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Volumn 1, Issue 3, 2006, Pages 358-365

Synthesis and preliminary biological evaluation of 2′-substituted 2-(3′-carboxybicyclo[1.1.1]-pentyl)glycine derivatives as group I selective metabotropic glutamate receptor ligands

(12) Pellicciari, Roberto a Filosa, Rosanna a Fulco, Maria Carmela a Marinozzi, Maura a Macchiarulo, Antonio a Novak, Clemens a,c Natalini, Benedetto a Hermit, Mette Brunsgaard b Nielsen, Søren b Sager, Thomas Nikolaj b Stensbøl, Tine Bryan b Thomsen, Christian b

a UNIVERSITY OF PERUGIA (Italy)

b H LUNDBECK A S (Denmark)

c UNIVERSITY OF VIENNA (Austria)

Author keywords

Bicyclo 1.1.1 pentane; Group I mGluR antagonists; Neurochemistry; Polycycles; Receptors

Indexed keywords

BICYCLO COMPOUND; DRUG DERIVATIVE; GLYCINE; LIGAND; METABOTROPIC RECEPTOR; UPF 596;

ARTICLE; CHEMICAL STRUCTURE; DRUG EFFECT; METABOLISM; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

BICYCLO COMPOUNDS; GLYCINE; LIGANDS; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, MOLECULAR; RECEPTORS, METABOTROPIC GLUTAMATE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33646530328 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200500071 Document Type: Article

Times cited : (25)

References (28)

1
- 0030995878
- P. J. Conn, J.-P. Pin, Annu. Rev. Pharmacol. Toxicol. 1997, 37, 205-237.
- (1997) Annu. Rev. Pharmacol. Toxicol. , vol.37 , pp. 205-237
- Conn, P.J.¹ Pin, J.-P.²

2
- 0032907608
- R. Anwyl, Brain Res. Rev. 1999, 29, 83-120.
- (1999) Brain Res. Rev. , vol.29 , pp. 83-120
- Anwyl, R.¹

3
- 0037832971
- H. Bräuner-Osborne, J. Egebjerg, E. Ø. Nielsen, U. Madsen, P. Krogsgaard-Larsen, J. Med. Chem. 2000, 43, 2609-2645.
- (2000) J. Med. Chem. , vol.43 , pp. 2609-2645
- Bräuner-Osborne, H.¹ Egebjerg, J.² Nielsen, E.Ø.³ Madsen, U.⁴ Krogsgaard-Larsen, P.⁵

4
- 12444302830
- G. Costantino, A. Macchiarulo, R. Pellicciari, Expert Opin. Ther. Targets 2001, 5, 669-683.
- (2001) Expert Opin. Ther. Targets , vol.5 , pp. 669-683
- Costantino, G.¹ Macchiarulo, A.² Pellicciari, R.³

5
- 0001050064
- M. A. Varney, R. W. Gereau, Curr. Drug Targets: CNS Neurol. Disord. 2002, 1, 283-296.
- (2002) Curr. Drug Targets: CNS Neurol. Disord. , vol.1 , pp. 283-296
- Varney, M.A.¹ Gereau, R.W.²

6
- 0042868860
- W. Spooren, T. Ballard, F. Gasparini, M. Amalric, V. Mutel, R. Schreiber, Behav. Pharmacol. 2003, 14, 257-277.
- (2003) Behav. Pharmacol. , vol.14 , pp. 257-277
- Spooren, W.¹ Ballard, T.² Gasparini, F.³ Amalric, M.⁴ Mutel, V.⁵ Schreiber, R.⁶

7
- 0012662271
- J. Doherty, R. Dingledine, Curr. Drug Targets: CNS Neurol. Disord. 2002, 1, 251-260.
- (2002) Curr. Drug Targets: CNS Neurol. Disord. , vol.1 , pp. 251-260
- Doherty, J.¹ Dingledine, R.²

8
- 8844263762
- J. N. C. Kew, Pharmacol. Ther. 2004, 104, 233-244.
- (2004) Pharmacol. Ther. , vol.104 , pp. 233-244
- Kew, J.N.C.¹

