopus 로고    scopus 로고
    • Pharmacokinetics and metabolism in early drug discovery
    • Smith D.A., and van de Waterbeemd H. Pharmacokinetics and metabolism in early drug discovery. Curr. Opin. Chem. Biol. 3 (1999) 373-378
    • (1999) Curr. Opin. Chem. Biol. , vol.3 , pp. 373-378
    • Smith, D.A.1    van de Waterbeemd, H.2
  • 5
    • 2942525302 scopus 로고    scopus 로고
    • Applications of high-throughput ADME in drug discovery
    • Kassel D.B. Applications of high-throughput ADME in drug discovery. Curr. Opin. Chem. Biol. 8 (2004) 339-345
    • (2004) Curr. Opin. Chem. Biol. , vol.8 , pp. 339-345
    • Kassel, D.B.1
  • 6
    • 0034955150 scopus 로고    scopus 로고
    • Pharmacokinetic theory of cassette dosing in drug discovery screening
    • White R.E., and Manitpisitkul R. Pharmacokinetic theory of cassette dosing in drug discovery screening. Drug Metab. Dispos. 29 (2001) 957-966
    • (2001) Drug Metab. Dispos. , vol.29 , pp. 957-966
    • White, R.E.1    Manitpisitkul, R.2
  • 7
    • 0034949807 scopus 로고    scopus 로고
    • Cassette dosing pharmacokinetics: valuable tool or flawed science?
    • Christ D.D. Cassette dosing pharmacokinetics: valuable tool or flawed science?. Drug Metab. Dispos. 29 (2001) 957-966
    • (2001) Drug Metab. Dispos. , vol.29 , pp. 957-966
    • Christ, D.D.1
  • 8
    • 0033136333 scopus 로고    scopus 로고
    • Novel in vivo procedure for rapid pharmacokinetic screening of discovery compounds in rat
    • Cox K.A., et al. Novel in vivo procedure for rapid pharmacokinetic screening of discovery compounds in rat. DDT 4 (1999) 232-237
    • (1999) DDT , vol.4 , pp. 232-237
    • Cox, K.A.1
  • 9
    • 33747193298 scopus 로고    scopus 로고
    • An efficient approach for the rapid assessment of oral rat exposures for new chemical entities in drug discovery
    • Han H.-K., et al. An efficient approach for the rapid assessment of oral rat exposures for new chemical entities in drug discovery. J. Pharm. Sci. 9 (2006) 1684-1692
    • (2006) J. Pharm. Sci. , vol.9 , pp. 1684-1692
    • Han, H.-K.1
  • 10
    • 0031000066 scopus 로고    scopus 로고
    • Simultaneous pharmacokinetic screening of a mixture of compounds in the dog using API LC/MS/MS analysis for increased throughput
    • Berman J., et al. Simultaneous pharmacokinetic screening of a mixture of compounds in the dog using API LC/MS/MS analysis for increased throughput. J. Med. Chem. 40 (1997) 827-829
    • (1997) J. Med. Chem. , vol.40 , pp. 827-829
    • Berman, J.1
  • 11
    • 0031906913 scopus 로고    scopus 로고
    • Sample pooling to expedite bioanalysis and pharmacokinetic research
    • Kuo B.S., et al. Sample pooling to expedite bioanalysis and pharmacokinetic research. J. Pharmaceut. Biomed. Anal. 16 (1998) 837-846
    • (1998) J. Pharmaceut. Biomed. Anal. , vol.16 , pp. 837-846
    • Kuo, B.S.1
  • 12
    • 3242778456 scopus 로고    scopus 로고
    • Whatever happened to cassette-dosing pharmacokinetics?
