Discovery and SAR of novel, potent and selective protein tyrosine phosphatase 1B inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 19, 2003, Pages 3129-3132

  Pei, Zhonghua ^a   Li, Xiaofeng ^a   Liu, Gang ^a   Abad Zapatero, Cele ^a   Lubben, Tom ^a   Zhang, Tianyuan ^a   Ballaron, Stephen J ^a   Hutchins, Charles W ^a   Trevillyan, James M ^a   Jirousek, Michael R ^a,b  

^a ABBOTT LABORATORIES   (United States)

^b PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

PROTEIN TYROSINE PHOSPHATASE 1B INHIBITOR; PROTEIN TYROSINE PHOSPHATASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME INHIBITION; STRUCTURE ACTIVITY RELATION; T LYMPHOCYTE;

EID: 10744220562     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00725-X     Document Type: Article

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