Characterization of tableting using the OSDRC system

Pharmaceutical Research

Volumn 24, Issue 10, 2007, Pages 1902-1909

  Shimizu, Kazuyuki ^a   Ando, Masaki ^a   Nakayama, Yukiharu ^a  

^a SANWA KAGAKU KENKYUSHO CO LTD   (Japan)

Author keywords

Compression; Conventional compression; Crushing strength; OSDRC; Tablet improvement

Indexed keywords

PHENACETIN;

ARTICLE; CRUSHING STRENGTH; DRUG GRANULATION; DRUG RESEARCH; POWDER; PRIORITY JOURNAL; TABLET COMPRESSION; TABLET FORMULATION; TABLET MANUFACTURE; TABLET PROPERTY; TABLET THICKNESS;

CELLULOSE; COMPRESSIVE STRENGTH; LACTOSE; PHENACETIN; POROSITY; POWDERS; PRESSURE; STEARIC ACIDS; TABLETS; TECHNOLOGY, PHARMACEUTICAL;

EID: 34548565780     PISSN: 07248741     EISSN: 1573904X     Source Type: Journal    
DOI: 10.1007/s11095-007-9315-3     Document Type: Article

References (32)

1. Y. Ozeki, Y. Watanabe, H. Okamoto, and K. Danjo. Development of dividable one-step dry-coated tablets (dividable-OSDRC) and their evaluation as a new platform for controlled drug release. Pharm. Res. 21:1177-1783 (2004).
2. Y. Ozeki, M. Ando, Y. Watanabe, and K. Danjo. Evaluation of novel one-step dry-coated tablets as a platform for delayed-release tablets. J. Control. Release. 95:51-60 (2004).
3. S. Ohmori, and T. Makino. Sustained-release phenylpropanolamine hydrochloride bilayer caplets containing the hydroxypropylmethylcellulose 2208 matrix. I. Formulation and dissolution characteristics. Chem. Pharm. Bull. (Tokyo). 48:678-682 (2000).
4. L. Yang, and R. Fassihi. Accessibility of solid core tablet for dissolution in an asymmetric triple-layer matrix system. J. Pharm. Pharmacol. 55:1331-1337 (2003).
5. N. A. Armstrong, N. M. A. H. Abourida, and L. Krijgsman. Multiple compression of powders in tablet press. J. Pharm. Pharmacol. 34:9-13 (1982).
6. C. J. de Blaey, A. B. Weekers-Andersen, and J. Polderman. Compression of pharmaceuticals. V. Formulation development of a new compound with the aid of quantitative force-displacement measurements. Pharm. Weekbl. 106:893-903 (1971).
7. K. Danjo, H. Kimura, and A. Otsuka. Infuence of punch velocity on the compressibility of granules. Drug Dev. Ind. Pharm. 22:933-942 (1996).
8. K. Danjo, A. Hiramatsu, and A. Otsuka. Effect of punch velocity on the compressibility and stress relaxation of particles and granules. J. Soc. Powder Technol. Jpn. 35:662-670 (1998).
9. A. Nokhodchi, J. L. Ford, and M. H. Rubinstein. The effect of particle size and viscosity grade on the compaction properties of hydroxypropylmethylcellulose 2208. Int. J. Pharm. 48:1122-1127 (1996).
10. K. Goto, H. Sunada, K. Danjyo, and Y. Yonezawa. Pharmaceutical evaluation of multipurpose excipients for direct compressed tablet manufacture: comparisons of the capabilities of multipurpose excipients with those in general use. Drug Dev. Ind. Pharm. 25:869-878 (1999).
11. H. Aoshima, A. Miyagisnima, Y. Nozawa, Y. Sadzuka, and T. Sonobe. Glycerin fatty acid esters as a new lubricant of tablets. Int. J. Pharm. 293:25-35 (2005).
12. K. D. Ertel, and J. T. Carstensen. Chemical, physical and lubricant properties of magnesium stearate. J. Pharm. Sci. 77:625-629 (1988).
13. H. Yuasa, M. Akutagawa, T. Hashizume, and Y. Kanaya. Studies on internal structure of tablets. VI. stress dispersion in tablets by excipients. Chem. Pharm. Bull. 44:378-382 (1996).
14. P. Ditrich, A. Bauer-Brandl, and R. Schubert. Influence of tableting forces and lubricant concentration on the adhesion strength in complex layer tablets. Drug Dev. Ind. Pharm. 26:745-754 (2000).
15. L. Yang, G. Venkatesh, and R. Fassihi. Compaction simulator study of a novel triple-layer tablet matrix for industrial tableting. Int. J. Pharm. 152:45-52 (1997).
