Microwave assisted solid-phase synthesis of trisubstituted 2-(2,6-purin-9-yl)acetamides

Tetrahedron Letters

Volumn 46, Issue 16, 2005, Pages 2873-2875

  Austin, Richard E ^a   Waldraff, Christian ^b   Al Obeidi, Fahad ^a  

^a Aventis Combinatorial Technol Ctr   (United States)

^b BAYER CROPSCIENCE AG   (Germany)

Author keywords

Combinatorial; Microwave; Purine; Solid phase

Indexed keywords

ACETAMIDE DERIVATIVE; AMINE; CARBON; HALOGEN; PURINE;

ARTICLE; IRRADIATION; MICROWAVE IRRADIATION; SOLID; SUBSTITUTION REACTION; SYNTHESIS;

EID: 15944379583     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2005.02.130     Document Type: Article

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21. 6): δ 8.58 (s, 1H), 5.10 (s, 2H)
22. 4): δ 8.12 (s, 1H), 7.79 (s, 1H), 7.60 (d, 1H, J = 7.6 Hz), 7.27 (m, 1H), 7.01 (m, 1H), 4.78 (s, 2H), 3.67-3.56 (m, 6H), 3.26 (m, 2H), 2.64-2.33 (m, 12H), 1.76-1.60 (m, 6H), 1.47 (m, 2H)