2-Alkylthio-substituted platelet P2Y12 receptor antagonists reveal pharmacological identity between the rat brain Gi-linked ADP receptors and P2Y12

Neuropharmacology

Volumn 45, Issue 1, 2003, Pages 145-154

  Vasiljev, Kati S ^a   Uri, Asko ^b   Laitinen, Jarmo T ^a  

^a UNIVERSITY OF EASTERN FINLAND   (Finland)

^b UNIVERSITY OF TARTU   (Estonia)

Author keywords

AR C compounds; Gi linked P2Y receptors; Platelet P2Y12 receptor antagonists; Presynaptic P2Y receptors; White matter tracts; 35S GTP S autoradiography

Indexed keywords

ADENOSINE ASPARTATE CONJUGATE; ADENOSINE DIPHOSPHATE; ADENOSINE TRIPHOSPHATE DERIVATIVE; ADENYLATE CYCLASE; AR C69581; AR C69931; AR C70300; AR C78511; BETA,GAMMA DICHLOROMETHYLENE 2 PROPYLTHIOADENOSINE TRIPHOSPHATE; G PROTEIN COUPLED RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); PURINE P2Y RECEPTOR; PURINERGIC RECEPTOR BLOCKING AGENT; SULFUR 35; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BINDING AFFINITY; BRAIN REGION; BRAIN TISSUE; CONTROLLED STUDY; DATA ANALYSIS; DRUG CONJUGATION; DRUG POTENCY; ENZYME INHIBITION; GLIOMA CELL; HUMAN; HUMAN CELL; IC 50; MALE; NONHUMAN; PRIORITY JOURNAL; PROTEIN FUNCTION; PROTEIN LOCALIZATION; RAT; RECEPTOR AFFINITY; STIMULATION; THROMBOCYTE; THROMBOCYTE MEMBRANE; WHITE MATTER;

EID: 0038177945     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(03)00142-4     Document Type: Article

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