Selective interactions of perylene derivatives having different side chains with inter- and intramolecular G-quadruplex DNA structures. A correlation with telomerase inhibition

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 2, 2005, Pages 413-420

  Rossetti, Luigi ^a   Franceschin, Marco ^a   Schirripa, Stefano ^a   Bianco, Armandodoriano ^a   Ortaggi, Giancarlo ^a   Savino, Maria ^a  

^a SAPIENZA UNIVERSITY OF ROME   (Italy)

Author keywords

G Quadruplex; Perylene diimides; Telomerase inhibitors

Indexed keywords

N,N' BIS[2 (1 PIPERAZINO)ETHYL] 3,4,9,10 PERYLENETETRACARBOXYLIC DIIMIDE; N,N' BIS[2 (1 PIPERIDINO)ETHYL] 3,4,9,10 PERYLENETETRACARBOXYLIC DIIMIDE; N,N' BIS[2 (2 PYRIDINO)ETHYL] 3,4,9,10 PERYLENETETRACARBOXYLIC DIIMIDE; N,N' BIS[2 (4 MORPHOLINO)ETHYL] 3,4,9,10 PERYLENETETRACARBOXYLIC DIIMIDE; N,N' BIS[2 [2 (1 METHYL)PYRIDINO]ETHYL] 3,4,9,10 PERYLENETETRACARBOXYLIC DIIMIDE; N,N' BIS[2 [2 (1 METHYL)PYRROLIDINO]ETHYL] 3,4,9,10 PERYLENETETRACARBOXYLIC DIIMIDE; N,N' BIS[3 (4 MORPHOLINO)PROPYL] 3,4,9,10 PERYLENETETRACARBOXYLIC DIIMIDE; PERYLENE; TELOMERASE; UNCLASSIFIED DRUG;

ARTICLE; CORRELATION ANALYSIS; DNA STRUCTURE; DRUG EFFICACY; ELECTRICITY; ENZYME INHIBITION; MOLECULAR INTERACTION;

BASE SEQUENCE; DNA; DRUG INTERACTIONS; ENZYME INHIBITORS; HUMANS; PERYLENE; TELOMERASE;

EID: 10644290098     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.10.061     Document Type: Article

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