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Volumn 62, Issue 3, 2006, Pages 241-246

Influence of cyclodextrins and chitosan, separately or in combination, on glyburide solubility and permeability

Author keywords

Caco 2 cells; Chitosan; Cyclodextrins; Glyburide; Permeability; Solubility

Indexed keywords

CHITOSAN; CYCLODEXTRIN DERIVATIVE; GLIBENCLAMIDE; MACROCYCLIC COMPOUND;

EID: 33644827423     PISSN: 09396411     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejpb.2005.08.010     Document Type: Article
Times cited : (53)

References (47)
  • 2
    • 0022909293 scopus 로고
    • Correlations between in vitro dissolution, in vivo bioavailability and hypoglycaemic effect of oral glibenclamide
    • J.B. Chalk, M. Patterson, M.T. Smith, and M.J. Eadie Correlations between in vitro dissolution, in vivo bioavailability and hypoglycaemic effect of oral glibenclamide Eur. J. Clin. Pharmacol. 31 1986 177 182
    • (1986) Eur. J. Clin. Pharmacol. , vol.31 , pp. 177-182
    • Chalk, J.B.1    Patterson, M.2    Smith, M.T.3    Eadie, M.J.4
  • 3
    • 0027772495 scopus 로고
    • Pharmaceutical quality of glibenclamide products: A multinational postmarket comparative study
    • H. Blume, S.L. Ali, and M. Siewert Pharmaceutical quality of glibenclamide products: a multinational postmarket comparative study Drug Dev. Ind. Pharm. 19 1993 2713 2741
    • (1993) Drug Dev. Ind. Pharm. , vol.19 , pp. 2713-2741
    • Blume, H.1    Ali, S.L.2    Siewert, M.3
  • 4
    • 3042618323 scopus 로고    scopus 로고
    • Deactivation of amorphous glibenclamide during dissolution
    • D. Cordes, and B.W. Müller Deactivation of amorphous glibenclamide during dissolution Eur. J. Pharm. Sci. 4 1996 S187 P3.087
    • (1996) Eur. J. Pharm. Sci. , vol.4 , pp. 187
    • Cordes, D.1    Müller, B.W.2
  • 5
    • 0030016875 scopus 로고    scopus 로고
    • Characterization of glyburide polyethylene glycol solid dispersions
    • G.V. Bertageri, and K.R. Makarla Characterization of glyburide polyethylene glycol solid dispersions Drug Dev. Ind. Pharm. 22 1996 731 734
    • (1996) Drug Dev. Ind. Pharm. , vol.22 , pp. 731-734
    • Bertageri, G.V.1    Makarla, K.R.2
  • 6
    • 0029820163 scopus 로고    scopus 로고
    • Dissolution properties of glibenclamide in combinations with polyvinylpyrrolidone
    • M. Iwata, and H. Ueda Dissolution properties of glibenclamide in combinations with polyvinylpyrrolidone Drug Dev. Ind. Pharm. 22 1996 1161 1165
    • (1996) Drug Dev. Ind. Pharm. , vol.22 , pp. 1161-1165
    • Iwata, M.1    Ueda, H.2
  • 7
    • 0028280539 scopus 로고
    • Solubilization of glibenclamide with β-cyclodextrin and its derivatives
    • N.M. Sanghavi, H. Venkatesh, and V. Tandel Solubilization of glibenclamide with β-cyclodextrin and its derivatives Drug Dev. Ind. Pharm. 20 1994 1275 1283
    • (1994) Drug Dev. Ind. Pharm. , vol.20 , pp. 1275-1283
    • Sanghavi, N.M.1    Venkatesh, H.2    Tandel, V.3
  • 8
    • 3042550643 scopus 로고    scopus 로고
    • Development and evaluation of glyburide fast dissolving tablets using solid dispersion technique
    • M. Valleri, P. Mura, F. Maestrelli, M. Cirri, and R. Ballerini Development and evaluation of glyburide fast dissolving tablets using solid dispersion technique Drug Dev. Ind. Pharm. 30 2004 525 534
