Novel peptide inhibitors of Leishmania gp63 based on the cleavage site of MARCKS (myristoylated alanine-rich C kinase substrate)-related protein

Biochemical Journal

Volumn 367, Issue 3, 2002, Pages 761-769

  Corradin, Sally ^a   Ransijn, Adriana ^a   Corradin, Giampietro ^a   Bouvier, Jacques ^a   Delgado, Maria Belen ^a   Fernandez Carneado, Jimena ^a   Mottram, Jeremy C ^a   Vergères, Guy ^a   Mauël, Jacques ^a  

^a UNIVERSITY OF LAUSANNE   (Switzerland)

Author keywords

Metalloprotease; Tat; Transduction

Indexed keywords

AMINO ACIDS; CELLS; ENZYMES; HYDROLYSIS; PHYSIOLOGY;

PHOSPHORYLATION;

BIOCHEMISTRY;

1,10 PHENANTHROLINE; ANTIPROTOZOAL AGENT; ASPARTIC ACID; BENZYLOXYCARBONYLTYROSYLLEUCYLHYDROXAMATE; CARBONIC ACID DERIVATIVE; MARCKS PROTEIN; MARCKS RELATED PROTEIN; MEMBRANE PROTEIN; METALLOPROTEINASE; PROTEIN GP63; PROTEIN KINASE C; PROTOZOAL PROTEIN; SERINE; TRANSACTIVATOR PROTEIN; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ANTIPROTOZOAL ACTIVITY; ARTICLE; CHEMICAL MODIFICATION; CONTROLLED STUDY; ENZYME SUBSTRATE; INHIBITION KINETICS; LEISHMANIA; MACROPHAGE; NONHUMAN; PRIORITY JOURNAL; PROMASTIGOTE; PROTEIN DEGRADATION; PROTEIN DOMAIN; PROTEIN PHOSPHORYLATION; PROTEIN SYNTHESIS; SIGNAL TRANSDUCTION; STRUCTURE ACTIVITY RELATION;

AMINO ACID SEQUENCE; ANIMALS; CIRCULAR DICHROISM; HYDROLYSIS; LEISHMANIA MAJOR; MEMBRANE PROTEINS; METALLOENDOPEPTIDASES; MICROSCOPY, FLUORESCENCE; MOLECULAR SEQUENCE DATA; PEPTIDES; PROTEASE INHIBITORS; RECOMBINANT PROTEINS; SUBSTRATE SPECIFICITY;

HUMAN IMMUNODEFICIENCY VIRUS 1; PROTOZOA;

EID: 0036847052     PISSN: 02646021     EISSN: None     Source Type: Journal    
DOI: 10.1042/BJ20020386     Document Type: Article

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