SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 4, 2006, Pages 1049-1053

A novel nicotinic acetylcholine receptor antagonist radioligand for PET studies

(6) Ding, Yu Shin a Kil, Kun Eek a Lin, Kuo Shyan b Ma, Wei c Yokota, Yasuno c Carroll, Ivy F c

a BROOKHAVEN NATIONAL LABORATORY (United States)

b UNIVERSITY OF PITTSBURGH SCHOOL OF MEDICINE (United States)

c RTI INTERNATIONAL (United States)

Author keywords

Antagonist; C 11; nAChR; PET

Indexed keywords

CARBON 11; EPIBATIDINE; N METHYL 3' IODO EPIBATIDINE; NICOTINIC ACETYLCHOLINE RECEPTOR ANTAGONIST; NICOTINIC RECEPTOR; NICOTINIC RECEPTOR BLOCKING AGENT; RADIOLIGAND; TRACER; UNCLASSIFIED DRUG;

ARTICLE; BABOON; BLOOD ANALYSIS; BODY TEMPERATURE; HOT PLATE TEST; IMAGING SYSTEM; ISOTOPE LABELING; LIPOPHILICITY; NONHUMAN; PLASMA PROTEIN BINDING; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; REPRODUCIBILITY; SIGNAL NOISE RATIO; TAIL FLICK TEST;

ANIMALS; BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING, COMPETITIVE; BRAIN; CARBON RADIOISOTOPES; DRUG EVALUATION, PRECLINICAL; LIGANDS; MOLECULAR STRUCTURE; NICOTINE; NICOTINIC ANTAGONISTS; PAPIO; POSITRON-EMISSION TOMOGRAPHY; RECEPTORS, NICOTINIC; STRUCTURE-ACTIVITY RELATIONSHIP; TIME FACTORS;

PAPIO HAMADRYAS; PRIMATES;

EID: 30344466062 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.10.075 Document Type: Article

Times cited : (19)

References (27)

1
- 4344692338
- H. Eyre, R. Kahn, R.M. Robertson, N.G. Clark, C. Doyle, T. Gansler, T. Glynn, Y. Hong, R.A. Smith, K. Taubert, and M.J. Thun CA Cancer J. Clin. 54 2004 190
- (2004) CA Cancer J. Clin. , vol.54 , pp. 190
- Eyre, H.¹ Kahn, R.² Robertson, R.M.³ Clark, N.G.⁴ Doyle, C.⁵ Gansler, T.⁶ Glynn, T.⁷ Hong, Y.⁸ Smith, R.A.⁹ Taubert, K.¹⁰ Thun, M.J.¹¹

2
- 0031953997
- E.F. Domino Neuropsychopharmacology 18 1998 456
- (1998) Neuropsychopharmacology , vol.18 , pp. 456
- Domino, E.F.¹

3
- 0030069188
- R. Peto, A.D. Lopez, J. Boreham, M. Thun, C.J. Heath, and R. Doll Br. Med. Bull. 52 1996 12
- (1996) Br. Med. Bull. , vol.52 , pp. 12
- Peto, R.¹ Lopez, A.D.² Boreham, J.³ Thun, M.⁴ Heath, C.J.⁵ Doll, R.⁶

4
- 0029943635
- F.E. Pontieri, G. Tanda, F. Orzi, and G. Di Chiara Nature 382 1996 255
- (1996) Nature , vol.382 , pp. 255
- Pontieri, F.E.¹ Tanda, G.² Orzi, F.³ Di Chiara, G.⁴

5
- 10544241544
- Y.-S. Ding, S.J. Gatley, J.S. Fowler, N.D. Volkow, D. Aggarwal, J. Logan, S.L. Dewey, F. Liang, F.I. Carroll, and M.J. Kuhar Synapse 24 1996 403
- (1996) Synapse , vol.24 , pp. 403
- Ding, Y.-S.¹ Gatley, S.J.² Fowler, J.S.³ Volkow, N.D.⁴ Aggarwal, D.⁵ Logan, J.⁶ Dewey, S.L.⁷ Liang, F.⁸ Carroll, F.I.⁹ Kuhar, M.J.¹⁰

