CGP7930: A positive allosteric modulator of the GABAB receptor

CNS Drug Reviews

Volumn 13, Issue 3, 2007, Pages 308-316

  Adams, C L ^a,b   Lawrence, A J ^b,c  

^a MONASH UNIVERSITY   (Australia)

^b FLOREY INSTITUTE OF NEUROSCIENCE AND MENTAL HEALTH   (Australia)

^c UNIVERSITY OF MELBOURNE   (Australia)

Author keywords

Alcohol; CGP7930; Drug seeking; GABAB receptors

Indexed keywords

(((3 (1 (3 CARBOXYPHENYL)ETHYL)AMINO)2 HYDROXYPROPYL)CYCLOHEXYLMETHYL PHOSPHINIC ACID); (3 (3',5' DI TERT BUTYL 4' HYDROXY)PHENYL 2,2 DIMETHYLPROPANOLO); (N,N' DICYCLOPENTYL 2 METHYLSULFANYL 5 NITRO PYRIMIDINE 4,6 DIAMINE); 4 AMINOBUTYRIC ACID B RECEPTOR; 4 AMINOBUTYRIC ACID B RECEPTOR STIMULATING AGENT; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; 5,5 DIMETHYL 2 MORPHOLINEACETIC ACID; [3 [1 (3 CARBOXYPHENYL)ETHYLAMINO] 2 HYDROXYPROPYL]CYCLOHEXYLMETHYLPHOSPHINIC ACID; ACTIVATING TRANSCRIPTION FACTOR 4; ALCOHOL; BACLOFEN; CALCIUM; CGP 7930; COCAINE; GS 39783; NICOTINE; UNCLASSIFIED DRUG;

ALLOSTERISM; ANALGESIA; ANXIETY; DEPRESSION; DRUG ACTIVITY; DRUG EFFECT; DRUG POTENCY; DRUG STRUCTURE; HUMAN; HYPNOSIS; HYPOTENSION; IN VITRO STUDY; IN VIVO STUDY; LIGAND BINDING; NERVE CELL; NONHUMAN; REVIEW; SEDATION; SIGNAL TRANSDUCTION; TRANQUILIZING ACTIVITY;

ANIMALS; PHENOLS; RECEPTORS, GABA-B; STEREOISOMERISM;

EID: 34748898892     PISSN: 1080563X     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1527-3458.2007.00021.x     Document Type: Review

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