Agonist-independent effect of an allosteric enhancer of the A1 adenosine receptor in CHO cells stably expressing the recombinant human A1 receptor

Journal of Pharmacology and Experimental Therapeutics

Volumn 281, Issue 2, 1997, Pages 761-768

  Kollias Baker, C A ^a,d   Ruble, J ^a   Jacobson, M ^c   Harrison, J K ^b   Ozeck, M ^b   Shryock, J C ^a   Belardinelli, L ^a,b  

^a UNIVERSITY OF FLORIDA COLLEGE OF MEDICINE   (United States)

^b UNIVERSITY OF FLORIDA   (United States)

^c MERCK RESEARCH LABORATORIES   (United States)

^d UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINO 4,5 DIMETHYL 3 (3 TRIFLUOROBENZOYL)THIOPHENE; 2 AMINO 4,5 DIMETHYL 3 (3 TRIFLUOROMETHYLBENZOYL)THIOPHENE; 8 CYCLOPENTYL 1,3 DIPROPYLXANTHINE; ADENOSINE; ADENOSINE 5' O (3 THIOTRIPHOSPHATE); ADENOSINE A1 RECEPTOR; ADENOSINE A1 RECEPTOR AGONIST; ADENOSINE A1 RECEPTOR ANTAGONIST; ADENOSINE DEAMINASE; BENZOTHIOPHENE DERIVATIVE; CYCLIC AMP; CYCLOHEXYLADENOSINE; PHENYLISOPROPYLADENOSINE; RECOMBINANT PROTEIN; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING KINETICS; CHO CELL; CONTROLLED STUDY; DRUG ACTIVITY; DRUG MECHANISM; DRUG RECEPTOR BINDING; NONHUMAN; PRIORITY JOURNAL;

ADENOSINE; ADENOSINE DEAMINASE; ALLOSTERIC REGULATION; ANIMALS; CHO CELLS; CRICETINAE; CYCLIC AMP; FORSKOLIN; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; RECEPTORS, PURINERGIC P1; RECOMBINANT PROTEINS; THIOPHENES; XANTHINES;

EID: 0030926208     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (18)

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