    • (2004) Drug Dev. Ind. Pharm. , vol.30 , pp. 525-534
    • Valleri, M.1    Mura, P.2    Maestrelli, F.3    Cirri, M.4    Ballerini, R.5
  • 9
    • 0029072198 scopus 로고
    • Enhancement of dissolution rate and hypoglicemic activity of glibenclamide with β-cyclodextrin
    • R.J. Babu, and K.J. Pandit Enhancement of dissolution rate and hypoglicemic activity of glibenclamide with β-cyclodextrin S.T.P. Pharma Sci. 5 1995 196 200
    • (1995) S.T.P. Pharma Sci. , vol.5 , pp. 196-200
    • Babu, R.J.1    Pandit, K.J.2
  • 10
    • 0031786697 scopus 로고    scopus 로고
    • Co-administration of a water-soluble polymer increases the usefulness of cyclodextrins in solid oral dosage forms
    • J. Savolainen, K. Jarvinen, H. Taipale, P. Jarho, T. Loftsson, and T. Jarvinen Co-administration of a water-soluble polymer increases the usefulness of cyclodextrins in solid oral dosage forms Pharm. Res. 15 1998 1696 1701
    • (1998) Pharm. Res. , vol.15 , pp. 1696-1701
    • Savolainen, J.1    Jarvinen, K.2    Taipale, H.3    Jarho, P.4    Loftsson, T.5    Jarvinen, T.6
  • 11
    • 0031783879 scopus 로고    scopus 로고
    • Chitosan and its use as a pharmaceutical excipient
    • L. Illum Chitosan and its use as a pharmaceutical excipient Pharm. Res. 15 1998 1326 1331
    • (1998) Pharm. Res. , vol.15 , pp. 1326-1331
    • Illum, L.1
  • 12
    • 0031714427 scopus 로고    scopus 로고
    • Chitosan: A unique polysaccharide for drug delivery
    • O. Felt, P. Buri, and R. Gurny Chitosan: a unique polysaccharide for drug delivery Drug Dev. Ind. Pharm. 24 1998 979 993
    • (1998) Drug Dev. Ind. Pharm. , vol.24 , pp. 979-993
    • Felt, O.1    Buri, P.2    Gurny, R.3
  • 13
    • 0034005095 scopus 로고    scopus 로고
    • Chitosan, a drug carrier for the 21th century
    • W. Paul, and C.P. Sharma Chitosan, a drug carrier for the 21th century S.T.P. Pharma Sci. 10 2000 5 22
    • (2000) S.T.P. Pharma Sci. , vol.10 , pp. 5-22
    • Paul, W.1    Sharma, C.P.2
  • 14
    • 0025215648 scopus 로고
    • Enhancement of dissolution rates of several drugs by low molecular chitosan and alginate
    • S. Shiraishi, M. Arahira, T. Imai, and M. Otagiri Enhancement of dissolution rates of several drugs by low molecular chitosan and alginate Chem. Pharm. Bull. 38 1990 185 187
    • (1990) Chem. Pharm. Bull. , vol.38 , pp. 185-187
    • Shiraishi, S.1    Arahira, M.2    Imai, T.3    Otagiri, M.4
  • 15
    • 0345195980 scopus 로고    scopus 로고
    • Effect of chitosan and chitosan glutamate enhancing the dissolution properties of the poorly water soluble drug nifedipine
    • A. Portero, C. Remuñan-Lopez, and J.L. Vila-Jato Effect of chitosan and chitosan glutamate enhancing the dissolution properties of the poorly water soluble drug nifedipine Int. J. Pharm. 175 1998 75 84
    • (1998) Int. J. Pharm. , vol.175 , pp. 75-84
    • Portero, A.1    Remuñan-Lopez, C.2    Vila-Jato, J.L.3
  • 16
    • 0344281695 scopus 로고    scopus 로고
    • Development and characterization of naproxen-chitosan solid systems with improved drug dissolution properties
    • P. Mura, N. Zerrouk, N. Mennini, F. Maestrelli, and C. Chemtob Development and characterization of naproxen-chitosan solid systems with improved drug dissolution properties Eur. J. Pharm. Sci. 19 2003 67 75
    • (2003) Eur. J. Pharm. Sci. , vol.19 , pp. 67-75