    • Manitpisitkul P., and White R.E. Whatever happened to cassette-dosing pharmacokinetics?. DDT 9 (2004) 652-658
    • (2004) DDT , vol.9 , pp. 652-658
    • Manitpisitkul, P.1    White, R.E.2
  • 13
    • 0031915533 scopus 로고    scopus 로고
    • Rapid determination of oral pharmacokinetics and plasma free fraction using cocktail approaches: methods and application
    • Allen M.C., et al. Rapid determination of oral pharmacokinetics and plasma free fraction using cocktail approaches: methods and application. Pharm. Res. 15 (1998) 93-97
    • (1998) Pharm. Res. , vol.15 , pp. 93-97
    • Allen, M.C.1
  • 14
    • 0035100437 scopus 로고    scopus 로고
    • Cassette-accelerated rapid rat screen: a systematic procedure for the dosing and liquid chromatography/atmospheric pressure ionization tandem mass spectrometric analysis of new chemical entities as part of new drug discovery
    • Korfmacher W.A., et al. Cassette-accelerated rapid rat screen: a systematic procedure for the dosing and liquid chromatography/atmospheric pressure ionization tandem mass spectrometric analysis of new chemical entities as part of new drug discovery. Rapid Commun. Mass Spectrom. 15 (2001) 335-340
    • (2001) Rapid Commun. Mass Spectrom. , vol.15 , pp. 335-340
    • Korfmacher, W.A.1
  • 15
    • 33747031401 scopus 로고    scopus 로고
    • Rapid in vivo oral screening in rats: reliability, acceptance criteria and filtering efficiency
    • Mei H., et al. Rapid in vivo oral screening in rats: reliability, acceptance criteria and filtering efficiency. AAPS J. 8 (2006) E493-E500
    • (2006) AAPS J. , vol.8
    • Mei, H.1
  • 16
    • 13144276327 scopus 로고    scopus 로고
    • In vivo pharmacokinetic screening in cassette dosing experiments; the use of on-line Prospekt liquid chromatography/atmospheric pressure chemical ionization tandem mass spectrometry technology in drug discovery
    • Beaudry F., et al. In vivo pharmacokinetic screening in cassette dosing experiments; the use of on-line Prospekt liquid chromatography/atmospheric pressure chemical ionization tandem mass spectrometry technology in drug discovery. Rapid Commun. Mass Spectrom. 12 (1998) 1216-1222
    • (1998) Rapid Commun. Mass Spectrom. , vol.12 , pp. 1216-1222
    • Beaudry, F.1
  • 17
    • 4444352458 scopus 로고    scopus 로고
    • Automated 96-well liquid-liquid back extraction liquid chromatography-tandem mass spectrometry method for the determination of ABT-202 in human plasma
    • Xu N., et al. Automated 96-well liquid-liquid back extraction liquid chromatography-tandem mass spectrometry method for the determination of ABT-202 in human plasma. J. Pharm. Biomed. Anal. 36 (2004) 189-195
    • (2004) J. Pharm. Biomed. Anal. , vol.36 , pp. 189-195
    • Xu, N.1
  • 18
    • 0034212552 scopus 로고    scopus 로고
    • Bioanalytical high-throughput selected reaction monitoring-LC/MS determination of selected estrogen receptor modulators in human plasma: 2000 samples/day
    • Zweigenbaum J., and Henion J. Bioanalytical high-throughput selected reaction monitoring-LC/MS determination of selected estrogen receptor modulators in human plasma: 2000 samples/day. Anal. Chem. 72 (2000) 2446-2454
    • (2000) Anal. Chem. , vol.72 , pp. 2446-2454
    • Zweigenbaum, J.1    Henion, J.2
  • 19
    • 0036164807 scopus 로고    scopus 로고
    • Direct cocktail analysis of drug discovery compounds in pooled plasma samples using liquid chromatography-tandem mass spectrometry
    • Hsieh Y., et al. Direct cocktail analysis of drug discovery compounds in pooled plasma samples using liquid chromatography-tandem mass spectrometry. J. Chromatogr. B: Analyt. Technol. Biomed. Life Sci. 767 (2002) 353-362
    • (2002) J. Chromatogr. B: Analyt. Technol. Biomed. Life Sci. , vol.767 , pp. 353-362
    • Hsieh, Y.1
  • 20
    • 3042599892 scopus 로고    scopus 로고
    • SOS - a sample ordering system for delivering 'assay-ready' compound plates for drug screening
