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Volumn 965, Issue , 2002, Pages 92-108

Preclinical evaluation of GBR12909 decanoate as a long-acting medication for methamphetamine dependence

Author keywords

Cocaine; DA transporter; Drug addiction; GBR decanoate; GBR12909; Methamphetamine; Pharmacotherapies; Psychomotor stimulants

Indexed keywords

DOPAMINE 2 RECEPTOR STIMULATING AGENT; DOPAMINE 3 RECEPTOR STIMULATING AGENT; DOPAMINE TRANSPORTER; METHAMPHETAMINE; PROLACTIN; QUINPIROLE; VANOXERINE;

EID: 0036296960     PISSN: 00778923     EISSN: None     Source Type: Book Series    
DOI: 10.1111/j.1749-6632.2002.tb04154.x     Document Type: Conference Paper
Times cited : (17)

References (70)
  • 1
    • 0029582665 scopus 로고
    • Increasing morbidity and mortality associated with abuse of methamphetamine - United States, 1991-1994
    • (1995) MMWR Morb. Mort. Wkly. Rep. , vol.44 , pp. 882-886
  • 3
    • 0009590419 scopus 로고    scopus 로고
  • 5
    • 0009640177 scopus 로고    scopus 로고
  • 12
    • 0033984392 scopus 로고    scopus 로고
    • Neurochemical neutralization of methamphetamine with high-affinity nonselective inhibitors of biogenic amine transporters: A pharmacological strategy for treating stimulant abuse
    • (2000) Synapse , vol.35 , pp. 222-227
    • Rothman, R.B.1
  • 13
    • 25744449012 scopus 로고
    • High affinity dopamine uptake inhibitors as potential cocaine antagonists
    • (1990) Life. Sci. , vol.46
    • Rothman, R.B.1
  • 15
    • 0029348098 scopus 로고
    • A review of the effects of dopaminergic agents on humans, animals, and drug seeking behavior, and its implications for medication development: Focus on GBR12909
    • (1995) Mol. Neurobiol. , vol.11 , pp. 1-19
    • Rothman, R.B.1    Glowa, J.R.2
  • 17
    • 0027174387 scopus 로고
    • Identification of a GBR12935 homolog, LR111, which is over 4000-fold selective for the dopamine transporter, relative to serotonin and norepinephrine transporters
    • (1993) Synapse , vol.14 , pp. 34-39
    • Rothman, R.B.1
  • 20
    • 0029072718 scopus 로고
    • Photoaffinity-labeled ligand binding domains on dopamine transporters identified by peptide mapping
    • (1995) Mol. Pharmacol. , vol.47 , pp. 956-964
    • Vaughan, R.A.1
  • 25
    • 0029120376 scopus 로고
    • Effects of dopamine reuptake inhibitors on food and cocaine maintained responding. II: Comparisons with other drugs and repeated administrations
    • (1995) Exp. Clin. Psychopharmacol. , vol.3
    • Glowa, J.R.1
  • 26
    • 0029909269 scopus 로고    scopus 로고
    • Differential reinforcing effects of cocaine and GBR-12909: Biochemical evidence for divergent neuroadaptive changes in the mesolimbic dopaminergic system
    • (1996) J. Neurosci. , vol.16 , pp. 7416-7427
    • Tella, S.R.1
  • 30
    • 0030473214 scopus 로고    scopus 로고
    • Sustained decrease in cocaine-maintained responding in rhesus monkeys with 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-hydroxy-3-phenylpropyl) piperazinyl decanoate, a long-acting ester derivative of GBR 12909
    • (1996) J. Med. Chem. , vol.39 , pp. 4689-4691
    • Glowa, J.R.1
  • 31
    • 0033518262 scopus 로고    scopus 로고
    • Oxygenated analogs of 1-[2-(diphenylmethoxy)ethyl]- and 1-[2-[bis-(4-fluorophenyl)methoxy]ethyl] 4-(3-phenylpropyl)piperazines (GBR12935 and GBR12909) as potential extended-action cocaine-abuse therapeutic agents
    • (1999) J. Med. Chem. , vol.42 , pp. 5029-5042
    • Lewis, D.B.1
  • 32
    • 0017111032 scopus 로고