    • Mura, P.1    Zerrouk, N.2    Mennini, N.3    Maestrelli, F.4    Chemtob, C.5
  • 17
    • 0346094166 scopus 로고    scopus 로고
    • Comparison of the effect of chitosan and polyvynilpyrrolidone on dissolution properties and analgesic effect of naproxen, Eur
    • N. Zerrouk, N. Mennini, F. Maestrelli, C. Chemtob, and P. Mura Comparison of the effect of chitosan and polyvynilpyrrolidone on dissolution properties and analgesic effect of naproxen, Eur J. Pharm. Biopharm. 57 2004 93 99
    • (2004) J. Pharm. Biopharm. , vol.57 , pp. 93-99
    • Zerrouk, N.1    Mennini, N.2    Maestrelli, F.3    Chemtob, C.4    Mura, P.5
  • 19
    • 0032119526 scopus 로고    scopus 로고
    • Cyclodextrin drug carrier systems
    • K. Uekama, F. Hirayama, and I. Tetsumi Cyclodextrin drug carrier systems Chem. Rev. 98 1998 2045 2076
    • (1998) Chem. Rev. , vol.98 , pp. 2045-2076
    • Uekama, K.1    Hirayama, F.2    Tetsumi, I.3
  • 20
    • 0141701162 scopus 로고    scopus 로고
    • Cyclodextrins as permeation enhancers: Some theoretical evaluations and in vitro testing
    • M. Másson, T. Loftsson, G. Másson, and E. Stefánsson Cyclodextrins as permeation enhancers: some theoretical evaluations and in vitro testing J. Control. Rel. 59 1999 107 118
    • (1999) J. Control. Rel. , vol.59 , pp. 107-118
    • Másson, M.1    Loftsson, T.2    Másson, G.3    Stefánsson, E.4
  • 21
    • 0033105151 scopus 로고    scopus 로고
    • Cyclodextrins in peptide and protein delivery
    • T. Irie, and K. Uekama Cyclodextrins in peptide and protein delivery Adv. Drug Del. Rev. 36 1999 101 123
    • (1999) Adv. Drug Del. Rev. , vol.36 , pp. 101-123
    • Irie, T.1    Uekama, K.2
  • 22
    • 0033106031 scopus 로고    scopus 로고
    • Cyclodextrins in transdermal and rectal delivery
    • H. Matsuda, and H. Arima Cyclodextrins in transdermal and rectal delivery Adv. Drug Del. Rev. 36 1999 81 99
    • (1999) Adv. Drug Del. Rev. , vol.36 , pp. 81-99
    • Matsuda, H.1    Arima, H.2
  • 24
    • 0021984043 scopus 로고
    • Selective transfer of 1-hexylcarbamoyl-5-fluorouracil into lymphatics by combination of β-cyclodextrin polymer complexation and absorption promotor in the rat
    • Y. Kaji, K. Uekama, H. Yoshikawa, K. Takada, and S. Muranishi Selective transfer of 1-hexylcarbamoyl-5-fluorouracil into lymphatics by combination of β-cyclodextrin polymer complexation and absorption promotor in the rat Int. J. Pharm. 24 1985 79 89
    • (1985) Int. J. Pharm. , vol.24 , pp. 79-89
    • Kaji, Y.1    Uekama, K.2    Yoshikawa, H.3    Takada, K.4    Muranishi, S.5
  • 25
    • 0029556984 scopus 로고
    • Modification of rectal absorption of morphine from suppositories with a combination of α-cyclodextrin and viscosity-enhancing polymer
    • K. Uekama, T. Kondo, and K. Nakamura Modification of rectal absorption of morphine from suppositories with a combination of α-cyclodextrin and viscosity-enhancing polymer J. Pharm. Sci. 84 1995 15 20
    • (1995) J. Pharm. Sci. , vol.84 , pp. 15-20
    • Uekama, K.1    Kondo, T.2    Nakamura, K.3
  • 26
    • 0024989124 scopus 로고
    • Effect of β-cyclodextrin on the in-vitro permeation rate and in-vivo rectal absorption of acetaminophen hydrogel preparations
    • S.Y. Lin, and J.C. Yang Effect of β-cyclodextrin on the in-vitro permeation rate and in-vivo rectal absorption of acetaminophen hydrogel preparations Pharm Acta Helv. 65 1990 262 268
