Synthesis and DNA-binding ability of pyrrolo[2,1-c][1,4]benzodiazepine- azepane conjugates

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 5, 2006, Pages 1160-1163

  Kamal, Ahmed ^a   Reddy, D Rajasekhar ^a   Reddy, P S Murali Mohan ^a   Rajendar, ^a  

^a INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

Author keywords

DNA binding ability; Hydroxyazepane; Pyrrolobenzodiazepine

Indexed keywords

ALKANE; ANTIBIOTIC AGENT; PYRROLO[2,1 C][1,4]BENZODIAZEPINE AZEPANE DERIVATIVE; PYRROLO[2,1 C][1,4]BENZODIAZEPINE DERIVATIVE; SIBIROMYCIN; SPACER DNA; UNCLASSIFIED DRUG;

ARTICLE; CATTLE; CONJUGATE; CONTROLLED STUDY; DNA BINDING; DNA DENATURATION; DNA HELIX; DRUG DNA BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; MELTING POINT; NONHUMAN; TEMPERATURE;

ANIMALS; AZEPINES; BENZODIAZEPINES; CATTLE; DNA; MOLECULAR STRUCTURE; NUCLEIC ACID DENATURATION; PYRROLES; TEMPERATURE;

BOS TAURUS;

EID: 31344463267     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.11.090     Document Type: Article

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