    • 14c-fluphenazine enanthate and decanoate esters administered in sesame oil to dogs
    • (1976) J. Pharm. Sci. , vol.65 , pp. 502-507
    • Dreyfuss, J.1
  • 34
    • 6844236997 scopus 로고    scopus 로고
    • 125I]RTI-55 in membranes prepared from human, monkey and guinea pig caudate
    • (1998) Synapse , vol.28 , pp. 322-338
    • Rothman, R.B.1
  • 35
    • 0028153669 scopus 로고
    • 125I]RTI-55: In vitro binding and autoradiographic characterization
    • (1994) J. Neurochem. , vol.62 , pp. 549-556
    • Staley, J.K.1
  • 36
    • 0034113934 scopus 로고    scopus 로고
    • Effects of phentermine and fenfluramine on extracellular dopamine and serotonin in rat nucleus accumbens: Therapeutic implications
    • (2000) Synapse , vol.36 , pp. 102-113
    • Baumann, M.H.1
  • 37
    • 0028069868 scopus 로고
    • Behavioral and neurochemical data suggest functional differences between dopamine D2 and D3 receptors
    • (1994) Eur. J. Pharmacol. , vol.263 , pp. 235-243
    • Svensson, K.1
  • 39
    • 0034628982 scopus 로고    scopus 로고
    • Differential neuroendocrine responsiveness to morphine in Lewis, Fischer 344, and ACI inbred rats
    • (2000) Brain Res. , vol.858 , pp. 320-326
    • Baumann, M.H.1
  • 45
    • 15844384993 scopus 로고    scopus 로고
    • Striatal dopamine nerve terminal markers in human chronic methamphetamine users
    • (1996) Nat. Med. , vol.2 , pp. 699-703
    • Wilson, J.M.1
  • 46
    • 17344365599 scopus 로고    scopus 로고
    • 11C]WIN-35,428 positron emission tomograpgy studies and direct in vitro determinations
    • (1998) J. Neurosci. , vol.18 , pp. 419-427
    • Villemagne, V.L.1
  • 47
    • 0025853962 scopus 로고
    • Cocaine addiction: Psychology and neurophysiology
    • (1991) Science , vol.253 , pp. 1580-1586
    • Gawin, F.1
  • 50
    • 0028914666 scopus 로고
    • Biogenic amine flux mediated by cloned transporters stably expressed in cultured cell lines: Amphetamine specificity for inhibition and efflux
    • (1995) Mol. Pharmacol. , vol.47 , pp. 544-550
    • Wall, S.C.1    Gu, H.2    Rudnick, G.3
  • 51
    • 0028944943 scopus 로고
    • Hippocampus norepinephrine, caudate dopamine and serotonin, and behavioral responses to stereoisomers of amphetamine and methamphetamine
    • (1995) J. Neurosci. , vol.15 , pp. 1308-1317
    • Kuczenski, R.1
  • 52
    • 0029010295 scopus 로고
    • Pharmacokinetic and pharmacodynamic analysis of the action of amphetamine and D-methamphetamine on dopamine terminals
    • (1995) J. Pharmacol. Exp. Ther. , vol.274 , pp. 90-96
    • Melega, W.P.1
  • 53
    • 0033695201 scopus 로고    scopus 로고
    • Methamphetamine dependence: Medication development efforts based on a dual deficit model of stimulant addiction
    • (2000) Ann. N.Y. Acad. Sci. , vol.914 , pp. 71-81
    • Rothman, R.B.1
  • 54
    • 0002121961 scopus 로고    scopus 로고
    • Effects of GBR12909 on responding maintained under a progressive-ratio schedule of methamphetamine delivery in rhesus monkeys
    • (2001) Drug Alcohol Depend. , vol.63
    • Glowa, J.R.1
  • 63
    • 0021253334 scopus 로고
    • Electrophysiological evidence for A10 dopamine autoreceptor subsensitivity following chronic D-amphetamine treatment
    • (1984) Brain Res. , vol.309 , pp. 283-292
    • White, F.J.1    Wang, R.Y.2
  • 66
    • 0026800560 scopus 로고
    • Do autoreceptors mediate dopamine agonist-induced yawning and suppression of exploration? A critical review
    • (1992) Psychopharmacology , vol.106 , pp. 1-14
    • Stahle, L.1
  • 70


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