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Volumn 7, Issue 16, 2005, Pages 3549-3552

Pd-catalyzed tandem C-N/C-C coupling of gem-dihalovinyl systems: A modular synthesis of 2-substituted indoles

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EID: 23944442185     PISSN: 15237060     EISSN: None     Source Type: Journal    
DOI: 10.1021/ol051286l     Document Type: Article
Times cited : (160)

References (36)
  • 1
    • 0003441482 scopus 로고    scopus 로고
    • John Wiley & Sons Ltd.: Chichester, U.K.
    • For a comprehensive monograph, see: Tsuji, J. Palladium Reagents and Catalysis; John Wiley & Sons Ltd.: Chichester, U.K., 2004.
    • (2004) Palladium Reagents and Catalysis
    • Tsuji, J.1
  • 4
    • 0034006847 scopus 로고    scopus 로고
    • For a review on the preparation of gem-dibromovinyl compounds, see: Eymery, F.; Iorga, B.; Savignac, P. Synthesis 2000, 185-213.
    • (2000) Synthesis , pp. 185-213
    • Eymery, F.1    Iorga, B.2    Savignac, P.3
  • 9
    • 0347653093 scopus 로고    scopus 로고
    • During our investigation, Bisseret and co-workers disclosed a related example of this reaction yielding N-acetyl-2-arylindole in moderate yield. Thielges, S.; Meddah, E.; Bisseret, P.; Eustache, J. Tetrahedron Lett. 2004, 45, 907. The scope of this reaction was not reported.
    • (2004) Tetrahedron Lett. , vol.45 , pp. 907
    • Thielges, S.1    Meddah, E.2    Bisseret, P.3    Eustache, J.4
  • 10
    • 1942534021 scopus 로고    scopus 로고
    • For recent reviews on indole-containing natural products, see: (a) Somei, M.; Yamada, F. Nat. Prod. Rep. 2004, 21, 278.
    • (2004) Nat. Prod. Rep. , vol.21 , pp. 278
    • Somei, M.1    Yamada, F.2
  • 14
    • 0003979828 scopus 로고    scopus 로고
    • Academic Press: San Diego
    • (b) Indoles; Sundberg, R. J., Ed,; Academic Press: San Diego, 1996.
    • (1996) Indoles
    • Sundberg, R.J.1
  • 20
    • 33645396760 scopus 로고    scopus 로고
    • note
    • 2O (90%) or Fe/HOAc (85%) reduction. This can also be carried out in a convenient one-pot preparation on a relatively large scale (>40 g) in 85% overall isolated yield. For experimental procedures for the preparation of all substrates in Table 2, please refer to Supporting Information.
  • 27
    • 33645402824 scopus 로고    scopus 로고
    • Patent Appl. US 2004058977
    • (b) Guo, Z.; Cheng, G.; Chu, F. U.S. Patent Appl. US 2004058977; Chem. Abstr. 2004, 140, 270734.
    • (2004) Chem. Abstr. , vol.140 , pp. 270734
    • Guo, Z.1    Cheng, G.2    Chu, F.U.S.3
  • 31
    • 33645397229 scopus 로고    scopus 로고
    • Patent WO 9,805,639, 1998
    • Gungor, T.; Teulon, J.-M. Patent WO 9,805,639, 1998; Chem. Abstr. 1998, 128, 180330.
    • (1998) Chem. Abstr. , vol.128 , pp. 180330
    • Gungor, T.1    Teulon, J.-M.2
  • 34
    • 33645403241 scopus 로고    scopus 로고
    • U.S. Patent 6,790,539, 2004
    • Lin, T.-s. U.S. Patent 6,790,539, 2004; Chem. Abstr. 2004, 140, 136161.
    • (2004) Chem. Abstr. , vol.140 , pp. 136161
    • Lin, T.-S.1
  • 36
    • 33645415074 scopus 로고    scopus 로고
    • Aldrich currently supplies a special catalog of more than 250 boronic acids and esters. This can be found at http://www.aldrich-sigma.com.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.