9
- 0027448332
- S. A. Eaton, D. E. Jane, P. L. Jones, R. H. Porter, P. C. Pook, D. C. Sunter, P. M. Udvarhelyi, P. T. Roberts, J. C. Watkins, Eur. J. Pharmacol. 1993, 244, 195-197.
- (1993) Eur. J. Pharmacol. , vol.244 , pp. 195-197
- Eaton, S.A.¹ Jane, D.E.² Jones, P.L.³ Porter, R.H.⁴ Pook, P.C.⁵ Sunter, D.C.⁶ Udvarhelyi, P.M.⁷ Roberts, P.T.⁸ Watkins, J.C.⁹

10
- 0029126126
- a) R. Pellicciari, R. Luneia, G. Costantino, M. Marinozzi, B. Natalini, P. Jakobsen, A. Kanstrup, G. Lombardi, F. Moroni, C. Thomsen, J. Med. Chem. 1995, 38, 3717-3719;
- (1995) J. Med. Chem. , vol.38 , pp. 3717-3719
- Pellicciari, R.¹ Luneia, R.² Costantino, G.³ Marinozzi, M.⁴ Natalini, B.⁵ Jakobsen, P.⁶ Kanstrup, A.⁷ Lombardi, G.⁸ Moroni, F.⁹ Thomsen, C.¹⁰

11
- 1942476154
- b) B. Natalini, M. Marinozzi, K. Bade, R. Sardella, C. Thomsen, R. Pellicciari, Chirality 2004, 16, 314-317;
- (2004) Chirality , vol.16 , pp. 314-317
- Natalini, B.¹ Marinozzi, M.² Bade, K.³ Sardella, R.⁴ Thomsen, C.⁵ Pellicciari, R.⁶

12
- 0037363728
- c) J. M. Mathiesen, N. Svendsen, H. Bräuner-Osborne, C. Thomsen, M. T. Ramirez, Br. J. Pharmacol. 2003, 138, 1026-1030.
- (2003) Br. J. Pharmacol. , vol.138 , pp. 1026-1030
- Mathiesen, J.M.¹ Svendsen, N.² Bräuner-Osborne, H.³ Thomsen, C.⁴ Ramirez, M.T.⁵

13
- 0032885411
- D. E. Pellegrini-Giampietro, F. Peruginelli, E. Meli, A. Cozzi, S. Albani-Torregrossa, R. Pellicciari, F. Moroni, Neuropharmacology 1999, 38, 1607-1619.
- (1999) Neuropharmacology , vol.38 , pp. 1607-1619
- Pellegrini-Giampietro, D.E.¹ Peruginelli, F.² Meli, E.³ Cozzi, A.⁴ Albani-Torregrossa, S.⁵ Pellicciari, R.⁶ Moroni, F.⁷

14
- 0030014882
- R. Pellicciari, M. Raimondo, M. Marinozzi, B. Natalini, G. Costantino, C. Thomsen, J. Med. Chem. 1996, 39, 2874-2876.
- (1996) J. Med. Chem. , vol.39 , pp. 2874-2876
- Pellicciari, R.¹ Raimondo, M.² Marinozzi, M.³ Natalini, B.⁴ Costantino, G.⁵ Thomsen, C.⁶

15
- 0032537619
- R. Pellicciari, G. Costantino, E. Giovagnoni, L. Mattoli, I. Brabet, J.-P. Pin, Bioorg. Med. Chem. Lett. 1998, 8, 1569-1573.
- (1998) Bioorg. Med. Chem. Lett. , vol.8 , pp. 1569-1573
- Pellicciari, R.¹ Costantino, G.² Giovagnoni, E.³ Mattoli, L.⁴ Brabet, I.⁵ Pin, J.-P.⁶

16
- 0033006689
- G. Mannaioni, S. Attucci, A. Missanelli, R. Pellicciari, R. Corradetti, F. Moroni, Neuropharmacology 1999, 38, 917-926.
- (1999) Neuropharmacology , vol.38 , pp. 917-926
- Mannaioni, G.¹ Attucci, S.² Missanelli, A.³ Pellicciari, R.⁴ Corradetti, R.⁵ Moroni, F.⁶

