Imidazo[1,2-a]pyridines: A potent and selective class of cyclin-dependent kinase inhibitors identified through structure-based hybridisation

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 18, 2003, Pages 3021-3026

  Anderson, Malcolm ^a   Beattie, John F ^a   Breault, Gloria A ^a   Breed, Jason ^a   Byth, Kate F ^a   Culshaw, Janet D ^a   Ellston, Rebecca P A ^a   Green, Stephen ^a   Minshull, Claire A ^a   Norman, Richard A ^a   Pauptit, Richard A ^a   Stanway, Judith ^a   Thomas, Andrew P ^a   Jewsbury, Philip J ^a  

^a ASTRAZENECA   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; CYCLIN DEPENDENT KINASE 2; CYCLIN DEPENDENT KINASE 4; CYCLIN DEPENDENT KINASE INHIBITOR; PYRIDINE DERIVATIVE; PYRIMIDINE DERIVATIVE;

ARTICLE; COMPARATIVE STUDY; DRUG BINDING; DRUG SCREENING; HYBRIDIZATION; IC 50; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

EID: 12444257368     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00638-3     Document Type: Article

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