Biochemical and electrophysiological studies on (S)-(+)-2-(3'-carboxybicyclo[1.1.1]pentyl)-glycine (CBPG), a novel mGlu5 receptor agonist endowed with mGlu1 receptor antagonist activity

Neuropharmacology

Volumn 38, Issue 7, 1999, Pages 917-926

  Mannaioni, Guido ^a   Attucci, Sabina ^a   Missanelli, Andrea ^a   Pellicciari, Roberto ^b   Corradetti, Renato ^a   Moroni, Flavio ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

^b UNIVERSITY OF PERUGIA   (Italy)

Author keywords

(RS) 1 aminoindan 1,5 dicarboxylic acid (AIDA); (RS) 2 chloro 5 hydroxyphenylglycine (CHPG); (S) (+) 2 (3' carboxybicyclo 1.1.1 pentyl) glycine (CBPG); (S) 3,5 dihydroxyphenylglycine (DHPG); Hippocampus; mGluR

Indexed keywords

1 AMINO 1,5 INDANDICARBOXYLIC ACID; 2 (3 CARBOXYBICYCLO[1.1.1]PENTYL)GLYCINE; 2 CHLORO 5 HYDROXYPHENYLGLYCINE; 3,5 DIHYDROXYPHENYLGLYCINE; ALPHA AMINO 3 HYDROXY 5 METHYL 4 ISOXAZOLEPROPIONIC ACID; CYCLIC AMP; GLUTAMATE RECEPTOR; METABOTROPIC RECEPTOR; N METHYL DEXTRO ASPARTIC ACID; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BRAIN SLICE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DEPOLARIZATION; HIPPOCAMPUS; MALE; NERVE POTENTIAL; NEUROTRANSMISSION; NONHUMAN; PRIORITY JOURNAL; PYRAMIDAL NERVE CELL; RAT; SECOND MESSENGER;

ANIMALS; BICYCLO COMPOUNDS; BRAIN; CELL MEMBRANE; CELLS, CULTURED; CRICETINAE; ELECTROPHYSIOLOGY; EXCITATORY AMINO ACID ANTAGONISTS; GLYCINE; MALE; METHOXYHYDROXYPHENYLGLYCOL; NEURONS; PHENYLACETATES; PYRAMIDAL TRACTS; RATS; RATS, WISTAR; RECEPTORS, METABOTROPIC GLUTAMATE; SECOND MESSENGER SYSTEMS; TRANSFECTION;

EID: 0033006689     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(99)00021-0     Document Type: Article

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