    • Brideau C., et al. SOS - a sample ordering system for delivering 'assay-ready' compound plates for drug screening. JALA 9 (2004) 123-127
    • (2004) JALA , vol.9 , pp. 123-127
    • Brideau, C.1
  • 21
    • 0031884052 scopus 로고    scopus 로고
    • Automated 96-well solid phase extraction for the determination of doramectin in cattle plasma
    • Harrison A.C., and Walker D.K. Automated 96-well solid phase extraction for the determination of doramectin in cattle plasma. J. Pharmaceut. Biomed. Anal. 16 (1998) 777-783
    • (1998) J. Pharmaceut. Biomed. Anal. , vol.16 , pp. 777-783
    • Harrison, A.C.1    Walker, D.K.2
  • 22
    • 0033788742 scopus 로고    scopus 로고
    • AutoScan: an automated workstation for rapid determination of mass and tandem mass spectrometry conditions for quantitative bioanalytical mass spectrometry
    • Whalen K.M., et al. AutoScan: an automated workstation for rapid determination of mass and tandem mass spectrometry conditions for quantitative bioanalytical mass spectrometry. Rapid Commun. Mass Spectrom. 14 (2000) 2074-2079
    • (2000) Rapid Commun. Mass Spectrom. , vol.14 , pp. 2074-2079
    • Whalen, K.M.1
  • 23
    • 10844283579 scopus 로고    scopus 로고
    • Automatic mass spectrometry method development for drug discovery: applications in metabolic stability assays
    • Chovan L.E., et al. Automatic mass spectrometry method development for drug discovery: applications in metabolic stability assays. Rapid Commun. Mass Spectrom. 18 (2004) 3105-3112
    • (2004) Rapid Commun. Mass Spectrom. , vol.18 , pp. 3105-3112
    • Chovan, L.E.1
  • 24
    • 33646745530 scopus 로고    scopus 로고
    • A centralized approach to tandem mass spectrometry method development for high-throughput ADME screening
    • Whalen K., et al. A centralized approach to tandem mass spectrometry method development for high-throughput ADME screening. Rapid Commun. Mass Spectrom. 20 (2006) 1497-1503
    • (2006) Rapid Commun. Mass Spectrom. , vol.20 , pp. 1497-1503
    • Whalen, K.1
  • 25
    • 41549110460 scopus 로고    scopus 로고
    • Unattended LC/MS/MS method development for drug discovery: application for in-vitro ADME assays and in-vivo snapshot animal PK studies
    • (Abstract 522)
    • Gordon W.P., et al. Unattended LC/MS/MS method development for drug discovery: application for in-vitro ADME assays and in-vivo snapshot animal PK studies. Drug Metab. Rev. 37 s2 (2005) 284 (Abstract 522)
    • (2005) Drug Metab. Rev. , vol.37 , Issue.SUPPL.2 , pp. 284
    • Gordon, W.P.1
  • 26
    • 0034880597 scopus 로고    scopus 로고
    • Pharmacokinetics and its role in small molecule drug discovery research
    • Jang J.R., et al. Pharmacokinetics and its role in small molecule drug discovery research. Med. Res. Rev. 21 (2001) 382-396
    • (2001) Med. Res. Rev. , vol.21 , pp. 382-396
    • Jang, J.R.1
  • 27
    • 41549097042 scopus 로고    scopus 로고
    • Snapshot PK: a high throughput approach for in vivo preclinical PK studies
    • (Abstract 389)
    • Liu B., et al. Snapshot PK: a high throughput approach for in vivo preclinical PK studies. Drug Metab. Rev. 37 s2 (2005) 214 (Abstract 389)
    • (2005) Drug Metab. Rev. , vol.37 , Issue.SUPPL.2 , pp. 214
    • Liu, B.1
  • 28
    • 26844558233 scopus 로고    scopus 로고
    • Optimizing an ultrafast generic high-performance liquid chromatography/tandem mass spectrometry method for faster discovery pharmacokinetic sample throughput
    • Dunn-Meynell K.W., Wainhaus S., and Korfmacher W.A. Optimizing an ultrafast generic high-performance liquid chromatography/tandem mass spectrometry method for faster discovery pharmacokinetic sample throughput. Rapid Commun. Mass Spectrom. 19 (2005) 2905-2910
    • (2005) Rapid Commun. Mass Spectrom. , vol.19 , pp. 2905-2910
    • Dunn-Meynell, K.W.1    Wainhaus, S.2    Korfmacher, W.A.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.