Inhibitory effect of 4-(2-aminoethyl)-benzenesulfonyl fluoride, a serine protease inhibitor, on PI3K inhibitor-induced CHOP expression

European Journal of Pharmacology

Volumn 554, Issue 1, 2007, Pages 8-11

  Hosoi, Toru ^a   Hyoda, Kanae ^b   Okuma, Yasunobu ^c   Nomura, Yasuyuki ^b,d   Ozawa, Koichiro ^a  

^a HIROSHIMA UNIVERSITY   (Japan)

^b HOKKAIDO UNIVERSITY   (Japan)

^c CHIBA INSTITUTE OF SCIENCE   (Japan)

^d YOKOHAMA COLLEGE OF PHARMACY   (Japan)

Author keywords

4 (2 Aminoethyl) benzenesulfonyl fluoride (AEBSF); CHOP; Endoplasmic reticulum stress; Phosphatidylinositol 3 kinase (PI3K)

Indexed keywords

4 (2 AMINOETHYL) BENZENESULFONYL FLUORIDE; GROWTH ARREST AND DNA DAMAGE INDUCIBLE PROTEIN 153; MESSENGER RNA; PHOSPHATIDYLINOSITOL 3 KINASE INHIBITOR; SERINE PROTEINASE INHIBITOR; TRANSCRIPTION FACTOR;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG EFFECT; DRUG MECHANISM; ENDOPLASMIC RETICULUM; INHIBITION KINETICS; MOUSE; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION;

1-PHOSPHATIDYLINOSITOL 3-KINASE; ANIMALS; CELLS, CULTURED; ENDOPLASMIC RETICULUM; GENE EXPRESSION REGULATION; MICE; RNA, MESSENGER; SERINE ENDOPEPTIDASES; SERINE PROTEINASE INHIBITORS; SULFONES; TRANSCRIPTION FACTOR CHOP;

EID: 33751417807     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2006.09.063     Document Type: Article

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