Structural basis for antagonist-mediated recruitment of nuclear co-repressors by PPARα

Nature

Volumn 415, Issue 6873, 2002, Pages 813-817

  Xu, H Eric ^a   Stanley, Thomas B ^a   Montana, Valerie G ^a   Lambert, Millard H ^a   Shearer, Barry G ^a   Cobb, Jeffery E ^a   McKee, David D ^a   Galardi, Cristin M ^a   Plunket, Kelli D ^a   Nolte, Robert T ^a   Parks, Derek J ^a   Moore, John T ^a   Kliewer, Steven A ^a   Willson, Timothy M ^a   Stimmel, Julie B ^a  

^a GLAXOSMITHKLINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CRYSTAL STRUCTURE; GENES; HORMONES; MUTAGENESIS; PROTEINS;

NUCLEAR RECEPTORS;

BIODIVERSITY;

GW 6471; HISTONE DEACETYLASE; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA ANTAGONIST; PROTEIN INHIBITOR; PROTEIN SMRT; REGULATOR PROTEIN; UNCLASSIFIED DRUG;

BIOCHEMISTRY; CRYSTAL STRUCTURE; GENE;

ARTICLE; CRYSTAL STRUCTURE; DRUG MECHANISM; DRUG STRUCTURE; LIGAND BINDING; PRIORITY JOURNAL; RECEPTOR BINDING; STRUCTURE ANALYSIS;

EID: 18244393501     PISSN: 00280836     EISSN: None     Source Type: Journal    
DOI: 10.1038/415813a     Document Type: Article

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