Accelerating drug discovery by integrative implementation of laboratory automation in the work flow

Current Medicinal Chemistry

Volumn 9, Issue 23, 2002, Pages 2179-2190

  Nettekoven, Matthias ^a   Thomas, Andrew W ^a  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

Author keywords

Case studies; Combinatorial chemistry; Drug discovery; Integrative workflow concept; Laboratory automation; Parallel synthesis

Indexed keywords

4 (4 FLUOROPHENYL) 2 (4 METHYLSULFINYLPHENYL) 5 (4 PYRIDYL)IMIDAZOLE; 4 (4 FLUOROPHENYL) 2 (5 METHYL 5 MORPHOLINOCARBONYL 1,3 DIOXAN 2 YL) 5 (4 PYRIDINYL)IMIDAZOLE; ADENOSINE A2A RECEPTOR ANTAGONIST; ANTIRHEUMATIC AGENT; PYRIDINE DERIVATIVE; RPR 132331; RPR 201227A; RPR 203494; RPR 238677; TRIAZOLOPYRIDINE DERIVATIVE; TUMOR NECROSIS FACTOR ALPHA; UNCLASSIFIED DRUG;

ANALYTICAL EQUIPMENT; ARTICLE; COMBINATORIAL CHEMISTRY; CONTROLLED STUDY; DATA ANALYSIS; DRUG DEVELOPMENT; DRUG RESEARCH; DRUG SYNTHESIS; HUMAN; JOB PERFORMANCE; LABORATORY AUTOMATION; ORGANIC CHEMISTRY; ROBOTICS; TECHNOLOGY; APPARATUS, EQUIPMENT AND SUPPLIES; AUTOMATION; CHEMISTRY; DRUG DESIGN; DRUG SCREENING; INSTRUMENTATION; METHODOLOGY; REVIEW;

AUTOMATION; CHEMISTRY, PHARMACEUTICAL; COMBINATORIAL CHEMISTRY TECHNIQUES; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; EQUIPMENT AND SUPPLIES;

EID: 0036427644     PISSN: 09298673     EISSN: None     Source Type: Journal    
DOI: 10.2174/0929867023368764     Document Type: Article

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