Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56Lck

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 22, 2003, Pages 4007-4010

  Wityak, John ^a   Das, Jagabandhu ^a   Moquin, Robert V ^a   Shen, Zhongqi ^a   Lin, James ^a   Chen, Ping ^a   Doweyko, Arthur M ^a   Pitt, Sidney ^a   Pang, Suhong ^a   Shen, Ding Ren ^a   Fang, Qiong ^a   De Fex, Henry F ^a   Schieven, Gary L ^a   Kanner, Steven B ^a   Barrish, Joel C ^a  

^a BRISTOL MYERS SQUIBB   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINO 5 CARBOXAMIDOTHIAZOLE; IMIDAZOQUINOLINE DERIVATIVE; PROTEIN P56; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG ACTIVITY; DRUG CONFORMATION; DRUG IDENTIFICATION; DRUG SCREENING; DRUG SYNTHESIS; HUMAN; NONHUMAN; SAPONIFICATION; SEQUENCE HOMOLOGY; STRUCTURE ACTIVITY RELATION;

EID: 10744220619     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.08.054     Document Type: Article

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