Inverse agonism of histamine H2 antagonists accounts for upregulation of spontaneously active histamine H2 receptors

Proceedings of the National Academy of Sciences of the United States of America

Volumn 93, Issue 13, 1996, Pages 6802-6807

  Smit, Martine J ^a,b   Leurs, Rob ^a   Alewijnse, Astrid E ^a   Blauw, Joeri ^a   Van Nieuw Amerongen, Gerard P ^a   Van De Vrede, Yvonne ^a   Roovers, Edwin ^a   Timmerman, Henk ^a  

^a VU UNIVERSITY AMSTERDAM   (Netherlands)

^b CITY UNIVERSITY OF NEW YORK   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 (2 HYDROXYETHYL) 1 PIPERAZINEETHANESULFONIC ACID; BURIMAMIDE; CIMETIDINE; CYCLIC AMP; FORSKOLIN; HISTAMINE; HISTAMINE H2 RECEPTOR; HISTAMINE H2 RECEPTOR ANTAGONIST; IODOAMINOPOTENTIDINE I 125; ISOBUTYLMETHYLXANTHINE; RADIOPHARMACEUTICAL AGENT; RANITIDINE; TIOTIDINE; UNCLASSIFIED DRUG; VUF 8299;

ANIMAL CELL; ARTICLE; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENTIATION; DRUG RECEPTOR BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR DENSITY; RECEPTOR UPREGULATION;

ANIMALS; BURIMAMIDE; CHO CELLS; CIMETIDINE; CRICETINAE; CYCLIC AMP; FORSKOLIN; HISTAMINE AGONISTS; HISTAMINE H2 ANTAGONISTS; RANITIDINE; RECEPTORS, HISTAMINE H2; TRANSFECTION; UP-REGULATION;

EID: 0029948346     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.93.13.6802     Document Type: Article

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