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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 10, 2002, Pages 1379-1382

Synthesis of highly potent and selective hetaryl ureas as integrin αVβ3-receptor antagonists

(10) Lange, Udo E W b Graef, Claudia b Lauterbach, Arnulf b Subkowski, Thomas b Zechel, Christian b Backfisch, Gisela c Delzer, Jürgen c Geneste, Hervé c Hornberger, Wilfried c Kling, Andreas c

a ABBOTT GMBH AND CO KG (Germany)

b BASF SE (Germany)

c NONE

Author keywords

[No Author keywords available]

Indexed keywords

ABCIXIMAB; HETARYLUREA; INTEGRIN RECEPTOR; UNCLASSIFIED DRUG; UREA DERIVATIVE;

ANIMAL CELL; ARTICLE; CELL ASSAY; CONTROLLED STUDY; DRUG ACTIVITY; DRUG EFFICACY; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ANIMALS; CELL ADHESION; CHO CELLS; CRICETINAE; DRUG DESIGN; HUMANS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MUSCLE, SMOOTH; RECEPTORS, VITRONECTIN; STRUCTURE-ACTIVITY RELATIONSHIP; UREA;

EID: 18344375818 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(02)00161-0 Document Type: Article

Times cited : (21)

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