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Volumn 40, Issue 11, 2005, Pages 1123-1128

Synthesis and biological activity of alpha-bromoacryloyl lexitropsin conjugates

(8) Romagnoli, Romeo a Baraldi, Pier Giovanni a Iaconinoto, Maria Antonietta a Carrion, Maria Dora a Tabrizi, Mojgan Aghazadeh a Gambari, Roberto a Borgatti, Monica a Heilmann, Jörg b

a UNIVERSITY OF FERRARA (Italy)

b UNIVERSITY OF REGENSBURG (Germany)

Author keywords

Alpha bromoacryloyl; Benzoheterocycle; DNA minor groove binders; Glutathione

Indexed keywords

3 [1 METHYL 3 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)INDOLE 2 CARBOXAMIDO]PYRAZOLE 5 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; 3 [1 METHYL 4 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)INDOLE 2 CARBOXAMIDO]IMIDAZOLE 2 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; 3 [1 METHYL 4 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)INDOLE 2 CARBOXAMIDO]PYRROLE 2 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; 3 [3 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)BENZOFURANE 2 CARBOXAMIDO]PYRAZOLE 5 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; 3 [3 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)BENZOTHIOPHENE 2 CARBOXAMIDO]PYRAZOLE 5 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; 3 [4 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)BENZOFURANE 2 CARBOXAMIDO]IMIDAZOLE 2 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; 3 [4 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)BENZOFURANE 2 CARBOXAMIDO]PYRROLE 2 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; 3 [4 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)BENZOTHIOPHENE 2 CARBOXAMIDO]IMIDAZOLE 2 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; 3 [4 [1 METHYL 5 (ALPHA BROMOACRYLAMIDO)BENZOTHIOPHENE 2 CARBOXAMIDO]PYRROLE 2 CARBOXAMIDO]DIMETHYLAMINOPROPYLAMINOLEXITROPSIN; ALPHA BROMOACRYLOYL LEXITROPSIN; ANTILEUKEMIC AGENT; GLUTATHIONE; LEXITROPSIN; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL STRAIN K 562; CELL STRAIN KB; CONTROLLED STUDY; CYTOTOXICITY; DRUG ACTIVITY; DRUG CONJUGATION; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; HUMAN; HUMAN CELL; LEUKEMIA L 1210; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTINEOPLASTIC AGENTS, ALKYLATING; BENZOFURANS; DRUG SCREENING ASSAYS, ANTITUMOR; HETEROCYCLIC COMPOUNDS; HUMANS; IMIDAZOLES; MICE; MOLECULAR STRUCTURE; NETROPSIN; PYRAZOLES; PYRROLES; STRUCTURE-ACTIVITY RELATIONSHIP; THIOPHENES; TUMOR CELLS, CULTURED;

EID: 26844451868 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2005.05.003 Document Type: Article

Times cited : (5)

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