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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 3, 2002, Pages 441-446

Synthesis and SAR of N-substituted dibenzazepinone derivatives as novel potent and selective αVβ3 antagonists

(12) Kling, Andreas a Backfisch, Gisela a Delzer, Jürgen a Geneste, Hervé a Graef, Claudia a Holzenkamp, Uta a Hornberger, Wilfried a Lange, Udo E W b Lauterbach, Arnulf a Mack, Helmut a Seitz, Werner b Subkowski, Thomas a

a Knoll AG (Germany)

b BASF SE (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

DIBENZAZEPINE DERIVATIVE; GUANIDINE; RECEPTOR BLOCKING AGENT; VITRONECTIN RECEPTOR;

ARTICLE; CELL STRAIN CACO 2; COLON ADENOCARCINOMA; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; PHARMACOPHORE; STRUCTURE ACTIVITY RELATION;

DIBENZAZEPINES; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; FIBRINOLYTIC AGENTS; GUANIDINE; INDICATORS AND REAGENTS; MASS SPECTROMETRY; PLATELET GLYCOPROTEIN GPIIB-IIIA COMPLEX; RECEPTORS, VITRONECTIN; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 18244403789 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(01)00773-9 Document Type: Article

Times cited : (34)

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