6
- 0032892066
- Y.-S. Ding, P. Molina, J. Fowler, J. Logan, N. Volkow, M. Kuhar, and F. Carroll Nucl. Med. Biol. 26 1999 139
- (1999) Nucl. Med. Biol. , vol.26 , pp. 139
- Ding, Y.-S.¹ Molina, P.² Fowler, J.³ Logan, J.⁴ Volkow, N.⁵ Kuhar, M.⁶ Carroll, F.⁷

7
- 0033978293
- Y.-S. Ding, N.D. Volkow, J. Logan, V. Garza, N. Pappas, P. King, and J.S. Fowler Synapse 35 2000 234
- (2000) Synapse , vol.35 , pp. 234
- Ding, Y.-S.¹ Volkow, N.D.² Logan, J.³ Garza, V.⁴ Pappas, N.⁵ King, P.⁶ Fowler, J.S.⁷

8
- 0034066935
- Y.-S. Ding, J. Logan, R. Bermel, V. Garza, O. Rice, J.S. Fowler, and N.D. Volkow J. Neurochem. 74 2000 1514
- (2000) J. Neurochem. , vol.74 , pp. 1514
- Ding, Y.-S.¹ Logan, J.² Bermel, R.³ Garza, V.⁴ Rice, O.⁵ Fowler, J.S.⁶ Volkow, N.D.⁷

9
- 0034182449
- Y.-S. Ding, N. Liu, T. Wang, J. Marecek, V. Garza, I. Ojima, and J.S. Fowler Nucl. Med. Biol. 27 2000 381
- (2000) Nucl. Med. Biol. , vol.27 , pp. 381
- Ding, Y.-S.¹ Liu, N.² Wang, T.³ Marecek, J.⁴ Garza, V.⁵ Ojima, I.⁶ Fowler, J.S.⁷

10
- 0036169966
- M. Fujita, J.P. Seibyl, D.B. Vaupel, G. Tamagnan, M. Early, S.S. Zoghbi, R.M. Baldwin, A.G. Horti, A.O. Koren, A.G. Mukhin, S. Khan, A. Bozkurt, A.S. Kimes, E.D. London, and R.B. Innis Eur. J. Nucl. Med. Mol. Imaging 29 2002 183
- (2002) Eur. J. Nucl. Med. Mol. Imaging , vol.29 , pp. 183
- Fujita, M.¹ Seibyl, J.P.² Vaupel, D.B.³ Tamagnan, G.⁴ Early, M.⁵ Zoghbi, S.S.⁶ Baldwin, R.M.⁷ Horti, A.G.⁸ Koren, A.O.⁹ Mukhin, A.G.¹⁰ Khan, S.¹¹ Bozkurt, A.¹² Kimes, A.S.¹³ London, E.D.¹⁴ Innis, R.B.¹⁵

11
- 0037927968
- A.S. Kimes, A.G. Horti, E.D. London, S.I. Chefer, C. Contoreggi, M. Ernst, P. Friello, A.O. Koren, V. Kurian, J.A. Matochik, O. Pavlova, D.B. Vaupel, and A.G. Mukhin FASEB J. 17 2003 1331
- (2003) FASEB J. , vol.17 , pp. 1331
- Kimes, A.S.¹ Horti, A.G.² London, E.D.³ Chefer, S.I.⁴ Contoreggi, C.⁵ Ernst, M.⁶ Friello, P.⁷ Koren, A.O.⁸ Kurian, V.⁹ Matochik, J.A.¹⁰ Pavlova, O.¹¹ Vaupel, D.B.¹² Mukhin, A.G.¹³