17
- 0035080723
- G. Costantino, K. Maltoni, M. Marinozzi, E. Camaioni, L. Prezeau, J.-P. Pin, R. Pellicciari, Bioorg. Med. Chem. 2001, 9, 221-227.
- (2001) Bioorg. Med. Chem. , vol.9 , pp. 221-227
- Costantino, G.¹ Maltoni, K.² Marinozzi, M.³ Camaioni, E.⁴ Prezeau, L.⁵ Pin, J.-P.⁶ Pellicciari, R.⁷

18
- 0000741608
- and references therein
- M. D. Levin, P. Kaszynski, J. Michl, Chem. Rev. 2000, 100, 169-234, and references therein.
- (2000) Chem. Rev. , vol.100 , pp. 169-234
- Levin, M.D.¹ Kaszynski, P.² Michl, J.³

19
- 0003695886
- R. E. Robinson, J. Michl, J. Org. Chem. 1989, 54, 2051-2053.
- (1989) J. Org. Chem. , vol.54 , pp. 2051-2053
- Robinson, R.E.¹ Michl, J.²

20
- 0001020947
- P. Kaszynski, J. Michl, J. Org. Chem. 1988, 53, 4593-4594.
- (1988) J. Org. Chem. , vol.53 , pp. 4593-4594
- Kaszynski, P.¹ Michl, J.²

21
- 12644312578
- A. J. Mancuso, S.-L Huang, D. Swern, J. Org. Chem. 1978, 43, 2480-2482.
- (1978) J. Org. Chem. , vol.43 , pp. 2480-2482
- Mancuso, A.J.¹ Huang, S.-L.² Swern, D.³

22
- 0029164282
- T. K. Chakraborty, K. A. Hussian, G. V. Reddy, Tetrahedron 1995, 51, 9179-9190.
- (1995) Tetrahedron , vol.51 , pp. 9179-9190
- Chakraborty, T.K.¹ Hussian, K.A.² Reddy, G.V.³

23
- 0029956082
- R. Pellicciari, M. Marinozzi, B. Natalini, G. Costantino, R. Luneia, G. Giorgi, F. Moroni, C. Thomsen, J. Med. Chem. 1996, 39, 2259-2269.
- (1996) J. Med. Chem. , vol.39 , pp. 2259-2269
- Pellicciari, R.¹ Marinozzi, M.² Natalini, B.³ Costantino, G.⁴ Luneia, R.⁵ Giorgi, G.⁶ Moroni, F.⁷ Thomsen, C.⁸

24
- 0001044552
- M. Ballestri, C. Chatgilialoglu, K. B. Clark, D. Griller, B. Giese, B. Kopping, J. Org. Chem. 1991, 56, 678-683.
- (1991) J. Org. Chem. , vol.56 , pp. 678-683
- Ballestri, M.¹ Chatgilialoglu, C.² Clark, K.B.³ Griller, D.⁴ Giese, B.⁵ Kopping, B.⁶

25
- 11644261806
- G. M. Morris, D. S. Goodsell, R. S. Halliday, R. Huey, W. E. Hart, R. K. Belew, A. J. Olson, J. Comput. Chem. 1998, 19, 1639-1662.
- (1998) J. Comput. Chem. , vol.19 , pp. 1639-1662
- Morris, G.M.¹ Goodsell, D.S.² Halliday, R.S.³ Huey, R.⁴ Hart, W.E.⁵ Belew, R.K.⁶ Olson, A.J.⁷

26
- 33646500074
- Accelrys, San Diego, CA
- Cerius-2, Accelrys, San Diego, CA.
- Cerius-2

27
- 0042041206
- A. K. Rappe, C. J. Casewit, K. S. Colwell, W. A. Goddard, W. M. Skiff, J. Am. Chem. Soc. 1992, 114, 10024-10035.
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 10024-10035
- Rappe, A.K.¹ Casewit, C.J.² Colwell, K.S.³ Goddard, W.A.⁴ Skiff, W.M.⁵

28
- 0027495614
- K. G. Steppuhn, L. Turski, J. Pharmacol. Exp. Ther. 1993, 265, 1063-1070.
- (1993) J. Pharmacol. Exp. Ther. , vol.265 , pp. 1063-1070
- Steppuhn, K.G.¹ Turski, L.²

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