Distinct thermodynamic parameters of serotonin 5-HT3 agonists and antagonists to displace [3H] granisetron binding

Journal of Neurochemistry

Volumn 67, Issue 1, 1996, Pages 407-412

  Maksay, Gábor ^a  

^a CTRL RES INSTITUTE FOR CHEMISTRY   (Hungary)

Author keywords

Distinction of serotonin 5 HT3 agonists and antagonists; Granisetron binding; Neurotransmitter receptor ionophore complexes; Serotonin 5 HT3 receptors; Thermodynamics of binding

Indexed keywords

1 (3 CHLOROPHENYL)BIGUANIDE; 2 METHYLSEROTONIN; 4 AMINO 1 (6 CHLORO 2 PYRIDYL)PIPERIDINE; GRANISETRON; ION CHANNEL; ONDANSETRON; PHENYLBIGUANIDE; SEROTONIN 1 RECEPTOR; TROPISETRON; TUBOCURARINE CHLORIDE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; DRUG BINDING SITE; LIGAND BINDING; MOLECULAR INTERACTION; NEUROTRANSMITTER RELEASE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BINDING; SCATCHARD PLOT; SEROTONIN RELEASE; STRUCTURE ACTIVITY RELATION; THERMODYNAMICS;

ANIMALS; BINDING, COMPETITIVE; CEREBRAL CORTEX; GRANISETRON; HIPPOCAMPUS; LINEAR MODELS; MALE; NEURONS; RATS; RATS, WISTAR; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; SYNAPTOSOMES; THERMODYNAMICS; TIME FACTORS; TRITIUM;

ANIMALIA;

EID: 0029931275     PISSN: 00223042     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1471-4159.1996.67010407.x     Document Type: Article

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