    • (1990) Pharm Acta Helv. , vol.65 , pp. 262-268
    • Lin, S.Y.1    Yang, J.C.2
  • 27
    • 0026321138 scopus 로고
    • Cell culture as models for drug absorption across the intestinal mucosa
    • P. Artursson Cell culture as models for drug absorption across the intestinal mucosa Crit. Rev. Ther. Drug Carrier Syst. 8 1991 105 130
    • (1991) Crit. Rev. Ther. Drug Carrier Syst. , vol.8 , pp. 105-130
    • Artursson, P.1
  • 28
    • 0030023536 scopus 로고    scopus 로고
    • Comparison between active and passive drug transport in human intestinal epithelial (Caco-2) cells in vitro and human jejunum in vivo
    • H. Lennernäs, K. Palm, U. Fagerholm, and P. Artusson Comparison between active and passive drug transport in human intestinal epithelial (Caco-2) cells in vitro and human jejunum in vivo Int. J. Pharm. 127 1996 103 107
    • (1996) Int. J. Pharm. , vol.127 , pp. 103-107
    • Lennernäs, H.1    Palm, K.2    Fagerholm, U.3    Artusson, P.4
  • 29
    • 0031574261 scopus 로고    scopus 로고
    • Chitosans for enhanced delivery of therapeutics peptides across intestinal epithelia: In vitro evaluation in Caco-2 cell monolayers
    • A.F. Kotzé, B.J. de Leeuw, H.L. Lueßen, A.G. de Boer, J.C. Verhoef, and H.E. Junginger Chitosans for enhanced delivery of therapeutics peptides across intestinal epithelia: in vitro evaluation in Caco-2 cell monolayers Int. J. Pharm. 159 1997 243 253
    • (1997) Int. J. Pharm. , vol.159 , pp. 243-253
    • Kotzé, A.F.1    De Leeuw, B.J.2    Lueßen, H.L.3    De Boer, A.G.4    Verhoef, J.C.5    Junginger, H.E.6
  • 30
    • 0031742986 scopus 로고    scopus 로고
    • Link between drug absorption solubility and permeability measurements in Caco-2 cells
    • V. Pade, and S. Stavchansky Link between drug absorption solubility and permeability measurements in Caco-2 cells J. Pharm. Sci. 87 1998 1604 1607
    • (1998) J. Pharm. Sci. , vol.87 , pp. 1604-1607
    • Pade, V.1    Stavchansky, S.2
  • 31
    • 0343150936 scopus 로고    scopus 로고
    • The potential of mucoadhesive polymer in enhancing intestinal peptide drug absorption. III. Effect of chitosan-glutamate and carbomer on epithelial tight junctions in vitro
    • G. Borchard, H.L. Lueßen, A.G. de Boer, J.C. Verhoef, C. Lehr, and H.E. Junginger The potential of mucoadhesive polymer in enhancing intestinal peptide drug absorption. III. Effect of chitosan-glutamate and carbomer on epithelial tight junctions in vitro J. Control. Rel. 39 1996 131 138
    • (1996) J. Control. Rel. , vol.39 , pp. 131-138
    • Borchard, G.1    Lueßen, H.L.2    De Boer, A.G.3    Verhoef, J.C.4    Lehr, C.5    Junginger, H.E.6
  • 32
    • 0021038289 scopus 로고
    • An enzyme-release assay for natural cytotoxicity
    • C. Korzeniewski, and D.M. Callewaert An enzyme-release assay for natural cytotoxicity J. Immunol. Methods 64 1983 313 320
    • (1983) J. Immunol. Methods , vol.64 , pp. 313-320
    • Korzeniewski, C.1    Callewaert, D.M.2
  • 33
    • 0343036151 scopus 로고    scopus 로고
    • Corrections to the original LDH release assay for the evaluation of NK cell cytotoxicity
    • G. Konjevic, V. Jurisic, and I. Spuzic Corrections to the original LDH release assay for the evaluation of NK cell cytotoxicity J. Immunol. Methods 200 1997 199 201
