Alteration of intracellular histamine H2 receptor cycling precedes antagonist-induced upregulation

American Journal of Physiology - Gastrointestinal and Liver Physiology

Volumn 289, Issue 5 52-5, 2005, Pages

  Osawa, Satoshi ^a   Kajimura, Masayoshi ^a   Yamamoto, Seiji ^a   Ikuma, Mutsuhiro ^a   Mochizuki, Chihiro ^a   Iwasaki, Hirohiko ^a   Hishida, Akira ^a   Terakawa, Susumu ^a  

^a HAMAMATSU UNIVERSITY SCHOOL OF MEDICINE   (Japan)

Author keywords

Constitutive activity; Endocytosis; Internalization; Inverse agonist; Recycling

Indexed keywords

ADENYLATE CYCLASE; CIMETIDINE; CYCLOHEXIMIDE; FAMOTIDINE; GREEN FLUORESCENT PROTEIN; HISTAMINE; HISTAMINE H2 RECEPTOR; HISTAMINE H2 RECEPTOR ANTAGONIST; ISOBUTYLMETHYLXANTHINE; MESSENGER RNA; RANITIDINE; TIOTIDINE;

ARTICLE; BINDING AFFINITY; CELL MEMBRANE; CELL STRAIN HEK293; CONTROLLED STUDY; ENDOSOME; FLUORESCENCE; HUMAN; HUMAN CELL; INTERNALIZATION; PRIORITY JOURNAL; PROTEIN DEGRADATION; PROTEIN EXPRESSION; PROTEIN SYNTHESIS; PROTEIN TRANSPORT; RECEPTOR UPREGULATION; RECYCLING; STOMACH ACID SECRETION; STOMACH PARIETAL CELL;

CELL LINE; CIMETIDINE; FAMOTIDINE; HISTAMINE H2 ANTAGONISTS; HUMANS; PROTEIN TRANSPORT; RANITIDINE; RECEPTORS, HISTAMINE H2; RNA, MESSENGER; UP-REGULATION;

EID: 27444446541     PISSN: 01931857     EISSN: None     Source Type: Journal    
DOI: 10.1152/ajpgi.00536.2004     Document Type: Article

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