SCH-202676: An allosteric modulator of both agonist and antagonist binding to G protein-coupled receptors

Molecular Pharmacology

Volumn 59, Issue 1, 2001, Pages 30-37

  Fawzi, Ahmad B ^a   Macdonald, Douglas ^a,c   Benbow, Lawrence L ^a   Smith Torhan, April ^a   Zhang, Hongtao ^a   Weig, Blair C ^a   Ho, Ginny ^a   Tulshian, Deen ^a   Linder, Maurine E ^b   Graziano, Michael P ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

^b WASHINGTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

^c SANOFI   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE DIPHOSPHATE; ALPHA ADRENERGIC RECEPTOR; BETA ADRENERGIC RECEPTOR; DELTA OPIATE RECEPTOR; DOPAMINE 1 RECEPTOR; DOPAMINE 2 RECEPTOR; EPIDERMAL GROWTH FACTOR RECEPTOR; G PROTEIN COUPLED RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); KAPPA OPIATE RECEPTOR; MU OPIATE RECEPTOR; MUSCARINIC M1 RECEPTOR; MUSCARINIC M2 RECEPTOR; N (2,3 DIPHENYL 1,2,4 THIADIAZOL 5(2H) YLIDENE)METHANAMINE; PERTUSSIS TOXIN; RADIOLIGAND; THIADIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING SITE; CHO CELL; CONTROLLED STUDY; ESCHERICHIA COLI; HUMAN; HUMAN CELL; LEPIDOPTERA; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING;

EID: 0035170060     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.59.1.30     Document Type: Article

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