Molecular actions of propofol on human 5-HT3A receptors: Enhancement as well as inhibition by closely related phenol derivatives

Anesthesia and Analgesia

Volumn 106, Issue 3, 2008, Pages 846-857

  Barann, Martin ^a   Linden, Isabelle ^a   Witten, Stefan ^a   Urban, Bernd W ^a  

^a UNIVERSITY OF BONN   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

2 ISOPROPYLPHENOL; 5 HYDROXYINDOLE; BENZENE; COMPLEMENTARY DNA; HYDROXYL GROUP; PHENOL; PHENOL DERIVATIVE; PROPOFOL; SEROTONIN 3 RECEPTOR; SEROTONIN 3A RECEPTOR; SEROTONIN DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CELL STRAIN HEK293; CHEMOSENSITIVITY; CONCENTRATION RESPONSE; CONTROLLED STUDY; DESENSITIZATION; DRUG CONFORMATION; DRUG EFFECT; DRUG MECHANISM; DRUG POTENCY; DRUG TARGETING; EMBRYO; GENETIC TRANSFECTION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN CELL; HYDROPHOBICITY; IC 50; INHIBITION KINETICS; MOLECULAR DYNAMICS; PATCH CLAMP; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION;

EID: 39749114992     PISSN: 00032999     EISSN: None     Source Type: Journal    
DOI: 10.1213/ane.0b013e318162ca7c     Document Type: Article

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