    • (1997) J. Immunol. Methods , vol.200 , pp. 199-201
    • Konjevic, G.1    Jurisic, V.2    Spuzic, I.3
  • 35
    • 0032543172 scopus 로고    scopus 로고
    • Interactions of ketoprofen and ibuprofen with ß-cyclodextrins in solution and in the solid state
    • P. Mura, G.P. Bettinetti, A. Manderioli, M.T. Faucci, G. Bramanti, and M. Sorrenti Interactions of ketoprofen and ibuprofen with ß-cyclodextrins in solution and in the solid state Int. J. Pharm. 166 1998 189 203
    • (1998) Int. J. Pharm. , vol.166 , pp. 189-203
    • Mura, P.1    Bettinetti, G.P.2    Manderioli, A.3    Faucci, M.T.4    Bramanti, G.5    Sorrenti, M.6
  • 36
    • 1842832659 scopus 로고    scopus 로고
    • Comparative study of ibuproxam complexation with amorphous ß-cyclodextrin derivatives in solution and in the solid state
    • P. Mura, N. Zerrouk, M.T. Faucci, F. Maestrelli, and C. Chemtob Comparative study of ibuproxam complexation with amorphous ß-cyclodextrin derivatives in solution and in the solid state Eur. J. Pharm. Biopharm. 54 2002 181 191
    • (2002) Eur. J. Pharm. Biopharm. , vol.54 , pp. 181-191
    • Mura, P.1    Zerrouk, N.2    Faucci, M.T.3    Maestrelli, F.4    Chemtob, C.5
  • 37
    • 0028071051 scopus 로고
    • Effect of chitosan on the permeability of monolayers of intestinal epithelial cells (Caco2)
    • P. Artursson, T. Lindmark, S.S. Davis, and L. Illum Effect of chitosan on the permeability of monolayers of intestinal epithelial cells (Caco2) Pharm. Res. 11 1994 1358 1361
    • (1994) Pharm. Res. , vol.11 , pp. 1358-1361
    • Artursson, P.1    Lindmark, T.2    Davis, S.S.3    Illum, L.4
  • 38
    • 0030455292 scopus 로고    scopus 로고
    • Chitosan as absorption enhancers for poorly absorbable drugs.1. Influence of molecular weight and degree of acetylation on drug transport across human intestinal epithelial (Caco-2) cells
    • N.G.M. Schipper, M.V. Kjell, and P. Artursson Chitosan as absorption enhancers for poorly absorbable drugs.1. Influence of molecular weight and degree of acetylation on drug transport across human intestinal epithelial (Caco-2) cells Pharm. Res. 13 1996 1686 1692
    • (1996) Pharm. Res. , vol.13 , pp. 1686-1692
    • Schipper, N.G.M.1    Kjell, M.V.2    Artursson, P.3
  • 39
    • 0028875096 scopus 로고
    • Drug delivery studies in Caco-2 monolayers. IV. Absorption enhancer effects of cyclodextrins
    • L. Hovgaard, and H. Brondsted Drug delivery studies in Caco-2 monolayers. IV. Absorption enhancer effects of cyclodextrins Pharm. Res. 12 1995 1328 1332
    • (1995) Pharm. Res. , vol.12 , pp. 1328-1332
    • Hovgaard, L.1    Brondsted, H.2
  • 40
    • 0037432169 scopus 로고    scopus 로고
    • Involvement of cholesterol in the inhibitory effect of dimethyl-β-cyclodextrin on P-glycoprotein and MRP2 function in Caco-2 cells
    • K. Yunomae, H. Arima, F. Hirayama, and K. Uekama Involvement of cholesterol in the inhibitory effect of dimethyl-β-cyclodextrin on P-glycoprotein and MRP2 function in Caco-2 cells FEBS Lett. 536 2003 225 231
    • (2003) FEBS Lett. , vol.536 , pp. 225-231
    • Yunomae, K.1    Arima, H.2    Hirayama, F.3    Uekama, K.4
  • 41
    • 0030596496 scopus 로고    scopus 로고
    • Cyclodextrins - Useful excipients for oral peptide administration?
