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Bioorganic and Medicinal Chemistry

Volumn 13, Issue 9, 2005, Pages 3295-3308

Synthesis and pharmacological evaluation of benzamide derivatives as selective 5-HT4 receptor agonists

(5) Sonda, Shuji a Kawahara, Toshio a Katayama, Kenichi a Sato, Noriko a Asano, Kiyoshi a

a MITSUBISHI TANABE PHARMA CORPORATION (Japan)

Author keywords

5 HT4 agonist

Indexed keywords

4 AMINO 5 CHLORO 2 METHOXY N [1 (4 PHENOXYBUTYL)PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 (4 PHENOXYETHYL)PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 (4 PHENOXYPROPYL)PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 (5 PHENOXYPENTYL)PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 (6 PHENOXYHEXYL)PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 [3 (PHENYLTHIO)PROPYL]PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 [4 (PHENYLTHIO)BUTYL]PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 [5 (NAPHTHALEN 2 YL)PENTYL]PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 [5 (PHENYLSULFINYL)PENTYL]PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 [5 (PHENYLTHIO)PENTYL]PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO 2 METHOXY N [1 [6 (PHENYLTHIO)HEXYL]PIPERIDIN 4 YLMETHYL]BENZAMIDE; 4 AMINO 5 CHLORO N [1 (6 HYDROXY 6 PHENYLHEXYL)PIPERIDIN 4 YLMETHYL] 2 METHOXYBENZAMIDE; 4 AMINO 5 CHLORO N [1 [5 (4 CHLOROBENZYLOXY)PENTYL]PIPERIDIN 4 YLMETHYL] 2 METHOXYBENZAMIDE; 4 AMINO 5 CHLORO N [1 [5 (CYCLOHEXYLMETHOXY)PENTYL]PIPERIDIN 4 YLMETHYL] 2 METHOXYBENZAMIDE; 4 AMINO 5 CHLORO N [1 [6 (HYDROXYIMINO) 6 PHENYLHEXYL]PIPERIDIN 4 YLMETHYL] 2 METHOXYBENZAMIDE; 4 AMINO N [1 (4 BENZYLOXYBUTYL)PIPERIDIN 4 YLMETHYL] 5 CHLORO 2 METHOXYBENZAMIDE OXALATE; 4 AMINO N [1 (5 BENZYLOXYPENTYL)PIPERIDIN 4 YLMETHYL] 5 CHLORO 2 METHOXYBENZAMIDE OXALATE; 4 AMINO N [1 (6 BENZYLOXYHEXYL)PIPERIDIN 4 YLMETHYL] 5 CHLORO 2 METHOXYBENZAMIDE; 4 AMINO N [1 [5 (BENZYLTHIO)PENTYL]PIPERIDIN 4 YLMETHYL] 5 CHLORO 2 METHOXYBENZAMIDE OXALATE; BENZAMIDE DERIVATIVE; SEROTONIN 4 AGONIST; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DEFECATION; DRUG EFFECT; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GASTROINTESTINAL MOTILITY; MALE; NONHUMAN; RAT;

EID: 16244401471 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2005.02.016 Document Type: Article

Times cited : (18)

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