16. P. M. Belda, and J. B. Mielck. Considerations about the theoretically expected crushing strength of tablets from binary powder mixtures: double layer tablets versus arithmetic additivity rule. Eur. J. Pharm. Biopharm. 64:343-350 (2006).
17. W. I. Thomas, G. Rowley, and G. Doveston. An investigation of the influence of the core material properties on the compression and properties of dry-coated tablets. Drug Dev. Ind. Pharm. 24:973-978 (1998).
18. H. Murakami, T. Yoneyama, K. Nakajima, and M. Kobayashi. Correlation between loose density and compatibility of granules prepared by various granulation methods. Int. J. Pharm. 216:159-164 (2001).
19. J. Berggren, and G. Alderborn. Effect of drying rate on porosity and tabletting behavior of cellulose pellets. Int. J. Pharm. 227:81-96 (2001).
20. P. Di Martino, E. Joiris, and S. Martelli. Particle interaction of lubricated or unlubricated binary mixtures according to their particle size and densification mechanism. Farmaco. 59:747-758 (2004).
21. E. Joiris, P. Di Martino, C. Berneron, A. M. Guyot-Hermann, and J. C. Guyot. Compression behavior of orthorhombic paracetamol. Pharm. Res. 15:1122-1130 (1998).
22. Y. Shibata, M. Fujii, H. Okada, S. Noda, M. Kondoh, and Y. Watanabe. Evaluation of the compaction properties of a solid dispersion of indomethacin with crospovidone by tableting process analyzer. Chem. Pharm. Bull. (Tokyo). 53:759-763 (2005).
23. A. Munoz-Ruiz, M. Wihervaara, M. Hakkinken, M. Juslin, and P. Paronen. Frictional work in double-sided tablet compression. J. Pharm. Sci. 86:481-486 (1997).
24. Y. Shibata, M. Fujii, S. Noda, M. Kokudai, H. Okada, M. Kondoh, and Y. Watanabe. Fluidity and tableting characteristics of a powder solid dispersion of the low melting drugs ketoprofen and ibuprofen with crospovidone. Drug Dev. Ind. Pharm. 32:449-456 (2006).
25. H. Takeuchi, S. Nagira, H. Yamamoto, and Y. Kawashima. Die wall pressure measurement for evaluation of compaction property of pharmaceutical materials. Int. J. Pharm. 274:131-138 (2004).
26. Y. Ozeki, and K. Danjyo. Effect of punch velocity on the compression characteristics of one-step dry-coated tablets (OSDRC). J. Pharm. Sci Technol. Japan. 64:67-73 (2004).
27. J. J. Wang, M. A. Guillot, S. D. Bateman, and K. R. Morris. Modeling of adhesion in tablet compression. 2. Compaction studies using a compaction simulator and an instrumented tablet press. J. Pharm. Sci. 93:407-417 (2004).
28. M. Otsuka, M. Sato, and Y. Matsuda. Comparative evaluation of tableting compression behaviors by methods of internal and external lubricant addition: inhibition of enzymatic activity of trypsin preparation by using external lubricant addition during the tableting compression process. AAPS PharmSci. 3:E20 (2001).
29. Y. Ozeki, Y. Watanabe, S. Inoue, and K. Danjo. Comparison of the compression characteristics between new one-step dry-coated tablets (OSDRC) and dry-coated tablets (DC). Int. J. Pharm. 259:69-77 (2003).
30. T. Cutt, J. T. Fell, P. J. Rue, and M. S. Spring. Granulation and compaction of a model system 2. Stress relaxation. Int. J. Pharm. 39:157-161 (1987).
31. A. Nokhodchi, J. L. Ford, P. H. Rowe, and M. H. Rubinstein. The effect of compression rate and force on the compaction properties of different viscosity grades of hydroxypropylmethylcellulose 2208. Int. J. Pharm. 129:21-31 (1996).
32. Y. Ozeki, Y. Watanabe, S. Inoue, and K. Danjo. Evaluation of the compression characteristics and physical properties of the newly invented one-step dry-coated tablets. Int. J. Pharm. 267:69-78 (2003).