12
- 3242749145
- Y.-S. Ding, J.S. Fowler, J. Logan, G.-J. Wang, F. Telang, V. Garza, A. Biegon, D. Pareto, W. Rooney, C. Shea, D. Alexoff, N.D. Volkow, and F. Vocci Synapse 53 2004 184
- (2004) Synapse , vol.53 , pp. 184
- Ding, Y.-S.¹ Fowler, J.S.² Logan, J.³ Wang, G.-J.⁴ Telang, F.⁵ Garza, V.⁶ Biegon, A.⁷ Pareto, D.⁸ Rooney, W.⁹ Shea, C.¹⁰ Alexoff, D.¹¹ Volkow, N.D.¹² Vocci, F.¹³

13
- 14844302779
- H. McRobbie Br. J. Cardiol. 12 2005 37
- (2005) Br. J. Cardiol. , vol.12 , pp. 37
- McRobbie, H.¹

14
- 0030724888
- P.E. Molina, Y.-S. Ding, F.I. Carroll, F. Liang, N.D. Volkow, N. Pappas, M. Kuhar, N. Abumrad, S.J. Gatley, and J.S. Fowler Nucl. Med. Biol. 24 1997 743
- (1997) Nucl. Med. Biol. , vol.24 , pp. 743
- Molina, P.E.¹ Ding, Y.-S.² Carroll, F.I.³ Liang, F.⁴ Volkow, N.D.⁵ Pappas, N.⁶ Kuhar, M.⁷ Abumrad, N.⁸ Gatley, S.J.⁹ Fowler, J.S.¹⁰

15
- 4143122118
- F.I. Carroll, R. Ware, L.E. Brieaddy, H.A. Navarro, M.I. Damaj, and B.R. Martin J. Med. Chem. 47 2004 4588
- (2004) J. Med. Chem. , vol.47 , pp. 4588
- Carroll, F.I.¹ Ware, R.² Brieaddy, L.E.³ Navarro, H.A.⁴ Damaj, M.I.⁵ Martin, B.R.⁶

16
- 13944260442
- F.I. Carroll, W. Ma, Y. Yokota, J.R. Lee, L.E. Brieaddy, H.A. Navarro, M.I. Damaj, and B.R. Martin J. Med. Chem. 48 2005 1221
- (2005) J. Med. Chem. , vol.48 , pp. 1221
- Carroll, F.I.¹ Ma, W.² Yokota, Y.³ Lee, J.R.⁴ Brieaddy, L.E.⁵ Navarro, H.A.⁶ Damaj, M.I.⁷ Martin, B.R.⁸

17
- 23944507549
- Y. Huang, Z. Zhu, Y. Xiao, and M.E. Laruelle Bioorg. Med. Chem. Lett. 15 2005 4385
- (2005) Bioorg. Med. Chem. Lett. , vol.15 , pp. 4385
- Huang, Y.¹ Zhu, Z.² Xiao, Y.³ Laruelle, M.E.⁴

18
- 3242682430
- K.-S. Lin, and Y.-S. Ding Chirality 16 2004 475
- (2004) Chirality , vol.16 , pp. 475
- Lin, K.-S.¹ Ding, Y.-S.²

19
- 20544462558
- K.-S. Lin, and Y.-S. Ding Bioorg. Med. Chem. 13 2005 4658
- (2005) Bioorg. Med. Chem. , vol.13 , pp. 4658
- Lin, K.-S.¹ Ding, Y.-S.²

20
- 0242653791
- Y.-S. Ding, K.-S. Lin, V. Garza, P. Carter, D. Alexoff, J. Logan, C. Shea, Y. Xu, and P. King Synapse 50 2003 345
- (2003) Synapse , vol.50 , pp. 345
- Ding, Y.-S.¹ Lin, K.-S.² Garza, V.³ Carter, P.⁴ Alexoff, D.⁵ Logan, J.⁶ Shea, C.⁷ Xu, Y.⁸ King, P.⁹

