Parallel microwave-assisted library of imidazothiazol-3-ones and imidazothiazin-4-ones

Journal of Combinatorial Chemistry

Volumn 7, Issue 6, 2005, Pages 947-951

  Le Bas, Marie Delphine H ^a   O'Shea, Donal F ^a  

^a UNIVERSITY COLLEGE DUBLIN   (Ireland)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 28244492850     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc0500856     Document Type: Article

References (34)

1. For reviews see: (a) Kappe, C. O. Angew. Chem., Int. Ed. 2004, 43, 6250.
2. (b) Nüchter, M.; Ondruschka, B.; Bonrath, W.; Gum, A. Green Chem. 2004, 6, 128.
3. (c) Blackwell, H. E. Org. Biomol. Chem. 2003, 1, 1251.
4. (d) Mavandadi, F.; Lidström, P. Curr. Top. Med. Chem. 2004, 4, 773.
5. (e) Lew, A.; Krutznik, P. O.; Hart, M. E.; Chamberlin, A. R. J. Comb. Chem. 2002, 4, 95.
6. (a) Varma, R. S. Pure Appl. Chem. 2001, 73, 193.
7. (b) Usyatinsky, A. Ya.; Khmelnitsky, Y. L. Tetrahedron Lett. 2000, 41, 5031.
8. (c) Cotterill, I. C.; Usyatinsky, A. Ya.; Arnold, J. M.; Clark, D. S.; Dordick, J. S.; Michels, P. C.; Khmelnitsky, Y. L. Tetrahedron Lett. 1998, 39, 1117.
9. (a) Ferguson, J. D. Mol. Diversity 2003, 7, 281.
10. (b) Schanche, J.-S. Mol. Diversity 2003, 7, 293.
11. (a) Favretto, L. Mol. Diversity 2003, 7, 287.
12. (b) http://www.anton-paar.com.
13. Another approach to high-throughput microwave library synthesis has been recently proposed by exploiting microwave heating in conjunction with continuous flow microreactors. See: Comer, E.; Organ, M. G. J. Am. Chem. Soc. 2005, 127, 8160.
14. (a) Santagada, V.; Frecentese, F.; Perissutti, E.; Fiorino, F.; Severino, B.; Cirillo, D.; Terracciano, S.; Caliendo, G. J. Comb. Chem. 2005, 7, 618.
15. (b) Alcazar, J. J. Comb. Chem. 2005, 7, 353.
16. Coleman, C. M.; MacElroy, J. M. D.; Gallagher, J. F.; O'Shea, D. F. J. Comb. Chem. 2002, 4, 87.
17. LeBas, M.-D. H.; McKinley, N. F.; Hogan, A.-M. L.; O'Shea, D. F. J. Comb. Chem. 2005, 7, 503.
18. Ostresh, J. M.; Husar, G. M.; Blondelle, S. E.; Dorner, B.; Weber, P. A.; Houghten, R. A. Proc. Natl. Acad. Sci. U.S.A. 1994, 91, 11138.
19. Wipf, P.; Coleman, C. M.; Janjic, J. M.; Iyer, P. S.; Fodor, M. D.; Shafer, Y. A.; Stephenson, C. R. J.; Kendall, C.; Day, B. W. J. Comb. Chem. 2005, 7, 322.
20. Milestone MicroSYNTH laboratory microwave using the easy Wave control software with the manufacturers reference vessel containing an internal fiber-optic temperature sensor.
21. Asinger, F.; Gentz, F. Angew. Chem., Int. Ed. Engl. 1963, 2, 397.
22. Tanaka, M.; Koyanagi, M. Synthesis 1981, 973.
23. (a) Lange, U. E. W. Tetrahedron Lett. 2002, 43, 6857.
24. (b) Weinshenker, N. M.; Shen, C. M.; Wong, J. Y. Org. Synth. 1988, 50, 951.
25. For recent examples, see; (a) Donati, D.; Morelli, C.; Taddei, M. Tetrahedron Lett. 2005, 46, 2817.
26. (b) Crosignani, S.; White, P. D.; Linclau, B. J. Org. Chem. 2004, 69, 5897.
27. (c) Petricci, E.; Mugnaini, C.; Radi, M.; Corelli, F.; Botta, M. J. Org. Chem. 2004, 69, 7880.
28. (d) Lei, X.; Porco, J. A., Jr. Org. Lett. 2004, 6, 795.
29. (e) Sauer, D. R.; Kalvin, D.; Phelan, K. M. Org. Lett. 2003, 5, 4721.
30. (f) Crosignani, S.; White, P. D.; Linclau, B. Org. Lett. 2002, 4, 2961.
31. (g) Ley, S. V.; Taylor, S. J. Bioorg. Med. Chem. Lett. 2002, 12, 1813.
32. (h) Launay, D.; Booth, S.; Clemens, I.; Merritt, A.; Bradley, M. Tetrahedron Lett. 2002, 43, 7201.
33. (i) Westman, J. Org. Lett. 2001, 3, 3745.
34. (j) Ley, S. V.; Leach, A. G.; Storer, R. I. J. Chem. Soc., Perkin Trans. 1 2001, 358.