Characterization of Ro 04-6790 and Ro 63-0563: Potent and selective antagonists at human and rat 5-HT6 receptors

British Journal of Pharmacology

Volumn 124, Issue 3, 1998, Pages 556-562

  Sleight, Andrew J ^a   Boess, Frank G ^a   Bös, Michael ^a   Levet Trafit, Bernard ^a   Riemer, Claus ^a   Bourson, Anne ^a  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

Author keywords

5 HT6 receptor; 5 HT6 receptor antagonists; Ro 04 6790; Ro 63 0563; Stretching

Indexed keywords

4 AMINO N (2,6 BISMETHYLAMINOPYRIDIN 4 YL)BENZENE SULFONAMIDE; 4 AMINO N (2,6 BISMETHYLAMINOPYRIMIDIN 4 YL)BENZENE SULFONAMIDE; ANTISENSE OLIGONUCLEOTIDE; CYCLIC AMP; RECOMBINANT RECEPTOR; SEROTONIN 6 RECEPTOR; SEROTONIN ANTAGONIST; SEROTONIN RECEPTOR; SULFONAMIDE; UNCLASSIFIED DRUG;

ANIMAL BEHAVIOR; ANIMAL EXPERIMENT; ARTICLE; BINDING SITE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; HELA CELL; HUMAN; HUMAN CELL; INTRAPERITONEAL DRUG ADMINISTRATION; INTRAVENOUS DRUG ADMINISTRATION; MALE; MASTICATION; NONHUMAN; PRIORITY JOURNAL; RAT; STRETCHING; YAWNING;

EID: 0031748656     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701851     Document Type: Article

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