Facile synthesis of non-steroidal anti-inflammatory active bisbenzamide-containing compounds

Bioorganic and Medicinal Chemistry

Volumn 14, Issue 24, 2006, Pages 8527-8532

  Girgis, Adel S ^a   Ellithey, Mohey ^a  

^a NATIONAL RESEARCH CENTRE   (Egypt)

Author keywords

Anti inflammatory; Bisbenzaldehydes; Bisbenzamides; Bisoxazol 5(4H) ones

Indexed keywords

4,4' [1,2 ETHANEDIYLBIS(OXY 2,1 PHENYLENEMETHYLIDENE)]BIS(2 PHENYL 5(4H)OXAZOLONE); BENZAMIDE DERIVATIVE; BIS[1 [[(4 CHLOROPHENYL)AMINO]CARBONYL] 2[1,2 ETHANEDIYLBIS(OXY 2,1 PHENYLENE)]ETHENYL]BENZAMIDE; BIS[2 [1,2 ETHANEDIYLBIS(OXY 2,1 PHENYLENE)1 [[1 (4 METHYLPIPERAZINYL)] CARBONYL]ETHENYL]BENZAMIDE; BIS[2 [1,2 ETHANEDIYLBIS(OXY 2,1 PHENYLENE)] 1 [(1 PIPERIDINYL)CARBONYL] ETHENYL]BENZAMIDE; BIS[2 [1,2 ETHANEDIYLBIS(OXY 2,1 PHENYLENE)] 1 [(4 MORPHOLINYL)CARBONYL] ETHENYL]BENZAMIDE; BIS[2 [1,2 ETHANEDIYLBIS(OXY 2,1 PHENYLENE)] 1 [(PHENYLAMINO)CARBONYL] ETHENYL]BENZAMIDE; BIS[2 [1,2 ETHANEDIYLBIS(OXY 2,1 PHENYLENE)] 1 [[(4 METHOXYPHENYL)AMINO] CARBONYL]ETHENYL]BENZAMIDE; BIS[2 [1,2 ETHANEDIYLBIS(OXY 2,1 PHENYLENE)] [[(4 METHYLPHENYL)AMINO] CARBONYL]ETHENYL]BENZAMIDE; KETOPROFEN; NONSTEROID ANTIINFLAMMATORY AGENT; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; IN VIVO STUDY; NONHUMAN; PAW EDEMA; RAT;

ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; BENZAMIDES; CARRAGEENAN; EDEMA; FEMALE; FOOT; MOLECULAR STRUCTURE; RATS; RATS, WISTAR; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33750496596     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2006.08.032     Document Type: Article

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