21
- 22244464188
- Y.-S. Ding, K.S. Lin, H. Benveniste, and P. Carter J. Neurochem. 94 2005 337
- (2005) J. Neurochem. , vol.94 , pp. 337
- Ding, Y.-S.¹ Lin, K.S.² Benveniste, H.³ Carter, P.⁴

22
- 15044345704
- S. Chattopadhyay, B. Xue, D. Collins, R. Pichika, R. Bagnera, F.M. Leslie, B.T. Christian, B. Shi, T.K. Narayanan, S.G. Potkin, and J. Mukherjee J. Nucl. Med. 46 2005 130
- (2005) J. Nucl. Med. , vol.46 , pp. 130
- Chattopadhyay, S.¹ Xue, B.² Collins, D.³ Pichika, R.⁴ Bagnera, R.⁵ Leslie, F.M.⁶ Christian, B.T.⁷ Shi, B.⁸ Narayanan, T.K.⁹ Potkin, S.G.¹⁰ Mukherjee, J.¹¹

23
- 0032477904
- N.H. Lin, D.E. Gunn, Y. Li, Y. He, H. Bai, K.B. Ryther, T. Kuntzweiler, D.L. Donnelly-Roberts, D.J. Anderson, J.E. Campbell, J.P. Sullivan, S.P. Arneric, and M.W. Holladay Bioorg. Med. Chem. Lett. 8 1998 249
- (1998) Bioorg. Med. Chem. Lett. , vol.8 , pp. 249
- Lin, N.H.¹ Gunn, D.E.² Li, Y.³ He, Y.⁴ Bai, H.⁵ Ryther, K.B.⁶ Kuntzweiler, T.⁷ Donnelly-Roberts, D.L.⁸ Anderson, D.J.⁹ Campbell, J.E.¹⁰ Sullivan, J.P.¹¹ Arneric, S.P.¹² Holladay, M.W.¹³

24
- 0030026025
- Y.-S. Ding, S.J. Gatley, J.S. Fowler, R. Chen, N.D. Volkow, J. Logan, C.E. Shea, Y. Sugano, and J. Koomen Life Sci. 58 1996 195
- (1996) Life Sci. , vol.58 , pp. 195
- Ding, Y.-S.¹ Gatley, S.J.² Fowler, J.S.³ Chen, R.⁴ Volkow, N.D.⁵ Logan, J.⁶ Shea, C.E.⁷ Sugano, Y.⁸ Koomen, J.⁹

25
- 1542315606
- Y. Kiyono, N. Kanegawa, H. Kawashima, Y. Kitamura, Y. Iida, and H. Saji Nucl. Med. Biol. 31 2004 147
- (2004) Nucl. Med. Biol. , vol.31 , pp. 147
- Kiyono, Y.¹ Kanegawa, N.² Kawashima, H.³ Kitamura, Y.⁴ Iida, Y.⁵ Saji, H.⁶

26
- 0038792263
- C.A. Mathis, Y. Wang, D.P. Holt, G.-F. Huang, M.L. Debnath, and W.E. Klunk J. Med. Chem. 46 2003 2740
- (2003) J. Med. Chem. , vol.46 , pp. 2740
- Mathis, C.A.¹ Wang, Y.² Holt, D.P.³ Huang, G.-F.⁴ Debnath, M.L.⁵ Klunk, W.E.⁶

27
- 0037399615
- S.I. Chefer, E.D. London, A.O. Koren, O.A. Pavlova, V. Kurian, A.S. Kimes, A.G. Horti, and A.G. Mukhin Synapse 48 2003 25
- (2003) Synapse , vol.48 , pp. 25
- Chefer, S.I.¹ London, E.D.² Koren, A.O.³ Pavlova, O.A.⁴ Kurian, V.⁵ Kimes, A.S.⁶ Horti, A.G.⁷ Mukhin, A.G.⁸

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.