Activation of vanilloid receptor 1 by resiniferatoxin mobilizes calcium from inositol 1,4,5-trisphosphate-sensitive stores

British Journal of Pharmacology

Volumn 138, Issue 1, 2003, Pages 172-176

  Marshall, Ian C B ^a   Owen, Davina E ^a   Cripps, Tim V ^a   Davis, John B ^a   McNulty, Shaun ^a   Smart, Darren ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

Capsaicin; Confocal microscopy; Fluorometric imaging plate reader; Inositol 1,4,5 trisphosphate; Phospholipase C; Resiniferatoxin; Vanilloid receptor 1

Indexed keywords

1 [[6 (3 METHOXYESTRA 1,3,5(10) TRIEN 17BETA YL)AMINO]HEXYL] 1H PYRROLE 2,5 DIONE; 1 [[6 (3 METHOXYESTRA 1,3,5(10) TRIEN 17BETA YL)AMINO]HEXYL] 2,5 PYRROLIDINEDIONE; ADENOSINE TRIPHOSPHATASE (CALCIUM); ADENOSINE TRIPHOSPHATASE INHIBITOR; CALCIUM; CALCIUM CHANNEL; CAPSAICIN; CAPSAZEPINE; CARBACHOL; CHOLINERGIC RECEPTOR STIMULATING AGENT; FLUORESCENT DYE; INOSITOL 1,4,5 TRISPHOSPHATE; PHOSPHOLIPASE C INHIBITOR; RECEPTOR BLOCKING AGENT; RESINIFERATOXIN; RUTHENIUM RED; THAPSIGARGIN; VANILLOID RECEPTOR;

ARTICLE; CALCIUM CELL LEVEL; CALCIUM MOBILIZATION; CALCIUM TRANSPORT; CHANNEL GATING; CONFOCAL MICROSCOPY; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG MECHANISM; EMBRYO; FLUOROMETRY; HUMAN; HUMAN CELL; IC 50; LIGAND BINDING; PAIN; PRIORITY JOURNAL; SIGNAL TRANSDUCTION;

CALCIUM; CALCIUM SIGNALING; CELL LINE; DITERPENES; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; INOSITOL 1,4,5-TRISPHOSPHATE; RECEPTORS, DRUG; TRPV CATION CHANNELS;

EID: 0037272795     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0705003     Document Type: Article

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