Auto-modulation of neuroactive steroids on GABAA receptors: A novel pharmacological effect

Neuropharmacology

Volumn 52, Issue 2, 2007, Pages 672-683

  Wegner, Florian ^a   Rassler, Cornelia ^a   Allgaier, Clemens ^a   Strecker, Karl ^a   Wohlfarth, Kai ^a  

^a UNIVERSITY OF LEIPZIG   (Germany)

Author keywords

Alphaxalone; Auto modulation; Electrophysiology; GABAA receptor; Neuroactive steroid; Phosphorylation

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; ALFAXALONE; CYCLIC AMP DEPENDENT PROTEIN KINASE; INDIPLON; NEUROSTEROID; PENTOBARBITAL;

ALLOSTERISM; ARTICLE; CELL STRAIN HEK293; CONCENTRATION RESPONSE; CONTROLLED STUDY; HUMAN; HUMAN CELL; NEUROMODULATION; PATCH CLAMP; PHOSPHORYLATION; PRIORITY JOURNAL; SYNAPTIC INHIBITION;

CELL LINE; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG INTERACTIONS; ENZYME INHIBITORS; GABA AGONISTS; GAMMA-AMINOBUTYRIC ACID; GENE EXPRESSION; HUMANS; ISOXAZOLES; MEMBRANE POTENTIALS; PATCH-CLAMP TECHNIQUES; PREGNANEDIONES; PROTEIN SUBUNITS; RECEPTORS, GABA-A; RECOMBINANT PROTEINS; STEROIDS;

EID: 33846441234     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2006.09.009     Document Type: Article

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