Allosteric modulators affect the internalization of human adenosine A 1 receptors

European Journal of Pharmacology

Volumn 522, Issue 1-3, 2005, Pages 1-8

  Klaasse, Elisabeth C ^a   Van Den Hout, Gijs ^a   Roerink, Sophie F ^a   De Grip, Willem J ^b   Ijzerman, Ad P ^a   Beukers, Margot W ^a  

^a LEIDEN UNIVERSITY   (Netherlands)

^b LEIDEN UNIVERSITY   (Netherlands)

Author keywords

Allosteric modulation; Human adenosine A1 receptor; Internalization; PD 81,723; SCH 202676; YFP

Indexed keywords

2 AMINO 4,5 DIMETHYL 3 (3 TRIFLUOROMETHYLBENZOYL)THIOPHENE; ADENOSINE A1 RECEPTOR; ADENOSINE DERIVATIVE; N (2,3 DIPHENYL 1,2,4 THIADIAZOL 5(2H) YLIDENE)METHANAMINE; RADIOLIGAND;

ALLOSTERISM; ARTICLE; CELL LINE; CHO CELL; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DRUG EFFECT; HUMAN; HUMAN CELL; LIGAND BINDING; PRIORITY JOURNAL; RECEPTOR AFFINITY;

ADENOSINE; ALLOSTERIC REGULATION; ANIMALS; BINDING, COMPETITIVE; CHO CELLS; CRICETINAE; CRICETULUS; DOSE-RESPONSE RELATIONSHIP, DRUG; ENDOCYTOSIS; HUMANS; LUMINESCENT PROTEINS; MICROSCOPY, CONFOCAL; RADIOLIGAND ASSAY; RECEPTOR, ADENOSINE A1; RECOMBINANT FUSION PROTEINS; THIAZOLES; THIOPHENES; TRANSFECTION; TRITIUM; XANTHINES;

EID: 26844448531     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2005.08.052     Document Type: Article

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