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Volumn 417, Issue 1-2, 2001, Pages 51-58

Characterisation using FLIPR of human vanilloid VR1 receptor pharmacology

(9) Smart, Darren a Jerman, Jeffrey C a Gunthorpe, Martin J a Brough, Stephen J a Ranson, Jennie a Cairns, William a Hayes, Philip D a Randall, Andrew D a Davis, John B a

a GLAXOSMITHKLINE (United Kingdom)

Author keywords

Ca2+; Capsaicin; FLIPR; Ligand gated ion channel; Nociception; Vanilloid

Indexed keywords

ANANDAMIDE; CALCIUM CHANNEL; CALCIUM ION; CAPSAICIN; CAPSAZEPINE; ION CHANNEL; ISOVELLERAL; OLVANIL; RESINIFERATOXIN; RUTHENIUM; UNCLASSIFIED DRUG; VANILLOID RECEPTOR; VANILLOID RECEPTOR 1;

ARTICLE; CONTROLLED STUDY; DRUG POTENCY; HUMAN; HUMAN CELL; KIDNEY CELL; MEMBRANE PERMEABILITY; NOCICEPTION; NUCLEOTIDE SEQUENCE; PATCH CLAMP; PH; PRIORITY JOURNAL;

ALKALOIDS; ANILINE COMPOUNDS; ARACHIDONIC ACIDS; BENZOPHENANTHRIDINES; CALCIUM; CAPSAICIN; CELL LINE; DITERPENES; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME INHIBITORS; FLUORESCENCE; FLUOROMETRY; HUMANS; HYDROGEN-ION CONCENTRATION; MEMBRANE POTENTIALS; PHENANTHRIDINES; POLYUNSATURATED ALKAMIDES; PROTEIN KINASE C; RECEPTORS, DRUG; RUTHENIUM RED; SESQUITERPENES; TIME FACTORS; XANTHENES;

EID: 0035815294 PISSN: 00142999 EISSN: None Source Type: Journal
DOI: 10.1016/S0014-2999(01)00901-3 Document Type: Article

Times cited : (91)

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