Epibatidine analogues as selective ligands for the α xβ2-containing subtypes of nicotinic acetylcholine receptors

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 19, 2005, Pages 4385-4388

  Huang, Yiyun ^a   Zhu, Zhihong ^a   Xiao, Yingxian ^b   Laruelle, Marc ^a  

^a Department of Neurology and the Taub Institute for Research on Alzheimer's Disease and the Aging Brain   (United States)

^b GEORGETOWN UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Antagonist; Nicotinic receptors; Synthesis

Indexed keywords

EPIBATIDINE; LEAD; LIGAND; NICOTINE; NICOTINIC AGENT; RECEPTOR SUBTYPE;

ARTICLE; DRUG ACTIVITY; DRUG DESIGN; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; RECEPTOR AFFINITY;

BICYCLO COMPOUNDS, HETEROCYCLIC; CELL LINE; HUMANS; LIGANDS; NICOTINIC AGONISTS; PYRIDINES; RADIOLIGAND ASSAY; RECEPTORS, NICOTINIC; STRUCTURE-ACTIVITY RELATIONSHIP; TRANSFECTION;

EID: 23944507549     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.06.039     Document Type: Article

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