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Volumn 16, Issue 19, 2006, Pages 5217-5221
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From arylureas to biarylamides to aminoquinazolines: Discovery of a novel, potent TRPV1 antagonist
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Author keywords
Antagonist; Bioisostere; Pain; Quinazoline; TRPV1; Ureas; VR1
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Indexed keywords
AROMATIC AMIDE;
QUINAZOLINE DERIVATIVE;
RECEPTOR BLOCKING AGENT;
UNCLASSIFIED DRUG;
UREA DERIVATIVE;
VANILLOID RECEPTOR 1;
VANILLOID RECEPTOR 1 ANTAGONIST;
ANIMAL EXPERIMENT;
ARTICLE;
CONFORMATION;
CONTROLLED STUDY;
DRUG BIOAVAILABILITY;
DRUG POTENCY;
NONHUMAN;
RAT;
STRUCTURE ACTIVITY RELATION;
ADMINISTRATION, ORAL;
AMIDES;
ANALGESICS, NON-NARCOTIC;
ANIMALS;
BIOLOGICAL AVAILABILITY;
HUMANS;
MOLECULAR CONFORMATION;
PAIN;
QUINAZOLINES;
RATS;
SOLUBILITY;
STRUCTURE-ACTIVITY RELATIONSHIP;
TRPV CATION CHANNELS;
UREA;
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EID: 33747375663
PISSN: 0960894X
EISSN: None
Source Type: Journal
DOI: 10.1016/j.bmcl.2006.07.010 Document Type: Article |
Times cited : (33)
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References (15)
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