    • B. Haeberlin, T. Gengenbacher, A. Meinzer, and G. Fricker Cyclodextrins - useful excipients for oral peptide administration? Int. J. Pharm. 137 1996 103 110
    • (1996) Int. J. Pharm. , vol.137 , pp. 103-110
    • Haeberlin, B.1    Gengenbacher, T.2    Meinzer, A.3    Fricker, G.4
  • 42
    • 0035032440 scopus 로고    scopus 로고
    • Contribution of P-glycoprotein to the enhancing effects of dimethyl-β-cyclodextrin on oral bioavailability of tacrolimus
    • H. Arima, K. Yunomae, F. Hirayama, and K. Uekama Contribution of P-glycoprotein to the enhancing effects of dimethyl-β-cyclodextrin on oral bioavailability of tacrolimus J. Pharmacol. Exp. Therap. 297 2001 547 555
    • (2001) J. Pharmacol. Exp. Therap. , vol.297 , pp. 547-555
    • Arima, H.1    Yunomae, K.2    Hirayama, F.3    Uekama, K.4
  • 43
    • 10644250881 scopus 로고    scopus 로고
    • Cytotoxicity of thermosensitive polymers poly(N-isopropylacrylamide), poly(N-vinylcaprolactam) and amphiphilically modified poly(N-vinylcaprolactam)
    • H. Vihola, A. Laukkanen, L. Valtola, H. Tenhu, and J. Hirvonen Cytotoxicity of thermosensitive polymers poly(N-isopropylacrylamide), poly(N-vinylcaprolactam) and amphiphilically modified poly(N-vinylcaprolactam) Biomaterials 26 2005 3055 3064
    • (2005) Biomaterials , vol.26 , pp. 3055-3064
    • Vihola, H.1    Laukkanen, A.2    Valtola, L.3    Tenhu, H.4    Hirvonen, J.5
  • 44
    • 0034183589 scopus 로고    scopus 로고
    • Flutamide-hydroxypropyl-β-cyclodextrin complex: Formulation, physical characterization and absorption studies using the Caco-2 in vitro model
    • Z. Zuo, G. Twon, B. Stevenson, J. Diakur, and L.I. Wiebe Flutamide-hydroxypropyl-β-cyclodextrin complex: formulation, physical characterization and absorption studies using the Caco-2 in vitro model J. Pharm. Pharmaceut. Sci. 3 2000 220 227
    • (2000) J. Pharm. Pharmaceut. Sci. , vol.3 , pp. 220-227
    • Zuo, Z.1    Twon, G.2    Stevenson, B.3    Diakur, J.4    Wiebe, L.I.5
  • 46
    • 3242673511 scopus 로고    scopus 로고
    • Cyclodextrins in nasal delivery of low-molecular-weight heparins: In vivo and in vitro studies
    • T. Yang, A. Hussain, J. Paulson, T.J. Abbruscato, and F. Ahsan Cyclodextrins in nasal delivery of low-molecular-weight heparins: in vivo and in vitro studies Pharm Res. 21 2004 1127 1136
    • (2004) Pharm Res. , vol.21 , pp. 1127-1136
    • Yang, T.1    Hussain, A.2    Paulson, J.3    Abbruscato, T.J.4    Ahsan, F.5


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